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51

Molecular features of the prazosin molecule required for activation of Transport-P

Joaquim Fernando Mendes da Silva, Marcus Walters, Saad Al-Damluji, C. Robin Ganellin

Journal:

Bioorganic & Medicinal Chemistry

Year:

2008

Language:

english

File:

PDF, 254 KB

english, 2008

52

Defining determinant molecular properties for the blockade of the apamin-sensitive SKCa channel in guinea-pig hepatocytes: the influence of polarizability and molecular geometry

Dimitrios Galanakis, C.Robin Ganellin

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2004

Language:

english

File:

PDF, 274 KB

english, 2004

53

Bis-quinolinium cyclophanes: toward a pharmacophore model for the blockade of apamin-sensitive SKCa channels in sympathetic neurons

Dimitrios Galanakis, C.Robin Ganellin, Jian-Quing Chen, Diyan Gunasekera, Philip M Dunn

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2004

Language:

english

File:

PDF, 275 KB

english, 2004

54

Potential HIV protease inhibitors: Preparation of di-N-alkylated 2-, 6-, and 2,6-aminodeoxy-derivatives of d-glucose by direct displacement and by a novel reductive-alkylation procedure

Jiaqiang Cai, Bruce E. Davison, C.Robin Ganellin, Suvit Thaisrivongs, Keith S. Wibley

Journal:

Carbohydrate Research

Year:

1997

Language:

english

File:

PDF, 852 KB

english, 1997

55

Calculation of conformational free energy of histamine

L. Farnell, W.G. Richards, C.R. Ganellin

Journal:

Journal of Theoretical Biology

Year:

1974

Language:

english

File:

PDF, 185 KB

english, 1974

56

The dielectric properties of seven polar amidine-containing compounds of biological interest

Rodney C. Young, C.Robin Ganellin, Michael J. Graham, Michael L. Roantree, Edward H. Grant

Journal:

Tetrahedron Letters

Year:

1985

Language:

english

File:

PDF, 198 KB

english, 1985

57

University education of medicinal chemists: comparison of eight countries

C.Robin Ganellin, Lester A Mitscher, Bernd Clement, Toshi-Hiko Kobayashi, Emilio Kyburz, Olivier Lafont, Annie Marcincal, Antonio Monge, Giorgio Tarzia, John G Topliss

Journal:

European Journal of Medicinal Chemistry

Year:

2000

Language:

english

File:

PDF, 62 KB

english, 2000

58

Analogues and derivatives of ciproxifan, a novel prototype for generating potent histamine H3-receptor antagonists

Holger Stark, Xavier Ligneau, Bassem Sadek, C.Robin Ganellin, Jean-Michel Arrang, Jean-Charles Schwartz, Walter Schunack

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2000

Language:

english

File:

PDF, 153 KB

english, 2000

59

Imetit and N-methyl derivatives. The transition from potent agonist to antagonist at histamine H3 receptors.1

C.R. Ganellin, B. Bang-Andersen, Y.S. Khalaf, W. Tertiuk, J.M. Arrang, M. Garbarg, X. Ligneau, A. Rouleau, J.C. Schwartz

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1992

Language:

english

File:

PDF, 316 KB

english, 1992

60

Different antagonist binding properties of human and rat histamine H3 receptors

Holger Stark, Wolfgang Sippl, Xavier Ligneau, Jean-Michel Arrang, C.Robin Ganellin, Jean-Charles Schwartz, Walter Schunack

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 720 KB

english, 2001

61

Bis-quinolinium cyclophanes: A novel class of potent blockers of the apamin-sensitive Ca2+-activated K+ channel

Joaquin Campos Rosa, Bridgitte M Beckwith-Hall, Dimitrios Galanakis, C.Robin Ganellin, Philip M Dunn, Donald H Jenkinson

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1997

Language:

english

File:

PDF, 239 KB

english, 1997

62

(Partial) agonist/antagonist properties of novel diarylalkyl carbamates on histamine H3 receptors

Astrid Sasse, Holger Stark, Xavier Ligneau, Sigurd Elz, Sibylle Reidemeister, C.Robin Ganellin, Jean-Charles Schwartz, Walter Schunack

Journal:

Bioorganic & Medicinal Chemistry

Year:

2000

Language:

english

File:

PDF, 242 KB

english, 2000

63

Piperidino-Hydrocarbon compounds as novel non-Imidazole histamine H3-Receptor antagonists

Galina Meier, Xavier Ligneau, Heinz H Pertz, C.Robin Ganellin, Jean-Charles Schwartz, Walter Schunack, Holger Stark

Journal:

Bioorganic & Medicinal Chemistry

Year:

2002

Language:

english

File:

PDF, 166 KB

english, 2002

64

Imidazole derivatives as a novel class of hybrid compounds with inhibitory histamine N-methyltransferase potencies and histamine hH3 receptor affinities

Sven Graßmann, Joachim Apelt, Wolfgang Sippl, Xavier Ligneau, Heinz H Pertz, Yuan Hui Zhao, Jean-Michel Arrang, C.Robin Ganellin, Jean-Charles Schwartz, Walter Schunack, Holger Stark

Journal:

Bioorganic & Medicinal Chemistry

Year:

2003

Language:

english

File:

PDF, 406 KB

english, 2003

65

Dimaprit, [S-[3-(N,N-dimethylamino)propyl]isothiourea]. A highly specific histamine H2-receptor agonist. Part 2. Structure-activity considerations

G. J. Durant, C. R. Ganellin, M. E. Parsons

Journal:

Inflammation Research

Year:

1977

Language:

english

File:

PDF, 319 KB

english, 1977

66

The pressor activity of burimamide: A relationship between chemical constitution and pressor activity of burimamide and related histamine H2-receptor antagonists

C. R. Ganellin, D. A. A. Owen

Journal:

Inflammation Research

Year:

1977

Language:

english

File:

PDF, 275 KB

english, 1977

67

Dimaprit-[S-[3-(N,N-dimethylamino)propyl]isothiourea] —A highly specific histamine H2-receptor agonist. Part 1. Pharmacology

M. E. Parsons, D. A. A. Owen, C. R. Ganellin, G. J. durant

Journal:

Inflammation Research

Year:

1977

Language:

english

File:

PDF, 551 KB

english, 1977

68

Histamine-induced inhibition of lymphocyte proliferation and lysosomal enzyme release from polymorphs may not be mediated via H1- or H2-receptors

M. R. Vickers, K. Milliner, D. Martin, C. R. Ganellin

Journal:

Inflammation Research

Year:

1982

Language:

english

File:

PDF, 401 KB

english, 1982

69

Metiamide — An orally active histamine H2-receptor antagonist

J. W. Black, W. A. M. Duncan, J. C. Emmett, C. R. Ganellin, T. Hesselbo, M. E. Parsons, J. H. Wyllie

Journal:

Inflammation Research

Year:

1973

Language:

english

File:

PDF, 413 KB

english, 1973

70

Binding of [3H]cimetidine to rat brain tissue

Ian R. Smith, Mark T. Cleverley, C. Robin Ganellin, Kathleen M. Metters

Journal:

Inflammation Research

Year:

1980

Language:

english

File:

PDF, 410 KB

english, 1980

71

3-[4(5)-Imidazolyl] propylguanidine (SK&F 91486) — a partial agonist at histamine H2-receptors

M. E. Parsons, R. C. Blakemore, G. J. Durant, C. R. Ganellin, A. C. Rasmussen

Journal:

Inflammation Research

Year:

1975

Language:

english

File:

PDF, 82 KB

english, 1975

72

N-Methyldimaprit (SK&F92054). A chemical control for the histamine H2-receptor agonist dimaprit

R. C. Blakemore, C. R. Ganellin, B. K. Leigh, M. E. Parsons, C. A. Price, I. R. Smith, W. Tertiuk

Journal:

Inflammation Research

Year:

1986

Language:

english

File:

PDF, 557 KB

english, 1986

73

Dimaprit, [S-[3-(N,N-dimethylamino)propyl]isothiourea]. A highly specific histamine H2-receptor agonist. Part 2. Structure-activity considerations

G. J. Durant, C. R. Ganellin, M. E. Parsons

Journal:

Inflammation Research

Year:

1994

Language:

english

File:

PDF, 383 KB

english, 1994

74

Dimaprit—[S-[3-(N,N-dimethylamino)propyl]isothiourea]—A highly specific histamine H2-receptor agonist. Part 1, pharmacology

M. E. Parsons, D. A. A. Owen, C. R. Ganellin, G. J. Durant

Journal:

Inflammation Research

Year:

1994

Language:

english

File:

PDF, 624 KB

english, 1994

75

Metiamide—An orally active histamine H2-receptor antagonist

J. W. Black, W. A. M. Duncan, J. C. Emmett, C. R. Ganellin, T. Hesselbo, M. E. Parsons, J. H. Wyllie

Journal:

Inflammation Research

Year:

1994

Language:

english

File:

PDF, 505 KB

english, 1994

76

Tautomerism of 4-methylhistamine—Effect of the methyl substituent

J. C. Emmett, C. R. Ganellin, M. J. Graham, F. H. Holloway

Journal:

Inflammation Research

Year:

1979

Language:

english

File:

PDF, 156 KB

english, 1979

77

Personal reflections on Sir James Black (1924–2010) and histamine

C. Robin Ganellin

Journal:

Inflammation Research

Year:

2011

Language:

english

File:

PDF, 767 KB

english, 2011

78

Histamine H1-Receptor in Heart: Unique Electrophoretic Mobility and Autoradiographic Localization

M. Ruat, M. L. Bouthenet, J.-C. Schwartz, C. R. Ganellin

Journal:

Journal of Neurochemistry

Year:

1990

Language:

english

File:

PDF, 1.65 MB

english, 1990

79

Design of an Affinity Matrix for Purification of the Histamine H1 Receptor from Guinea Pig Cerebellum

M. Ruat, E. Traiffort, M. Garbarg, J. C. Schwartz, P. Demonchaux, R. J. Ife, W. Tertiuk, C. R. Ganellin

Journal:

Journal of Neurochemistry

Year:

1992

Language:

english

File:

PDF, 703 KB

english, 1992

80

The pharmacology of cimetidine, a new histamine H2-receptor antagonist

RW Brimblecombe, WAM Duncan, GJ Durant, CR Ganellin, ME Parsons, JW Black

Journal:

British Journal of Pharmacology

Year:

2010

Language:

english

File:

PDF, 185 KB

english, 2010

81

Definition and Antagonism of Histamine H2-receptors

BLACK, J. W., DUNCAN, W. A. M., DURANT, C. J., GANELLIN, C. R., PARSONS, E. M.

Journal:

Year:

1972

File:

PDF, 692 KB

1972

82

Sulphur-methylene isosterism in the developent of metiamide, a new histamine H2-receptor antagonist

BLACK, J. W., DURANT, G. J., EMMETT, J. C., GANELLIN, C. R.

Journal:

Year:

1974

File:

PDF, 356 KB

1974

83

Impromidine (SK&F 92676) is a very potent and specific agonist for histamine H2 receptors

DURANT, G. J., DUNCAN, W. A. M., GANELLIN, C. R., PARSONS, M. E., BLAKEMORE, R. C., RASMUSSEN, A. C.

Journal:

Year:

1978

File:

PDF, 399 KB

1978

84

10.1038/35048583

Arrang, Jean-Michel, Morisset, Séverine, Rouleau, Agnès, Ligneau, Xavier, Gbahou, Florence, Tardivel-Lacombe, Joël, Stark, Holger, Schunack, Walter, Ganellin, C. Robin

Journal:

Year:

2000

Language:

english

File:

PDF, 438 KB

english, 2000

85

Characterization and inhibition of a cholecystokinin-inactivating serine peptidase

Rose, Christiane, Vargas, Froylan, Facchinetti, Patricia, Bourgeat, Pierre, Bambal, Ramesh B., Bishop, Paul B., Chan, Suzanne M. T., Moore, Andrew N. J., Ganellin, C. Robin, Schwartz, Jean-Charles

Journal:

Year:

1996

File:

PDF, 1.89 MB

1996

86

Obituary: James Black (1924–2010)

Ganellin, Robin, Duncan, William

Journal:

Year:

2010

Language:

english

File:

PDF, 151 KB

english, 2010

87

Differences in the actions of some blockers of the calcium-activated potassium permeability in mammalian red cells

D C H Benton, C J Roxburgh, C R Ganellin, M A R Shiner, D H Jenkinson

Journal:

British Journal of Pharmacology

Year:

1999

Language:

english

File:

PDF, 387 KB

english, 1999

88

Compounds that block both intermediate-conductance (IKCa) and small-conductance (SKCa) calcium-activated potassium channels

M Malik-Hall, C R Ganellin, D Galanakis, D H Jenkinson

Journal:

British Journal of Pharmacology

Year:

2000

Language:

english

File:

PDF, 202 KB

english, 2000

89

Distinct pharmacology of rat and human histamine H3 receptors: role of two amino acids in the third transmembrane domain

X Ligneau, S Morisset, J Tardivel-Lacombe, F Gbahou, C R Ganellin, H Stark, W Schunack, J -C Schwartz, J -M Arrang

Journal:

British Journal of Pharmacology

Year:

2000

Language:

english

File:

PDF, 135 KB

english, 2000

90

Clotrimazole analogues: effective blockers of the slow afterhyperpolarization in cultured rat hippocampal pyramidal neurones

M M Shah, Z Miscony, M Javadzadeh-Tabatabaie, C R Ganellin, D G Haylett

Journal:

British Journal of Pharmacology

Year:

2001

Language:

english

File:

PDF, 214 KB

english, 2001

91

10.1021/jm00329a015

Ganellin, C. R., Spickett, R. G. W.

Journal:

Journal of Medicinal Chemistry

Year:

1965

Language:

english

File:

PDF, 893 KB

english, 1965

92

Compounds Affecting the Central Nervous System. IV. Substituted 2-Benzyl-3-dialkylaminoalkylindenes and Related Compounds

Ganellin, C. R., Loynes, J. M., Ridley, H. F., Spickett, R. G. W.

Journal:

Journal of Medicinal Chemistry

Year:

1967

Language:

english

File:

PDF, 934 KB

english, 1967

93

Compounds Affecting the Central Nervous System. V. Substituted 3-Dialkylaminoalkylindenes

Bavin, P. M. G., Ganellin, C, Loynes, J, Spickett, R G W

Journal:

Journal of Medicinal Chemistry

Year:

1969

Language:

english

File:

PDF, 483 KB

english, 1969

94

Synthesis and Structure-Activity Relationships of Dequalinium Analogs as K+ Channel Blockers. Investigations on the Role of the Charged Heterocycle

Jenkinson, Donald H., Galanakis, Dimitrios, Davis, Carole A., Herrero, Benedicto Del Rey, Ganellin, C. Robin, Dunn, Philip M.

Journal:

Journal of Medicinal Chemistry

Year:

1995

Language:

english

File:

PDF, 2.33 MB

english, 1995

95

ChemInform Abstract: Design of Potent Non-Thiourea H3-Receptor Histamine Antagonists.

C. R. GANELLIN, S. K. HOSSEINI, Y. S. KHALAF, W. TERTIUK, J.-M. ARRANG, M. GARBARG, X. LIGNEAU, J.-C. SCHWARTZ

Journal:

Year:

1995

File:

PDF, 33 KB

1995

96

ChemInform Abstract: New 3,4-O-Isopropylidene Derivatives of D- and L-Glucopyranosides.

J. CAI, B. E. DAVISON, C. R. GANELLIN, S. THAISRIVONGS

Journal:

Year:

1996

File:

PDF, 28 KB

1996

97

ChemInform Abstract: Synthesis and Authentication of Iodoazidophenpyramine, a Photoaffinity Reporter Ligand Previously Used for Histamine H1-Receptor Labelling.

G. SORBA, W. TERTIUK, C. R. GANELLIN

Journal:

Year:

1996

File:

PDF, 32 KB

1996

98

The synthesis of 1-substituted-2-(β-dimethylaminoethyl)benzimidazoles

C. R. Ganellin, H. F. Ridley, R. G. W. Spickett

Journal:

Journal of Heterocyclic Chemistry

Year:

1966

Language:

english

File:

PDF, 380 KB

english, 1966

99

Naming of substituted histamines

J. W. Black, C. R. Ganellin

Journal:

Cellular and Molecular Life Sciences

Year:

1974

Language:

english

File:

PDF, 608 KB

english, 1974

100

Inhibition of the antigen-induced activation of RBL-2H3 cells by cetiedil and some of its analogues

Jamshid Narenjkar, El-Sayed K. Assem, C.Robin Ganellin

Journal:

European Journal of Pharmacology

Year:

2004

Language:

english

File:

PDF, 529 KB

english, 2004