Chaim GILON: search on Z-Library

The world's largest scientific articles store. 70,000,000+ articles for free.

Don't use scam websites

1

1H-nmr studies of receptor-selective substance P analogues reveal distinct predominant conformations in DMSO-d6

Dina Levian-Teitelbaum, Nancy Kolodny, Michael Chorev, Zvi Selinger, Chaim Gilon

Journal:

Year:

1989

Language:

english

File:

PDF, 812 KB

english, 1989

2

Improving Oral Bioavailability of Peptides by Multiple N-Methylation: Somatostatin Analogues

Eric Biron, Jayanta Chatterjee, Oded Ovadia, Daniel Langenegger, Joseph Brueggen, Daniel Hoyer, Herbert A. Schmid, Raz Jelinek, Chaim Gilon, Amnon Hoffman, Horst Kessler

Journal:

Angewandte Chemie International Edition

Year:

2008

Language:

english

File:

PDF, 477 KB

english, 2008

3

Characterization of a putative pheromone biosynthesis-activating neuropeptide (PBAN) receptor from the pheromone gland of Heliothis peltigera

Altstein, Miriam, Gabay, Tal, Ben-Aziz, Orna, Daniel, Shai, Zeltser, Irina, Gilon, Chaim

Journal:

Invertebrate Neuroscience

Year:

1999

Language:

english

File:

PDF, 161 KB

english, 1999

4

The Molecular Basis of Memory

Marx, Gerard, Gilon, Chaim

Journal:

ACS Chemical Neuroscience

Year:

2012

Language:

english

File:

PDF, 2.20 MB

english, 2012

5

Characterization of a putative pheromone biosynthesis-activating neuropeptide (PBAN) receptor from the pheromone gland ofHeliothis peltigera

Miriam Altstein, Tal Gabay, Orna Ben-Aziz, Shai Daniel, Irina Zeltser, Chaim Gilon

Journal:

Invertebrate Neuroscience

Year:

1999

Language:

english

File:

PDF, 161 KB

english, 1999

6

Esterification of Polyethylene Glycols

Zalipsky, Samuel, Gilon, Chaim, Zilkha, Albert

Journal:

Journal of Macromolecular Science Part A - Chemistry

Year:

1984

Language:

english

File:

PDF, 319 KB

english, 1984

7

cis -Peptide Bonds: A Key for Intestinal Permeability of Peptides?

Marelli, Udaya Kiran, Ovadia, Oded, Frank, Andreas Oliver, Chatterjee, Jayanta, Gilon, Chaim, Hoffman, Amnon, Kessler, Horst

Journal:

Chemistry - A European Journal

Year:

2015

Language:

english

File:

PDF, 1.72 MB

english, 2015

8

Enhancing oral bioavailability of cyclic RGD hexa-peptides by the Lipophilic Prodrug Charge Masking approach: Redirection of peptide intestinal permeability from paracellular to transcellular pathway

Schumacher-Klinger, Adi, Fanous, Joseph, Merzbach, Shira, Weinmueller, Michael, Reichart, Florian, Räder, Andreas F. B., Gitlin-Domaglaska, Agata, Gilon, Chaim, Kessler, Horst, Hoffman, Amnon

Journal:

Molecular Pharmaceutics

Year:

2018

Language:

english

File:

PDF, 1.40 MB

english, 2018

9

Die Verbesserung der oralen Bioverfügbarkeit von Peptiden durch multiple N-Methylierung: Somatostatin-Analoga

Eric Biron, Jayanta Chatterjee, Oded Ovadia, Daniel Langenegger, Joseph Brueggen, Daniel Hoyer, Herbert A. Schmid, Raz Jelinek, Chaim Gilon, Amnon Hoffman, Horst Kessler

Journal:

Angewandte Chemie

Year:

2008

Language:

german

File:

PDF, 477 KB

german, 2008

10

A rapid method for the preparation of amino acid resin esters for merrifield solid-phase peptide synthesis

Michael W. Monahan, Chaim Gilon

Journal:

Year:

1973

Language:

english

File:

PDF, 389 KB

english, 1973

11

Synthesis of pyroglutamyl-histidyl-thiazolidine-4-carboxamide, a biologically active analog of the thyrotropin relasing factor

C. Grant Willson, Chaim Gilon, Bernard Donzel, Murray Goodman

Journal:

Year:

1976

Language:

english

File:

PDF, 284 KB

english, 1976

12

Sequential polypeptides by matrix-controlled thermal polymerization. Synthesis and racemization studies

Maria Sakarellos-Daitsiotis, Chaim Gilon, Constantinos Sakarellos, Murray Goodman

Journal:

Year:

1977

Language:

english

File:

PDF, 750 KB

english, 1977

13

Development of bifunctional photoactivatable benzophenone probes and their application to glycoside substrates

Nir Qvit, Galya Monderer-Rothkoff, Ayelet Ido, Deborah E. Shalev, Orna Amster-Choder, Chaim Gilon

Journal:

Year:

2008

Language:

english

File:

PDF, 510 KB

english, 2008

14

Structure-activity relationship and metabolic stability studies of backbone cyclization and N-methylation of melanocortin peptides

Yaniv Linde, Oded Ovadia, Eli Safrai, Zhimin Xiang, Federico P. Portillo, Deborah E. Shalev, Carrie Haskell-Luevano, Amnon Hoffman, Chaim Gilon

Journal:

Year:

2008

Language:

english

File:

PDF, 314 KB

english, 2008

15

Design and synthesis of backbone cyclic phosphorylated peptides: The IκB model

Nir Qvit, Ada Hatzubai, Deborah E. Shalev, Assaf Friedler, Yinon Ben-Neriah, Chaim Gilon

Journal:

Year:

2009

Language:

english

File:

PDF, 428 KB

english, 2009

16

1H-NMR studies on substance P hexapeptide analogs

Anthony Ribeiro, Oleg Jardetzky, Chaim Gilon, Dina Teitelbaum, Michael Chorev

Journal:

Year:

1983

Language:

english

File:

PDF, 323 KB

english, 1983

17

The crystal structure of the photosynthetic inhibitors DCMU and DTPU

Chaim Gilon, Shmuel Cohen, Yona Siderer

Journal:

Year:

1986

Language:

english

File:

PDF, 377 KB

english, 1986

18

Backbone cyclization: A new method for conferring conformational constraint on peptides

Chaim Gilon, David Halle, Michael Chorev, Zvi Selincer, Gerardo Byk

Journal:

Year:

1991

Language:

english

File:

PDF, 520 KB

english, 1991

19

Toward nonpeptidal substance P mimetic analogues: Design, synthesis, and biological activity

Michael Chorev, Eli Roubini, Chaim Gilon, Zvi Selincer

Journal:

Year:

1991

Language:

english

File:

PDF, 663 KB

english, 1991

20

ChemInform Abstract: New Perspective in Peptide Chemistry by N-Alkylation

Horst Kessler, Jayanta Chatterjee, Lucas Doedens, Florian Operrer, Eric Biron, Daniel Hoyer, Herbert Schmid, Chaim Gilon, Victor J. Hruby, Dale F. Mierke

Journal:

Year:

2011

File:

PDF, 18 KB

2011

21

Polydepsipeptides, 4 Synthesis of the alternating Polydepsipeptides Poly(Ala-Lac) and Poly(Val-Lac)

Dietmar Nissen, Chaim Gilon, Murray Goodman

Journal:

Macromolecular Chemistry and Physics

Year:

1975

Language:

english

File:

PDF, 1.33 MB

english, 1975

22

Building units for N-Backbone cyclic peptides. 2. Synthesis of protected N-(ω-thioalkylene) amino acids and their incorporation into dipeptide units

Gal Bilan, Chaim Gilon

Journal:

Year:

1995

Language:

english

File:

PDF, 636 KB

english, 1995

23

An improved method for the catalytic preparation of t-butyl esters of carboxylic and fatty acids

Harold Wiener, Chaim Gilon

Journal:

Journal of Molecular Catalysis

Year:

1986

Language:

english

File:

PDF, 461 KB

english, 1986

24

The effect of backbone cyclization on PK/PD properties of bioactive peptide-peptoid hybrids: The melanocortin agonist paradigm

Oded Ovadia, Yaniv Linde, Carrie Haskell-Luevano, Marvin L. Dirain, Tanya Sheynis, Raz Jelinek, Chaim Gilon, Amnon Hoffman

Journal:

Bioorganic & Medicinal Chemistry

Year:

2010

Language:

english

File:

PDF, 496 KB

english, 2010

25

Rational conversion of noncontinuous active region in proteins into a small orally bioavailable macrocyclic drug-like molecule: The HIV-1 CD4:gp120 paradigm

Mattan Hurevich, Avi Swed, Salim Joubran, Shira Cohen, Noam S. Freeman, Elena Britan-Rosich, Laurence Briant-Longuet, Martine Bardy, Christian Devaux, Moshe Kotler, Amnon Hoffman, Chaim Gilon

Journal:

Bioorganic & Medicinal Chemistry

Year:

2010

Language:

english

File:

PDF, 542 KB

english, 2010

26

Cyclic peptide inhibitors of HIV-1 integrase derived from the LEDGF/p75 protein

Zvi Hayouka, Mattan Hurevich, Aviad Levin, Hadar Benyamini, Anat Iosub, Michal Maes, Deborah E. Shalev, Abraham Loyter, Chaim Gilon, Assaf Friedler

Journal:

Bioorganic & Medicinal Chemistry

Year:

2010

Language:

english

File:

PDF, 965 KB

english, 2010

27

Synthesis of N′-substituted Ddz-protected hydrazines and their application in solid phase synthesis of aza-peptides

Noam S. Freeman, Mattan Hurevich, Chaim Gilon

Journal:

Year:

2009

Language:

english

File:

PDF, 587 KB

english, 2009

28

A novel method for the facile synthesis of depsipeptides

Chaim Gilon, Yakir Klausner, Alfred Hassner

Journal:

Tetrahedron Letters

Year:

1979

Language:

english

File:

PDF, 174 KB

english, 1979

29

Synthesis and biological activity of semipeptoid farnesyltransferase inhibitors

Hadas Reuveni, Alex Gitler, Enrique Poradosu, Chaim Gilon, Alexander Levitzki

Journal:

Bioorganic & Medicinal Chemistry

Year:

1997

Language:

english

File:

PDF, 762 KB

english, 1997

30

Novel method for the synthesis of urea backbone cyclic peptides using new Alloc-protected glycine building units

Mattan Hurevich, Yftah Tal-Gan, Shoshana Klein, Yaniv Barda, Alexander Levitzki, Chaim Gilon

Journal:

Journal of Peptide Science

Year:

2010

Language:

english

File:

PDF, 281 KB

english, 2010

31

A Bioactive Somatostatin Analog without a Type II′ β-Turn: Synthesis and Conformational Analysis in Solution

Shaokai Jiang, Sharon Gazal, Gary Gelerman, Ofer Ziv, Olga Karpov, Pninit Litman, Moshe Bracha, Michael Afargan, Chaim Gilon, Murray Goodman

Journal:

Journal of Peptide Science

Year:

2001

Language:

english

File:

PDF, 2.16 MB

english, 2001

32

Novel cyclic azo-bridged analogs of gonadotropin-releasing hormone

Gil Fridkin, Shai Rahimipour, Nurit Ben-Aroya, Aviva Kapitkovsky, Susanna Di-Segni, Masha Rosenberg, Irina Kustanovich, Yitzhak Koch, Chaim Gilon, Mati Fridkin

Journal:

Journal of Peptide Science

Year:

2006

Language:

english

File:

PDF, 239 KB

english, 2006

33

Backbone Cyclization of the C-terminal Part of Substance P. Part 1: The Important Role of the Sulphur in Position 11

Gal Bitan, Irena Zeltser, Gerardo Byk, David Halle, Yaffa Mashriki, Evgenia V. Gluhov, Inna Sukhotinsky, Menachem Hanani, Zvi Selinger, Chaim Gilon

Journal:

Journal of Peptide Science

Year:

1996

Language:

english

File:

PDF, 717 KB

english, 1996

34

New backbone cyclic substance P analogs

Gal Bitan, Stephan Behrens, Barbara Mathä, Yaffa Mashriki, Menachem Hanani, Horst Kessler, Chaim Gilon

Journal:

International Journal of Peptide Research and Therapeutics

Year:

1995

Language:

english

File:

PDF, 251 KB

english, 1995

35

Synthesis of a bicyclic BPTI mimetic containing 4-thioproline replacing Cys38

Ron Kasher, Gal Bitan, Christeen Halloun, Chaim Gilon

Journal:

International Journal of Peptide Research and Therapeutics

Year:

1998

Language:

english

File:

PDF, 187 KB

english, 1998

36

Rationally designed neuropeptide antagonists: A novel approach for generation of environmentally friendly insecticides

Chaim Gilon, Irina Zeltser, Shai Daniel, Orna Ben-Aziz, Irit Schefler, Miriam Altstein

Journal:

Invertebrate Neuroscience

Year:

1997

Language:

english

File:

PDF, 530 KB

english, 1997

37

Synthesis and structure–activity relationship studies of peptidomimetic PKB/Akt inhibitors: The significance of backbone interactions

Yftah Tal-Gan, Noam S. Freeman, Shoshana Klein, Alexander Levitzki, Chaim Gilon

Journal:

Bioorganic & Medicinal Chemistry

Year:

2010

Language:

english

File:

PDF, 903 KB

english, 2010

38

Ion-exchange chromatographic assay of peptidases acting on the C-terminal hexapeptide sequence of substance P

Ralph Laufer, Uri Wormser, Zvi Selinger, Michael Chorev, Chaim Gilon

Journal:

Journal of Chromatography A

Year:

1984

Language:

english

File:

PDF, 659 KB

english, 1984

39

Synthesis and biological activity of novel backbone-bicyclic Substance-P analogs containing lactam and disulfide bridges

GAL BITAN, INNA SUKHOTINSKY, YAFHA MASHRIKI, MENACHEM HANANI, ZVI SELINGER, CHAIM GILON

Journal:

Chemical Biology & Drug Design

Year:

1997

Language:

english

File:

PDF, 421 KB

english, 1997

40

Metabolic Stability of Peptidomimetics: N-Methyl and Aza Heptapeptide Analogs of a PKB/Akt Inhibitor

Yftah Tal-Gan, Noam S. Freeman, Shoshana Klein, Alexander Levitzki, Chaim Gilon

Journal:

Chemical Biology & Drug Design

Year:

2011

Language:

english

File:

PDF, 380 KB

english, 2011

41

Synthesis of a bicyclic BPTI mimetic containing 4-thioproline replacing Cys38

Ron Kasher, Gal Bitan, Christeen Halloun, Chaim Gilon

Journal:

International Journal of Peptide Research and Therapeutics

Year:

1998

Language:

english

File:

PDF, 81 KB

english, 1998

42

Effect of Structural and Conformation Modifications, Including Backbone Cyclization, of Hydrophilic Hexapeptides on Their Intestinal Permeability and Enzymatic Stability

Hess, Shmuel, Ovadia, Oded, Shalev, Deborah E., Senderovich, Hanoch, Qadri, Bashir, Yehezkel, Tamar, Salitra, Yoseph, Sheynis, Tania, Jelinek, Raz, Gilon, Chaim

Journal:

Journal of Medicinal Chemistry

Year:

2007

Language:

english

File:

PDF, 287 KB

english, 2007

43

Building Units for N-Backbone Cyclic Peptides. 3. Synthesis of Protected Nα-(ω-Aminoalkyl)amino Acids and Nα-(ω-Carboxyalkyl)amino Acids

Muller, Dan, Zeltser, Irena, Bitan, Gal, Gilon, Chaim

Journal:

Journal of Organic Chemistry

Year:

1997

Language:

english

File:

PDF, 227 KB

english, 1997

44

Intestinal Permeability of Cyclic Peptides: Common Key Backbone Motifs Identified

Beck, Johannes G., Chatterjee, Jayanta, Laufer, Burkhardt, Kiran, Marelli Udaya, Frank, Andreas O., Neubauer, Stefanie, Ovadia, Oded, Greenberg, Sarit, Gilon, Chaim, Hoffman, Amnon, Kessler, Horst

Journal:

Journal of the American Chemical Society

Year:

2012

Language:

english

File:

PDF, 3.56 MB

english, 2012

45

Importance of delaying balloon angioplasty in patients with unstable angina pectoris

Youseph Rozenman, Dan Gilon, Julian Zeilingher, Dan Sapoznikov, Chaim Lotan, Morris Mosseri, A. Teddy Weiss, Yonathan Hasin, Mervyn S. Gotsman

Journal:

Clinical Cardiology

Year:

1996

Language:

english

File:

PDF, 426 KB

english, 1996

46

Plasma lipoproteins are not related to restenosis after successful coronary angioplasty

Yoseph Rozenman, Dan Gilon, Sima Welber, Dan Sapoznikov, Chaim Lotan, Michael Geist, A.Teddy Weiss, Yonathan Hasin, Mervyn S. Gotsman

Journal:

The American Journal of Cardiology

Year:

1993

Language:

english

File:

PDF, 303 KB

english, 1993

47

Studying protein–peptide interactions using benzophenone units: A case study of protein kinase B/Akt and its inhibitor PTR6154

Yftah Tal-Gan, Shirly Naveh, Shoshana Klein, Ofra Moshel, Alexander Levitzki, Chaim Gilon

Journal:

Analytical Biochemistry

Year:

2012

Language:

english

File:

PDF, 509 KB

english, 2012

48

A comparative study of backbone versus side chain peptide cyclization: Application for HIV-1 integrase inhibitors

Zvi Hayouka, Aviad Levin, Mattan Hurevich, Deborah E. Shalev, Abraham Loyter, Chaim Gilon, Assaf Friedler

Journal:

Bioorganic & Medicinal Chemistry

Year:

2012

Language:

english

File:

PDF, 741 KB

english, 2012

49

Developing potent backbone cyclic peptides bearing the shared epitope sequence as rheumatoid arthritis drug-leads

Shirly Naveh, Yftah Tal-Gan, Song Ling, Amnon Hoffman, Joseph Holoshitz, Chaim Gilon

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2012

Language:

english

File:

PDF, 444 KB

english, 2012

50

Influence of coronary angioplasty on the progression of coronary atherosclerosis

Yoseph Rozenman, Dan Gilon, Sima Welber, Dan Sapoznikov, Chaim Lotan, Morris Mosseri, A.Teddy Weiss, Yonathan Hasin, Mervyn S. Gotsman

Journal:

The American Journal of Cardiology

Year:

1995

Language:

english

File:

PDF, 595 KB

english, 1995