CHRISTIAN SERGHERAERT: search on Z-Library

The world's largest scientific articles store. 70,000,000+ articles for free.

Don't use scam websites

1

Screening of Plasmodium falciparum iron superoxide dismutase inhibitors and accuracy of the SOD-assays

Laurent Soulère, Patrick Delplace, Elisabeth Davioud-Charvet, Sandrine Py, Christian Sergheraert, Jacques Périé, Isabelle Ricard, Pascal Hoffmann, Daniel Dive

Journal:

Bioorganic & Medicinal Chemistry

Year:

2003

Language:

english

File:

PDF, 150 KB

english, 2003

2

Conversion of Sterically Hindered Diacylated 1,2-Phenylenediamines into 2-Substituted Benzimidazoles

Charton, Julie, Girault-Mizzi, Sophie, Sergheraert, Christian

Journal:

CHEMICAL & PHARMACEUTICAL BULLETIN

Year:

2005

Language:

english

File:

PDF, 237 KB

english, 2005

3

ChemInform Abstract: Automated Parallel Synthesis of a Tetrahydroisoquinolin-Based Library: Potential Prolyl Endopeptidase Inhibitors.

Sandrine Vendeville, Line Bourel, Elisabeth Davioud-Charvet, Philippe Grellier, Benoit Deprez, Christian Sergheraert

Journal:

Year:

1999

File:

PDF, 29 KB

1999

4

ChemInform Abstract: PyBroP: A Convenient Activator for the Synthesis of Formamidines.

Sandrine Delarue, Christian Sergheraert

Journal:

Year:

1999

File:

PDF, 25 KB

1999

5

ChemInform Abstract: Synthesis and in vitro and in vivo Antimalarial Activity of New 4-Anilinoquinolines.

Sandrine Delarue, Sophie Girault, Louis Maes, Marie-Ange Debreu-Fontaine, Mehdi Labaeid, Philippe Grellier, Christian Sergheraert

Journal:

Year:

2001

File:

PDF, 25 KB

2001

6

ChemInform Abstract: “One-Pot” Synthesis and Antimalarial Activity of Formamidine Derivatives of 4-Anilinoquinoline.

Sandrine Delarue, Sophie Girault, Fouad Dali Ali, Louis Maes, Philippe Grellier, Christian Sergheraert

Journal:

Year:

2002

File:

PDF, 29 KB

2002

7

ChemInform Abstract: Convenient Synthesis of Tetrahydroisoquinoline-hydantoins.

Julie Charton, Sandrine Delarue, Sandrine Vendeville, Marie-Ange Debreu-Fontaine, Sophie Girault-Mizzi, Christian Sergheraert

Journal:

Year:

2002

File:

PDF, 26 KB

2002

8

Antitrypanosomal Activities and Cytotoxicity of 5-Nitro-2-furancarbohydrazides.

Regis Millet, Louis Maes, Valerie Landry, Christian Sergheraert, Elisabeth Davioud-Charvet

Journal:

Year:

2003

File:

PDF, 74 KB

2003

9

Design, Synthesis and Antimalarial Activity of Novel, Quinoline-Based, Zinc Metallo-Aminopeptidase Inhibitors.

Marian Flipo, Isabelle Florent, Philippe Grellier, Christian Sergheraert, Rebecca Deprez-Poulain

Journal:

Year:

2003

File:

PDF, 69 KB

2003

10

Synthesis and Antimalarial Evaluation of New 1,4-Bis(3-aminopropyl)piperazine Derivatives.

Adina Ryckebusch, Rebecca Deprez-Poulain, Marie-Ange Debreu-Fontaine, Richard Vandaele, Elisabeth Mouray, Philippe Grellier, Christian Sergheraert

Journal:

Year:

2004

File:

PDF, 77 KB

2004

11

Optimized Synthesis of Tetrahydroisoquinoline-Hydantoins.

Julie Charton, Amaury Cazenave Gassiot, Patricia Melnyk, Sophie Girault-Mizzi, Christian Sergheraert

Journal:

Year:

2005

File:

PDF, 144 KB

2005

12

Synthesis and Antimalarial Evaluation of New N1-(7-Chloro-4-quinolyl)-1,4-bis(3-aminopropyl)piperazine Derivatives.

Adina Ryckebusch, Marie-Ange Debreu-Fontaine, Elisabeth Mouray, Philippe Grellier, Christian Sergheraert, Patricia Melnyk

Journal:

Year:

2005

File:

PDF, 13 KB

2005

13

Conversion of Sterically Hindered Diacylated 1,2-Phenylenediamines into 2-Substituted Benzimidazoles.

Julie Charton, Sophie Girault-Mizzi, Christian Sergheraert

Journal:

Year:

2005

Language:

english

File:

PDF, 32 KB

english, 2005

14

Synthesis of 5,5′-Dithiobis(2-nitrobenzamides)as Alternative Substrates for Trypanothione Reductase and Thioredoxin Reductase: A Microtiter Colorimetric Assay for Inhibitor Screening

Elisabeth Davioud-Charvet, Katja Becker, Valérie Landry, Stephan Gromer, Cédric Logé, Christian Sergheraert

Journal:

Analytical Biochemistry

Year:

1999

Language:

english

File:

PDF, 87 KB

english, 1999

15

Synthesis and biological evaluation of benzimidazole derivatives as potent AMP-activated protein kinase activators

Julie Charton, Sophie Girault-Mizzi, Marie-Ange Debreu-Fontaine, Fabienne Foufelle, Isabelle Hainault, Jean-Guy Bizot-Espiard, Daniel-Henri Caignard, Christian Sergheraert

Journal:

Bioorganic & Medicinal Chemistry

Year:

2006

Language:

english

File:

PDF, 436 KB

english, 2006

16

Synthesis and antimalarial evaluation of new N1-(7-chloro-4-quinolyl)-1,4-bis(3-aminopropyl)piperazine derivatives

Adina Ryckebusch, Marie-Ange Debreu-Fontaine, Elisabeth Mouray, Philippe Grellier, Christian Sergheraert, Patricia Melnyk

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2005

Language:

english

File:

PDF, 284 KB

english, 2005

17

2-Amino diphenylsulfides as inhibitors of trypanothione reductase: modification of the side chain

Stéphanie Baillet, Eric Buisine, Dragos Horvath, Louis Maes, Beatrice Bonnet, Christian Sergheraert

Journal:

Bioorganic & Medicinal Chemistry

Year:

1996

Language:

english

File:

PDF, 869 KB

english, 1996

18

Synthesis and antimalarial evaluation of new 1,4-bis(3-aminopropyl)piperazine derivatives

Adina Ryckebusch, Rébecca Deprez-Poulain, Marie-Ange Debreu-Fontaine, Richard Vandaele, Elisabeth Mouray, Philippe Grellier, Christian Sergheraert

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2003

Language:

english

File:

PDF, 184 KB

english, 2003

19

Synthesis and pharmacological evaluation of Tic-hydantoin derivatives as selective σ1 ligands. Part 2

Amaury Cazenave Gassiot, Julie Charton, Sophie Girault-Mizzi, Pauline Gilleron, Marie-Ange Debreu-Fontaine, Christian Sergheraert, Patricia Melnyk

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2005

Language:

english

File:

PDF, 151 KB

english, 2005

20

Synthesis and pharmacological evaluation of Tic-hydantoin derivatives as selective σ1 ligands. Part 1

Julie Charton, Amaury Cazenave Gassiot, Sophie Girault-Mizzi, Marie-Ange Debreu-Fontaine, Patricia Melnyk, Christian Sergheraert

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2005

Language:

english

File:

PDF, 140 KB

english, 2005

21

Design, synthesis and in vitro antimalarial activity of an acylhydrazone library

Patricia Melnyk, Virginie Leroux, Christian Sergheraert, Philippe Grellier

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2006

Language:

english

File:

PDF, 145 KB

english, 2006

22

Synthesis and antimalarial activity of new analogues of amodiaquine

Sandrine Delarue-Cochin, Emilia Paunescu, Louis Maes, Elisabeth Mouray, Christian Sergheraert, Philippe Grellier, Patricia Melnyk

Journal:

European Journal of Medicinal Chemistry

Year:

2008

Language:

english

File:

PDF, 334 KB

english, 2008

23

Synthesis and antimalarial activity of carbamate and amide derivatives of 4-anilinoquinoline

Sandrine Delarue-Cochin, Philippe Grellier, Louis Maes, Elisabeth Mouray, Christian Sergheraert, Patricia Melnyk

Journal:

European Journal of Medicinal Chemistry

Year:

2008

Language:

english

File:

PDF, 482 KB

english, 2008

24

Optimized synthesis of tetrahydroisoquinoline-hydantoins

Julie Charton, Amaury Cazenave Gassiot, Patricia Melnyk, Sophie Girault-Mizzi, Christian Sergheraert

Journal:

Tetrahedron Letters

Year:

2004

Language:

english

File:

PDF, 281 KB

english, 2004

25

Derives soufres du methylcymantrene

Christian Sergheraert, Pierre Marcincal, Etienne Cuingnet

Journal:

Journal of Organometallic Chemistry

Year:

1977

File:

PDF, 561 KB

1977

26

Sulfonation du methyl cymantrene, analogues cymantreniques du tolbutamide

Christian Sergheraert, Pierre Marcincal, Etienne Cuingnet

Journal:

Journal of Organometallic Chemistry

Year:

1976

File:

PDF, 499 KB

1976

27

Convenient synthesis of tetrahydroisoquinoline-hydantoins

Julie Charton, Sandrine Delarue, Sandrine Vendeville, Marie-Ange Debreu-Fontaine, Sophie Girault-Mizzi, Christian Sergheraert

Journal:

Tetrahedron Letters

Year:

2001

Language:

english

File:

PDF, 93 KB

english, 2001

28

PyBroP: a convenient activator for the synthesis of formamidines

Sandrine Delarue, Christian Sergheraert

Journal:

Tetrahedron Letters

Year:

1999

Language:

english

File:

PDF, 185 KB

english, 1999

29

Parallel synthesis of a library of 1,4-naphthoquinones and automated screening of potential inhibitors of trypanothione reductase from Trypanosoma cruzi

Laurence Salmon-Chemin, Anick Lemaire, Stéphanie De Freitas, Benoı̂t Deprez, Christian Sergheraert, Elisabeth Davioud-Charvet

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2000

Language:

english

File:

PDF, 168 KB

english, 2000

30

Solid phase synthesis of trypanothione disulfide

Valéry Fauchet, Line Bourel, André Tartar, Christian Sergheraert

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1994

Language:

english

File:

PDF, 332 KB

english, 1994

31

Synthesis of non reducible inhibitors for trypanothione reductase from Trypanosoma cruzi.

Anne Tromelin, Mireille Moutiez, Djalal Meziane-Cherif, Marc Aumercier, André Tartar, Christian Sergheraert

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1993

Language:

english

File:

PDF, 344 KB

english, 1993

32

Antitrypanosomal activities and cytotoxicity of 5-nitro-2-furancarbohydrazides

Régis Millet, Louis Maes, Valérie Landry, Christian Sergheraert, Elisabeth Davioud-Charvet

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 129 KB

english, 2002

33

Design, synthesis and antimalarial activity of novel, quinoline-Based, zinc metallo-aminopeptidase inhibitors

Marian Flipo, Isabelle Florent, Philippe Grellier, Christian Sergheraert, Rebecca Deprez-Poulain

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2003

Language:

english

File:

PDF, 160 KB

english, 2003

34

Vasopressin trisulphide: synthesis, NMR study and affinity studies with V1 and V2 subtypes receptors

Mireille Moutiez, Guy Lippens, Christian Sergheraert, André Tartar

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1997

Language:

english

File:

PDF, 319 KB

english, 1997

35

Structure-activity relationships in 2-aminodiphenylsulfides against trypanothione reductase from Trypanosoma cruzi

Sophie Girault, Elisabeth Davioud-Charvet, Laurence Salmon, Amaya Berecibar, Marie-Ange Debreu, Christian Sergheraert

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1998

Language:

english

File:

PDF, 328 KB

english, 1998

36

Automated parallel synthesis of a tetrahydroisoquinolin-based library: Potential prolyl endopeptidase inhibitors

Sandrine Vendeville, Line Bourel, Elisabeth Davioud-Charvet, Philippe Grellier, Benoît Deprez, Christian Sergheraert

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1999

Language:

english

File:

PDF, 375 KB

english, 1999

37

Synthesis of polyamine derivatives for the preparation of affinity chromatography columns for the search of new Trypanosoma cruzi targets

Elisabeth Davioud-Charvet, Amaya Berecibar, Sophie Girault, Valérie Landry, Hervé Drobecq, Christian Sergheraert

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1999

Language:

english

File:

PDF, 307 KB

english, 1999

38

Potent and specific inhibitors of trypanothione reductase from Trypanosoma cruzi: bis(2-aminodiphenylsulfides) for fluorescent labeling studies

Sophie Girault, Elisabeth Davioud-Charvet, Louis Maes, Jean-François Dubremetz, Marie-Ange Debreu, Valérie Landry, Christian Sergheraert

Journal:

Bioorganic & Medicinal Chemistry

Year:

2001

Language:

english

File:

PDF, 763 KB

english, 2001

39

New spermine and spermidine derivatives as potent inhibitors of Trypanosoma cruzi Trypanothione Reductase

Béatrice Bonnet, David Soullez, Elisabeth Davioud-Charvet, Valérie Landry, Dragos Horvath, Christian Sergheraert

Journal:

Bioorganic & Medicinal Chemistry

Year:

1997

Language:

english

File:

PDF, 734 KB

english, 1997

40

Truncated beta-amyloid peptide species in pre-clinical Alzheimer's disease as new targets for the vaccination approach

Nicolas Sergeant, Stepanie Bombois, Antoine Ghestem, Hervé Drobecq, Vesna Kostanjevecki, Carla Missiaen, Annick Wattez, Jean-Phillipe David, Eugeen Vanmechelen, Christian Sergheraert, André Delacourte

Journal:

Journal of Neurochemistry

Year:

2003

Language:

english

File:

PDF, 255 KB

english, 2003

41

Design and synthesis of new leads for PKC bisubstrate inhibitors.

Martine He, Eric Buisine, André Tartar, Christian Sergheraert

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1994

Language:

english

File:

PDF, 406 KB

english, 1994

42

Comparison of the Inhibition of Human and Trypanosoma cruzi Prolyl Endopeptidases

Sandrine Vendeville, Filip Goossens, Marie-Ange Debreu-Fontaine, Valérie Landry, Elisabeth Davioud-Charvet, Philippe Grellier, Simon Scharpe, Christian Sergheraert

Journal:

Bioorganic & Medicinal Chemistry

Year:

2002

Language:

english

File:

PDF, 213 KB

english, 2002

43

Trypanothione reductase inhibition/trypanocidal activity relationships in a 1,4-bis(3-aminopropyl)piperazine series

Béatrice Bonnet, David Soullez, Sophie Girault, Louis Maes, Valérie Landry, Elisabeth Davioud-Charvet, Christian Sergheraert

Journal:

Bioorganic & Medicinal Chemistry

Year:

2000

Language:

english

File:

PDF, 223 KB

english, 2000

44

Lacrimal Gland Functions Are Differentially Controlled by Protein Kinase C Isoforms

DRISS ZOUKHRI, ROBIN R. HODGES, CHRISTIAN SERGHERAERT, DARLENE A. DARTT

Journal:

Annals of the New York Academy of Sciences

Year:

1998

File:

PDF, 269 KB

1998

45

Glucose regulates LXRα subcellular localization and function in rat pancreatic β-cells

Helleboid-Chapman, Audrey, Helleboid, Stéphane, Jakel, Heidelinde, Timmerman, Catherine, Sergheraert, Christian, Pattou, François, Fruchart-Najib, Jamila, Fruchart, Jean-Charles

Journal:

Year:

2006

Language:

english

File:

PDF, 635 KB

english, 2006

46

The rat lacrimal gland expresses the α isoform of PKC. Further evidence for the PMA-activated and phospholipid-independent protein kinase activity

Driss Zoukhri, Jean-Marc Pelosin, Philippe Mauduit, Edmond Chambaz, Christian Sergheraert, Bernard Rossignol

Journal:

Cellular Signalling

Year:

1992

Language:

english

File:

PDF, 564 KB

english, 1992

47

Photosubstitution of cymantrenylalanine as a tool in peptide chemistry : Synthesis and biological activity of new GnRH analogs

ANNIE RICOUART, PIERRETTE MAES, THIERRY BATTMANN, BERNARD KERDELHUE, ANDRÉ TARTAR, CHRISTIAN SERGHERAERT

Journal:

Chemical Biology & Drug Design

Year:

1988

Language:

english

File:

PDF, 524 KB

english, 1988

48

2- and 3-Substituted 1,4-Naphthoquinone Derivatives as Subversive Substrates of Trypanothione Reductase and Lipoamide Dehydrogenase from Trypanosoma cruzi: Synthesis and Correlation between Redox Cycling Activities and in Vitro Cytotoxicity

Salmon-Chemin, Laurence, Buisine, Eric, Yardley, Vanessa, Kohler, Sven, Debreu, Marie-Ange, Landry, Valérie, Sergheraert, Christian, Croft, Simon L., Krauth-Siegel, R. Luise, Davioud-Charvet, Elisabet

Journal:

Journal of Medicinal Chemistry

Year:

2001

Language:

english

File:

PDF, 468 KB

english, 2001

49

Inhibition of protein kinase C by retro-inverso pseudosubstrate analogues

Annie Ricouart, André Tartar, Christian Sergheraert

Journal:

Biochemical and Biophysical Research Communications

Year:

1989

Language:

english

File:

PDF, 491 KB

english, 1989

50

Comparative efficiency of simple lipopeptide constructs for in vivo induction of virus-specific CTL

Benoît Deprez, Jean-Pierre Sauzet, Christophe Boutillon, Frédéric Martinon, André Tartar, Christian Sergheraert, Jean-Gérard Guillet, Elisabeth Gomard, Hélène Gras-Masse

Journal:

Year:

1996

Language:

english

File:

PDF, 994 KB

english, 1996