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101

Synthesis of new 2,3-diaryl-1,3-thiazolidin-4-ones as anti-HIV agents

Angela Rao, Jan Balzarini, Anna Carbone, Alba Chimirri, Erik De Clercq, Anna Maria Monforte, Pietro Monforte, Christophe Pannecouque, Maria Zappalà

Journal:

Year:

2004

Language:

english

File:

PDF, 160 KB

english, 2004

102

Synthesis and anticonvulsant activity of N-3 substituted 2,3-benzodiazepines

Silvana Quartarone, Roberta Caruso, Valèrie Orlando, Emilio Russo, Giovambattista De Sarro, Alba Chimirri

Journal:

Year:

2004

Language:

english

File:

PDF, 195 KB

english, 2004

103

Comparative anticonvulsant activity of N-acetyl-1-aryl-6,7-dimethoxy-1,2,3,4-tetrahydroisoquinoline derivatives in rodents

Guido Ferreri, Alba Chimirri, Emilio Russo, Rosaria Gitto, Pietro Gareri, Angela De Sarro, Giovambattista De Sarro

Journal:

Pharmacology Biochemistry and Behavior

Year:

2004

Language:

english

File:

PDF, 377 KB

english, 2004

104

Group III mGlu receptor agonists potentiate the anticonvulsant effect of AMPA and NMDA receptor block

Giovambattista De Sarro, Alba Chimirri, Brian S Meldrum

Journal:

European Journal of Pharmacology

Year:

2002

Language:

english

File:

PDF, 240 KB

english, 2002

105

Synthesis and anticonvulsant properties of 2,3,3a,4-tetrahydro-1H-pyrrolo[1,2-a]benzimidazol-1-one derivatives

Alba Chimirri, Angela De Sarro, Giovambattista De Sarro, Rosaria Gitto, Maria Zappalà

Journal:

Year:

2001

Language:

english

File:

PDF, 106 KB

english, 2001

106

Synthesis and anti-HIV activity of 2,3-diaryl-1,3-thiazolidin-4-ones

Angela Rao, Anna Carbone, Alba Chimirri, Erik De Clercq, Anna Maria Monforte, Pietro Monforte, Christophe Pannecouque, Maria Zappalà

Journal:

Year:

2003

Language:

english

File:

PDF, 131 KB

english, 2003

107

Synthesis and pharmacological properties of new 3-ethoxycarbonyl-11H-[1,2,4]triazolo[4,5-c][2,3]benzodiazepines

A Chimirri, Rosaria Gitto, S Quartarone, V Orlando, A De Sarro, G.B De Sarro

Journal:

Year:

2002

Language:

english

File:

PDF, 156 KB

english, 2002

108

Binding modes of noncompetitive AMPA antagonists: a computational approach

Laura De Luca, Antonio Macchiarulo, Gabriele Costantino, Maria Letizia Barreca, Rosaria Gitto, Alba Chimirri, Roberto Pellicciari

Journal:

Year:

2003

Language:

english

File:

PDF, 1017 KB

english, 2003

109

Synthesis and anti-HIV activity of 2,3-diaryl-1,3-thiazolidin-4-(thi)one derivatives

Angela Rao, Anna Carbone, Alba Chimirri, Erik De Clercq, Anna Maria Monforte, Pietro Monforte, Christophe Pannecouque, Maria Zappalà

Journal:

Year:

2002

Language:

english

File:

PDF, 116 KB

english, 2002

110

Synthesis and anti-HIV activity of 1-(2,6-difluorophenyl)-1H,3H-thiazolo[3,4-a]benzimidazole structurally-related 1,2-substituted benzimidazoles

Angela Rao, Alba Chimirri, Erik De Clercq, Anna Maria Monforte, Pietro Monforte, Christophe Pannecouque, Maria Zappalà

Journal:

Year:

2002

Language:

english

File:

PDF, 182 KB

english, 2002

111

Anti-HIV agents: design and discovery of new potent RT inhibitors

Maria Letizia Barreca, Alba Chimirri, Erik De Clercq, Laura De Luca, Anna-Maria Monforte, Pietro Monforte, Angela Rao, Maria Zappalà

Journal:

Year:

2003

Language:

english

File:

PDF, 139 KB

english, 2003

112

Comparative anticonvulsant activity of some 2,3-benzodiazepine derivatives in rodents

Giovambattista De Sarro, Guido Ferreri, Pietro Gareri, Emilio Russo, Angela De Sarro, Rosaria Gitto, Alba Chimirri

Journal:

Pharmacology Biochemistry and Behavior

Year:

2003

Language:

english

File:

PDF, 280 KB

english, 2003

113

Anticonvulsant Activity of Azirino[1,2-d] [1,4]Benzodiazepines and Related 1,4-Benzodiazepines in Mice

Giovambattista De Sarro, Alba Chimirri, Ruth Mckernan, Kathleen Quirk, Piero Giusti, Angela De Sarro

Journal:

Pharmacology Biochemistry and Behavior

Year:

1997

Language:

english

File:

PDF, 248 KB

english, 1997

114

Relationship Between Anticonvulsant Activity and Plasma Level of Some 2,3-Benzodiazepines in Genetically Epilepsy-Prone Rats

Giovambattista De Sarro, Milena Rizzo, Vincenzo Antonio Sinopoli, Rosaria Gitto, Angela De Sarro, Maria Zappala, Alba Chimirri

Journal:

Pharmacology Biochemistry and Behavior

Year:

1998

Language:

english

File:

PDF, 138 KB

english, 1998

115

Anticonvulsant Activity and Plasma Level of 2,3-Benzodiazepin-4-ones (CFMs) in Genetically Epilepsy-Prone Rats

Giovambattista De Sarro, Milena Rizzo, Cinzia Spagnolo, Rosaria Gitto, Angela De Sarro, Gisella Scotto, Maria Zappala, Alba Chimirri

Journal:

Pharmacology Biochemistry and Behavior

Year:

1999

Language:

english

File:

PDF, 178 KB

english, 1999

116

18 Synthesis and metabolic study of 1H,3H-oxazolo[3,4-a]benzimidazoles, a new class of non-nucleoside HIV-1 RT inhibitors

A. Chimirri, E. De Clercq, A.M. Monforte, P. Monforte, C. Pannecouque, A. Rao, M. Witvrouw, M. Zappalà

Journal:

Antiviral Research

Year:

2000

Language:

english

File:

PDF, 54 KB

english, 2000

117

Azirino[1, 2-d][1, 4]benzodiazepine derivatives and related 1,4-benzodiazepines as anticonvulsant agents in DBA/2 mice

Giovambattista De Sarro, Alba Chimirri, Maria Zappala, Piero Guisti, Maria Lipartiti, Angela De Sarro

Journal:

General Pharmacology: The Vascular System

Year:

1996

Language:

english

File:

PDF, 813 KB

english, 1996

118

Docking Studies on a New Human Immodeficiency Virus Integrase−Mg−DNA Complex: Phenyl Ring Exploration and Synthesis of 1H-Benzylindole Derivatives through Fluorine Substitutions

Ferro, Stefania, De Luca, Laura, Barreca, Maria Letizia, Iraci, Nunzio, De Grazia, Sara, Christ, Frauke, Witvrouw, Myriam, Debyser, Zeger, Chimirri, Alba

Journal:

Journal of Medicinal Chemistry

Year:

2009

Language:

english

File:

PDF, 795 KB

english, 2009

119

Synthesis and Structural Features of New Cyclofunctionalized Benzimidazoles

Chimirri, Alba, Maria Monforte, Anna, Monforte, Pietro, Nicolò, Francesco, Rao, Angela, Zappalà, Maria

Journal:

Year:

2000

Language:

english

File:

PDF, 55 KB

english, 2000

120

GYKI 52466 and related 2,3-benzodiazepines as anticonvulsant agents in DBA/2 mice

Giovambattista De Sarro, Alba Chimirri, Angela De Sarro, Rosaria Gitto, Silvana Grasso, Piero Giusti, Astrid G. Chapman

Journal:

European Journal of Pharmacology

Year:

1995

Language:

english

File:

PDF, 1.09 MB

english, 1995

121

Analysis of the full-length integrase–DNA complex by a modified approach for DNA docking

Laura De Luca, Alessandro Pedretti, Giulio Vistoli, Maria Letizia Barreca, Luigi Villa, Pietro Monforte, Alba Chimirri

Journal:

Biochemical and Biophysical Research Communications

Year:

2003

Language:

english

File:

PDF, 147 KB

english, 2003

122

Molecular dynamics studies of the full-length integrase–DNA complex

Laura De Luca, Giulio Vistoli, Alessandro Pedretti, Maria Letizia Barreca, Alba Chimirri

Journal:

Biochemical and Biophysical Research Communications

Year:

2005

Language:

english

File:

PDF, 331 KB

english, 2005

123

Anti-enterovirus activity and structure–activity relationship of a series of 2,6-dihalophenyl-substituted 1H,3H-thiazolo[3,4-a]benzimidazoles

Armando M. De Palma, Ward Heggermont, Pieter Leyssen, Gerhard Pürstinger, Eva Wimmer, Erik De Clercq, Angela Rao, Anna-Maria Monforte, Alba Chimirri, Johan Neyts

Journal:

Biochemical and Biophysical Research Communications

Year:

2007

Language:

english

File:

PDF, 135 KB

english, 2007

124

Tn5 transposase as a useful platform to simulate HIV-1 integrase inhibitor binding mode

Maria Letizia Barreca, Francesco Ortuso, Nunzio Iraci, Laura De Luca, Stefano Alcaro, Alba Chimirri

Journal:

Biochemical and Biophysical Research Communications

Year:

2007

Language:

english

File:

PDF, 707 KB

english, 2007

125

Effects of non-competitive AMPA receptor antagonists injected into some brain areas of WAG/Rij rats, an animal model of generalized absence epilepsy

Rita Citraro, Emilio Russo, Santo Gratteri, Eugenio Donato Di Paola, Guido Ferreri Ibbadu, Carmela Curinga, Rosaria Gitto, Alba Chimirri, Giuseppe Donato, Giovambattista De Sarro

Journal:

Neuropharmacology

Year:

2006

Language:

english

File:

PDF, 1.06 MB

english, 2006

126

Enhancement of anti-absence effects of ethosuximide by low doses of a noncompetitive α-amino-3-hydroxy-5-methyl-4-isoxazolepropionic acid (AMPA) receptor antagonist in a genetic animal model of absence epilepsy

Emilio Russo, Rita Citraro, Salvatore De Fazio, Rosario Marra, Rosaria Gitto, Alba Chimirri, Giovambattista De Sarro, Eugenio Donato Di Paola

Journal:

Epilepsy & Behavior

Year:

2008

Language:

english

File:

PDF, 188 KB

english, 2008

127

Apoptotic effects of thiazolobenzimidazole derivatives on sensitive and multidrug resistant leukaemic cells

S Grimaudo, M.V Raimondi, F Capone, A Chimirri, F Poretto, A.M Monforte, D Simoni, M Tolomeo

Journal:

European Journal of Cancer

Year:

2001

Language:

english

File:

PDF, 280 KB

english, 2001

128

Selective induction of apoptosis in multidrug resistant HL60R cells by the thiazolobenzoimidazole derivative 1-(2,6-difluorophenyl)-1H,3H-thiazolo [3,4-a] benzimidazole (TBZ)

S Grimaudo, M Tolomeo, A Chimirri, M Zappala, R.A Gancitano, N D’Alessandro

Journal:

European Journal of Cancer

Year:

1998

Language:

english

File:

PDF, 580 KB

english, 1998

129

AMPA receptor antagonists

Chimirri, Alba, Gitto, Rosaria, Zappalà, Maria

Journal:

Expert Opinion on Therapeutic Patents

Year:

1999

Language:

english

File:

PDF, 140 KB

english, 1999

130

Synthesis and Biological Characterization of 3-Substituted 1 H -Indoles as Ligands of GluN2B-Containing N -Methyl- d -aspartate Receptors. Part 2

Gitto, Rosaria, De Luca, Laura, Ferro, Stefania, Buemi, Maria R., Russo, Emilio, De Sarro, Giovambattista, Chisari, Mariangela, Ciranna, Lucia, Chimirri, Alba

Journal:

Journal of Medicinal Chemistry

Year:

2012

Language:

english

File:

PDF, 395 KB

english, 2012

131

Insight into the Fundamental Interactions between LEDGF Binding Site Inhibitors and Integrase Combining Docking and Molecular Dynamics Simulations

De Luca, Laura, Morreale, Francesca, Chimirri, Alba

Journal:

Journal of Chemical Information and Modeling

Year:

2012

Language:

english

File:

PDF, 1.92 MB

english, 2012

132

Molecular Dynamics Studies of the Wild-Type and Double Mutant HIV-1 Integrase Complexed with the 5CITEP Inhibitor: Mechanism for Inhibition and Drug Resistance

Barreca, Maria L., Lee, Keun Woo, Chimirri, Alba, Briggs, James M.

Journal:

Biophysical Journal

Year:

2003

Language:

english

File:

PDF, 549 KB

english, 2003

133

Pharmacophore-Based Design of HIV-1 Integrase Strand-Transfer Inhibitors

Barreca, Maria Letizia, Ferro, Stefania, Rao, Angela, De Luca, Laura, Zappalà, Maria, Monforte, Anna-Maria, Debyser, Zeger, Witvrouw, Myriam, Chimirri, Alba

Journal:

Journal of Medicinal Chemistry

Year:

2005

Language:

english

File:

PDF, 239 KB

english, 2005

134

Protective activity of α-lactoalbumin (ALAC), a whey protein rich in tryptophan, in rodent models of epileptogenesis

Russo, E., Scicchitano, F., Citraro, R., Aiello, R., Camastra, C., Mainardi, P., Chimirri, S., Perucca, E., Donato, G., De Sarro, G.

Journal:

Year:

2012

Language:

english

File:

PDF, 354 KB

english, 2012

135

Design, Synthesis, Structure−Activity Relationships, and Molecular Modeling Studies of 2,3-Diaryl-1,3-thiazolidin-4-ones as Potent Anti-HIV Agents

Barreca, Maria L., Balzarini, Jan, Chimirri, Alba, Clercq, Erik De, Luca, Laura De, Höltje, Hans Dieter, Höltje, Monika, Monforte, Anna Maria, Monforte, Pietro, Pannecouque, Christophe, Rao, Angela, Z

Journal:

Journal of Medicinal Chemistry

Year:

2002

Language:

english

File:

PDF, 154 KB

english, 2002

136

Structural Basis for the Interaction Between Carbonic Anhydrase and 1,2,3,4-tetrahydroisoquinolin-2-ylsulfonamides

Mader, Pavel, Brynda, Jiří, Gitto, Rosaria, Agnello, Stefano, Pachl, Petr, Supuran, Claudiu T., Chimirri, Alba, Řezáčová, Pavlína

Journal:

Journal of Medicinal Chemistry

Year:

2011

Language:

english

File:

PDF, 4.08 MB

english, 2011

137

New AMPA antagonists in epilepsy

Russo, Emilio, Gitto, Rosaria, Citraro, Rita, Chimirri, Alba, De Sarro, Giovambattista

Journal:

Expert Opinion on Investigational Drugs

Year:

2012

Language:

english

File:

PDF, 602 KB

english, 2012

138

Indole derivatives as dual-effective agents for the treatment of neurodegenerative diseases: Synthesis, biological evaluation, and molecular modeling studies

Buemi, Maria Rosa, De Luca, Laura, Chimirri, Alba, Ferro, Stefania, Gitto, Rosaria, Alvarez-Builla, Julio, Alajarin, Ramon

Journal:

Bioorganic & Medicinal Chemistry

Year:

2013

Language:

english

File:

PDF, 642 KB

english, 2013

139

Computational Strategies in Discovering Novel Non-nucleoside Inhibitors of HIV-1 RT

Barreca, Maria Letizia, Rao, Angela, De Luca, Laura, Zappalà, Maria, Monforte, Anna-Maria, Maga, Giovanni, Pannecouque, Christophe, Balzarini, Jan, De Clercq, Erik, Chimirri, Alba, Monforte, Pietro

Journal:

Journal of Medicinal Chemistry

Year:

2005

Language:

english

File:

PDF, 297 KB

english, 2005

140

Binding Mode Prediction of Strand Transfer HIV-1 Integrase Inhibitors Using Tn5 Transposase as a Plausible Surrogate Model for HIV-1 Integrase

Barreca, Maria Letizia, De Luca, Laura, Iraci, Nunzio, Chimirri, Alba

Journal:

Journal of Medicinal Chemistry

Year:

2006

Language:

english

File:

PDF, 290 KB

english, 2006

141

3,5-Dihydro-4 H -2,3-benzodiazepine-4-thiones: A New Class of AMPA Receptor Antagonists

Chimirri, Alba, De Sarro, Giovambattista, De Sarro, Angela, Gitto, Rosaria, Quartarone, Silvana, Zappalà, Maria, Constanti, Andrew, Libri, Vincenzo

Journal:

Journal of Medicinal Chemistry

Year:

1998

Language:

english

File:

PDF, 221 KB

english, 1998

142

Design and synthesis of N1-aryl-benzimidazoles 2-substituted as novel HIV-1 non-nucleoside reverse transcriptase inhibitors

Monforte, Anna-Maria, Ferro, Stefania, De Luca, Laura, Lo Surdo, Giuseppa, Morreale, Francesca, Pannecouque, Christophe, Balzarini, Jan, Chimirri, Alba

Journal:

Bioorganic & Medicinal Chemistry

Year:

2014

Language:

english

File:

PDF, 540 KB

english, 2014

143

Diketoacid chelating ligands as dual inhibitors of HIV-1 integration process

Rogolino, Dominga, Carcelli, Mauro, Compari, Carlotta, De Luca, Laura, Ferro, Stefania, Fisicaro, Emilia, Rispoli, Gabriele, Neamati, Nouri, Debyser, Zeger, Christ, Frauke, Chimirri, Alba

Journal:

European Journal of Medicinal Chemistry

Year:

2014

Language:

english

File:

PDF, 210 KB

english, 2014

144

Structure-based screening for the discovery of new carbonic anhydrase VII inhibitors

De Luca, Laura, Ferro, Stefania, Damiano, Francesca M., Supuran, Claudiu T., Vullo, Daniela, Chimirri, Alba, Gitto, Rosaria

Journal:

European Journal of Medicinal Chemistry

Year:

2014

Language:

english

File:

PDF, 1.41 MB

english, 2014

145

Synthesis, modelling and biological characterization of 3-substituted-1H-indoles as ligands of GluN2B-containing N-methyl-d-aspartate receptors

Gitto, Rosaria, De Luca, Laura, Ferro, Stefania, Russo, Emilio, De Sarro, Giovambattista, Chisari, Mariangela, Ciranna, Lucia, Alvarez-Builla, Julio, Alajarin, Ramon, Buemi, Maria Rosa, Chimirri, Alba

Journal:

Bioorganic & Medicinal Chemistry

Year:

2014

Language:

english

File:

PDF, 892 KB

english, 2014

146

From NMDA receptor antagonists to discovery of selective σ2 receptor ligands

Gitto, Rosaria, De Luca, Laura, Ferro, Stefania, Scala, Angela, Ronsisvalle, Simone, Parenti, Carmela, Prezzavento, Orazio, Buemi, Maria Rosa, Chimirri, Alba

Journal:

Bioorganic & Medicinal Chemistry

Year:

2014

Language:

english

File:

PDF, 577 KB

english, 2014

147

A new potential approach to block HIV-1 replication via protein–protein interaction and strand-transfer inhibition

Ferro, Stefania, De Luca, Laura, Lo Surdo, Giuseppa, Morreale, Francesca, Christ, Frauke, Debyser, Zeger, Gitto, Rosaria, Chimirri, Alba

Journal:

Bioorganic & Medicinal Chemistry

Year:

2014

Language:

english

File:

PDF, 844 KB

english, 2014

148

Anticonvulsant activity of newly synthesized thiazolobenzodiazepines

Chimirri, A., De Sarro, G.B., Grasso, S., De Sarro, A.

Journal:

Pharmacological Research

Year:

1990

Language:

english

File:

PDF, 60 KB

english, 1990

149

Lamotrigine positively affects the development of psychiatric comorbidity in epileptic animals, while psychiatric comorbidity aggravates seizures

Russo, Emilio, Chimirri, Serafina, Aiello, Rossana, De Fazio, Salvatore, Leo, Antonio, Rispoli, Vincenzo, Marra, Rosario, Labate, Angelo, De Fazio, Pasquale, Citraro, Rita, De Sarro, Giovambattista

Journal:

Epilepsy & Behavior

Year:

2013

Language:

english

File:

PDF, 793 KB

english, 2013

150

Protective effects of some statins on epileptogenesis and depressive-like behavior in WAG/Rij rats, a genetic animal model of absence epilepsy

Citraro, Rita, Chimirri, Serafina, Aiello, Rossana, Gallelli, Luca, Trimboli, Francesca, Britti, Domenico, De Sarro, Giovambattista, Russo, Emilio

Journal:

Year:

2014

Language:

english

File:

PDF, 417 KB

english, 2014