D.H Caignard: search on Z-Library

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51

3-Benzo[b]furyl- and 3-benzo[b]thienylaminobutyric acids as GABAB ligands. Synthesis and structure-activity relationship studies

M Ansar, S Al Akoum Ebriki, R Mouhoub, P Berthelot, C Vaccher, MP Vaccher, N Flouquet, DH Caignard, P Renard, B Pirard, MC Rettori, G Evrard, F Durant, M Debaert

Journal:

European Journal of Medicinal Chemistry

Year:

1996

Language:

english

File:

PDF, 967 KB

english, 1996

52

Synthesis and evaluation of new 2-piperazinylbenzothiazoles with high 5-HT1A and 5-HT3 affinities

O Diouf, P Depreux, D Lesieur, JH Poupaert, DH Caignard

Journal:

European Journal of Medicinal Chemistry

Year:

1995

Language:

english

File:

PDF, 447 KB

english, 1995

53

Synthesis and biological evaluation of benzimidazole derivatives as potent AMP-activated protein kinase activators

Julie Charton, Sophie Girault-Mizzi, Marie-Ange Debreu-Fontaine, Fabienne Foufelle, Isabelle Hainault, Jean-Guy Bizot-Espiard, Daniel-Henri Caignard, Christian Sergheraert

Journal:

Bioorganic & Medicinal Chemistry

Year:

2006

Language:

english

File:

PDF, 436 KB

english, 2006

54

Synthesis and biological activity of conformationally restricted tricyclic analogs of the hormone melatonin

V. Leclerc, P. Depreux, D. Lesieur, D.H. Caignard, P. Renard, P. Delagrange, B. Guardiola-Lemaitre, P. Morgan

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1996

Language:

english

File:

PDF, 248 KB

english, 1996

55

N-substituted aminohydroxypyridines as potential non-opioid analgesic agents

M.C. Viaud, P. Jamoneau, J.G. Bizot-Espiard, B. Pfeiffer, P. Renard, D.H. Caignard, G. Adam, G. Guillaumet

Journal:

Bioorganic & Medicinal Chemistry

Year:

1995

Language:

english

File:

PDF, 794 KB

english, 1995

56

Design and synthesis of novel imidazoline derivatives with potent antihyperglycemic activity in a rat model of type 2 diabetes

Louis Crane, Maria Anastassiadou, Salomé El Hage, Jean Luc Stigliani, Geneviève Baziard-Mouysset, Marc Payard, Jean Michel Leger, Jean-Guy Bizot-Espiard, Alain Ktorza, Daniel-Henri Caignard, Pierre Re

Journal:

Bioorganic & Medicinal Chemistry

Year:

2006

Language:

english

File:

PDF, 365 KB

english, 2006

57

Novel 1,3-dicarbonyl compounds having 2(3H)-benzazolonic heterocycles as PPARγ agonists

Elodie Blanc-Delmas, Nicolas Lebegue, Valérie Wallez, Véronique Leclerc, Saïd Yous, Pascal Carato, Amaury Farce, Caroline Bennejean, Pierre Renard, Daniel-Henri Caignard, Valérie Audinot-Bouchez, Pasc

Journal:

Bioorganic & Medicinal Chemistry

Year:

2006

Language:

english

File:

PDF, 421 KB

english, 2006

58

Novel 5-azaindolocarbazoles as cytotoxic agents and Chk1 inhibitors

Myriam Lefoix, Gérard Coudert, Sylvain Routier, Bruno Pfeiffer, Daniel-Henri Caignard, John Hickman, Alain Pierré, Roy M. Golsteyn, Stéphane Léonce, Céline Bossard, Jean-Yves Mérour

Journal:

Bioorganic & Medicinal Chemistry

Year:

2008

Language:

english

File:

PDF, 349 KB

english, 2008

59

Design and synthesis of benzofuranic derivatives as new ligands at the melatonin-binding site MT3

Mohamed Ettaoussi, Basile Péres, Fréderique Klupsch, Philippe Delagrange, Jean-A. Boutin, Pierre Renard, Daniel-H. Caignard, Philippe Chavatte, Pascal Berthelot, Daniel Lesieur, Saïd Yous

Journal:

Bioorganic & Medicinal Chemistry

Year:

2008

Language:

english

File:

PDF, 188 KB

english, 2008

60

Synthesis of 3-phenylnaphthalenic derivatives as new selective MT2 melatoninergic ligands

Sophie Poissonnier-Durieux, Mohamed Ettaoussi, Basile Pérès, Jean A. Boutin, Valérie Audinot, Caroline Bennejean, Philippe Delagrange, Daniel Henri Caignard, Pierre Renard, Pascal Berthelot, Daniel Le

Journal:

Bioorganic & Medicinal Chemistry

Year:

2008

Language:

english

File:

PDF, 253 KB

english, 2008

61

Synthesis and pharmacological evaluation of a second generation of pyridothiadiazine 1,1-dioxides acting as AMPA potentiators

Pierre Francotte, Pascal de Tullio, Tchao Podona, Ousmane Diouf, Pierre Fraikin, Pierre Lestage, Laurence Danober, Jean-Yves Thomas, Daniel-Henri Caignard, Bernard Pirotte

Journal:

Bioorganic & Medicinal Chemistry

Year:

2008

Language:

english

File:

PDF, 382 KB

english, 2008

62

Design and synthesis of 3-phenyltetrahydronaphthalenic derivatives as new selective MT2 melatoninergic ligands. Part II

Sophie Durieux, Angéline Chanu, Christophe Bochu, Valérie Audinot, Sophie Coumailleau, Jean A. Boutin, Philippe Delagrange, Daniel H. Caignard, Caroline Bennejean, Pierre Renard, Daniel Lesieur, Pasca

Journal:

Bioorganic & Medicinal Chemistry

Year:

2009

Language:

english

File:

PDF, 380 KB

english, 2009

63

Synthesis of new carbo- and heterocyclic analogues of 8-HETE and evaluation of their activity towards the PPARs

Frédéric Caijo, Paul Mosset, René Grée, Valérie Audinot-Bouchez, Jean Boutin, Pierre Renard, Daniel-Henri Caignard, Catherine Dacquet

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2005

Language:

english

File:

PDF, 147 KB

english, 2005

64

Studies towards the conception of new selective PPARβ/δ ligands

Carine Ekambomé Basséne, Franck Suzenet, Nathalie Hennuyer, Bart Staels, Daniel-Henri Caignard, Catherine Dacquet, Pierre Renard, Gérald Guillaumet

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2006

Language:

english

File:

PDF, 135 KB

english, 2006

65

4,4-Dimethyl-1,2,3,4-tetrahydroquinoline-based PPARα/γ agonists. Part I: Synthesis and pharmacological evaluation

Cécile Parmenon, Jérôme Guillard, Daniel-Henri Caignard, Nathalie Hennuyer, Bart Staels, Valérie Audinot-Bouchez, Jean-Albert Boutin, Catherine Dacquet, Alain Ktorza, Marie-Claude Viaud-Massuard

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2008

Language:

english

File:

PDF, 182 KB

english, 2008

66

Synthesis and biological evaluation of novel benzodioxinocarbazoles (BDCZs) as potential anticancer agents

Nathalie Ayerbe, Sylvain Routier, Isabelle Gillaizeau, Carmen Maiereanu, Daniel-Henry Caignard, Alain Pierré, Stéphane Léonce, Gérard Coudert

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2010

Language:

english

File:

PDF, 1.56 MB

english, 2010

67

Design and synthesis of 1-(2-alkanamidoethyl)-6-methoxy-7-azaindole derivatives as potent melatonin agonists

Matthieu Jeanty, Franck Suzenet, Philippe Delagrange, Olivier Nosjean, Jean A. Boutin, Daniel H. Caignard, Gérald Guillaumet

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2011

Language:

english

File:

PDF, 627 KB

english, 2011

68

Synthesis of potential Rho-kinase inhibitors based on the chemistry of an original heterocycle: 4,4-Dimethyl-3,4-dihydro-1H-quinolin-2-one

Marie-Anne Letellier, Jérôme Guillard, Daniel-Henri Caignard, Gilles Ferry, Jean A. Boutin, Marie-Claude Viaud-Massuard

Journal:

European Journal of Medicinal Chemistry

Year:

2008

Language:

english

File:

PDF, 355 KB

english, 2008

69

Design and synthesis of naphthalenic derivatives as new ligands at the melatonin binding site MT3

Véronique Leclerc, Mohamed Ettaoussi, Marouan Rami, Amaury Farce, Jean Albert Boutin, Philippe Delagrange, Daniel-Henri Caignard, Pierre Renard, Pascal Berthelot, Saïd Yous

Journal:

European Journal of Medicinal Chemistry

Year:

2011

Language:

english

File:

PDF, 309 KB

english, 2011

70

Preparation and pharmacological evaluation of a novel series of 2-(phenylthio)benzo[b]thiophenes as selective MT2 receptor ligands

Christophe Mésangeau, Mikaël Fraise, Philippe Delagrange, Daniel Henri Caignard, Jean Albert Boutin, Pascal Berthelot, Saïd Yous

Journal:

European Journal of Medicinal Chemistry

Year:

2011

Language:

english

File:

PDF, 243 KB

english, 2011

71

Preparative enantiomeric separation of potent AMP-activated protein kinase activator by HPLC on amylose-based chiral stationary phase: Determination of enantiomeric purity and assignment of absolute configuration

Marie-Pierre Vaccher, Julie Charton, Abdelhalim Guelzim, Daniel-Henry Caignard, Jean-Paul Bonte, Claude Vaccher

Journal:

Journal of Pharmaceutical and Biomedical Analysis

Year:

2008

Language:

english

File:

PDF, 547 KB

english, 2008

72

Synthesis of tetracyclic dioxygenated isoquinolines and their cytotoxic activity

Manel Romero, Daniel-Henry Caignard, Pierre Renard, M. Dolors Pujol

Journal:

Year:

2008

Language:

english

File:

PDF, 288 KB

english, 2008

73

Synthesis of isoquinolines and tetrahydroisoquinolines as potential antitumour agents

A.S Capilla, M Romero, M.D Pujol, D.H Caignard, P Renard

Journal:

Year:

2001

Language:

english

File:

PDF, 138 KB

english, 2001

74

Synthesis and biological evaluation of 7-azaindolocarbazoles

Sylvain Routier, Nathalie Ayerbe, Jean-Yves Mérour, Gérard Coudert, Christian Bailly, Alain Pierré, Bruno Pfeiffer, Daniel-Henri Caignard, Pierre Renard

Journal:

Year:

2002

Language:

english

File:

PDF, 218 KB

english, 2002

75

An efficient method for the preparation of antitumoral α-keto-imines benzyldihydroisoquinolines by selective benzylic oxidation with C/Pd in acetonitrile

Inmaculada Andreu, Nuria Cabedo, Ghanem Atassi, Alain Pierre, Daniel H Caignard, Pierre Renard, Diego Cortes, Almudena Bermejo

Journal:

Tetrahedron Letters

Year:

2002

Language:

english

File:

PDF, 99 KB

english, 2002

76

First synthesis of symmetrical and non-symmetrical aza indolocarbazoles derivatives

Sylvain Routier, Gérard Coudert, Jean-Yves Mérour, Daniel Henri Caignard

Journal:

Tetrahedron Letters

Year:

2002

Language:

english

File:

PDF, 157 KB

english, 2002

77

The host—tumor immune conflict: from immunosuppression to resistance and destruction

Salem Chouaib, Carine Asselin-Paturel, Fathia Mami-Chouaib, Anne Caignard, Jean Yves Blay

Journal:

Immunology Today

Year:

1997

Language:

english

File:

PDF, 699 KB

english, 1997

78

Synthesis and structure–activity relationships of novel arylalkyl 4-benzyl piperazine derivatives as σ site selective ligands

Salomé Younes, Youssef Labssita, Geneviève Baziard-Mouysset, Marc Payard, Marie-Claire Rettori, Pierre Renard, Bruno Pfeiffer, Daniel-Henri Caignard

Journal:

European Journal of Medicinal Chemistry

Year:

2000

Language:

english

File:

PDF, 160 KB

english, 2000

79

Antitumor agents. Synthesis and biological evaluation of new compounds related to podophyllotoxin, containing the 2,3-dihydro-1,4-benzodioxin system

Alfons Sergi Capilla, Isabel Sánchez, Daniel H. Caignard, Pierre Renard, Maria Dolors Pujol

Journal:

European Journal of Medicinal Chemistry

Year:

2001

Language:

english

File:

PDF, 159 KB

english, 2001

80

6-Amino-2,4-lutidine carboxamides: α-aminoamide derivatives as systemic and topical inflammation inhibitors

Muriel Duflos, Jacqueline Courant, Guillaume Le Baut, Nicole Grimaud, Pierre Renard, Dominique Manechez, Daniel-Henri Caignard

Journal:

European Journal of Medicinal Chemistry

Year:

1998

Language:

english

File:

PDF, 1.02 MB

english, 1998

81

Synthesis and anti-inflammatory activity of N-(aza)arylcarboxamides derived from Trolox®

Claudie Moulin, Muriel Duflos, Guillaume Le Baut, Nicole Grimaud, Pierre Renard, Daniel-Henri Caignard

Journal:

European Journal of Medicinal Chemistry

Year:

1998

Language:

english

File:

PDF, 638 KB

english, 1998

82

Synthesis and pharmacological evaluation of novel 4-(4-fluorobenzoyl)piperidine derivatives as mixed 5-HT1A/5-HT2A/D2 receptor ligands

Ousmane Diouf, Pascal Carato, Isabelle Lesieur, Marie Claire Rettori, Daniel Henri Caignard

Journal:

European Journal of Medicinal Chemistry

Year:

1999

Language:

english

File:

PDF, 72 KB

english, 1999

83

Novel antitumor artemisinin derivatives targeting G1 phase of the cell cycle

Ying Li, Feng Shan, Jin-Ming Wu, Guang-Shao Wu, Jian Ding, Dong Xiao, Wei-Yi Yang, Ghanem Atassi, Stéphane Léonce, Daniel-Henri Caignard, Pierre Renard

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 177 KB

english, 2001

84

5-HT1A and 5-HT2A ligands with anxiolytic and antipanic-like properties

O. Diouf, P. Carato, P. Depreux, J.P. Bonte, D.H. Caignard, B. Guardiola-Lemaître, M.C. Rettori, C. Belzung, Daniel Lesieur

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1997

Language:

english

File:

PDF, 298 KB

english, 1997

85

Synthesis and pharmacological evaluation of imidazoline sites I1 and I2 selective ligands

Maria Anastassiadou, Saı̈da Danoun, Louis Crane, Geneviève Baziard-Mouysset *, Marc Payard *, Daniel-Henri Caignard, Marie-Claire Rettori, Pierre Renard

Journal:

Bioorganic & Medicinal Chemistry

Year:

2001

Language:

english

File:

PDF, 195 KB

english, 2001

86

Synthesis and cytotoxicity of dihydroartemisinin ethers containing cyanoarylmethyl group

Ying Li, Jin-Ming Wu, Feng Shan, Guang-Shao Wu, Jian Ding, Dong Xiao, Jia-Xian Han, Ghanem Atassi, Stéphane Leonce, Daniel-Henri Caignard, Pierre Renard

Journal:

Bioorganic & Medicinal Chemistry

Year:

2003

Language:

english

File:

PDF, 225 KB

english, 2003

87

Substituted pyrido[3,2-b]oxazin-3(4H)-ones: synthesis and evaluation of antinociceptive activity

L. Savelon, J.G. Bizot-Espiard, D.H. Caignard, B. Pfeiffer, P. Renard, M.C. Viaud, G. Guillaumet

Journal:

Bioorganic & Medicinal Chemistry

Year:

1998

Language:

english

File:

PDF, 216 KB

english, 1998

88

6-Aminoalkyloxazolo[4,5-b]pyridin-2(3H)-ones: Synthesis and Evaluation of Antinoceptive Activity

L. Savelon, J.G. Bizot-Espiard, D.H. Caignard, B. Pfeiffer, P. Renard, M.C. Viaud, G. Guillaumet

Journal:

Bioorganic & Medicinal Chemistry

Year:

1998

Language:

english

File:

PDF, 256 KB

english, 1998

89

Synthesis and structure–activity relationships of novel naphthalenic and bioisosteric related amidic derivatives as melatonin receptor ligands

Véronique Leclerc, Eric Fourmaintraux, Patrick Depreux, Daniel Lesieur, Peter Morgan, H.Edward Howell, Pierre Renard, Daniel-Henri Caignard, Bruno Pfeiffer, Philippe Delagrange, Béatrice Guardiola-Lem

Journal:

Bioorganic & Medicinal Chemistry

Year:

1998

Language:

english

File:

PDF, 253 KB

english, 1998

90

Tumor escape from killing: Role of killer inhibitory receptors and acquisition of tumor resistance to cell death

S. Chouaib, J. Thiery, A. Gati, N. Guerra, M. El Behi, G. Dorothée, F. Mami-Chouaib, D. Bellet, A. Caignard

Journal:

Tissue Antigens

Year:

2002

Language:

english

File:

PDF, 356 KB

english, 2002

91

Cytofluorescence localization of adriamycin in resistant colon cancer cells

Bruno Chauffert, François Martin, Anne Caignard, Jean-François Jeannin, Annick Leclerc

Journal:

Cancer Chemotherapy and Pharmacology

Year:

1984

Language:

english

File:

PDF, 502 KB

english, 1984

92

Histological reactivity of a monoclonal antibody against rat colon cancer cells on human and rat normal gut and colonic tumours

P. Genne, N. -O. Olsson, A. Caignard, R. Oriol, J. Bara, A. Hammann, F. Martin

Journal:

Virchows Archiv

Year:

1992

Language:

english

File:

PDF, 3.47 MB

english, 1992

93

Novel 2(3H)-Benzothiazolones as Highly Potent and Selective Sigma-1 Receptor Ligands

Saïd Yous, Valérie Wallez, Mirabelle Belloir, Daniel H. Caignard, Christopher R. McCurdy, Jacques H. Poupaert

Journal:

Medicinal Chemistry Research

Year:

2005

File:

PDF, 335 KB

2005

94

Effect of indomethacin on the growth of colon cancer cells in syngeneic rats

Nils O. Olsson, Anne Caignard, Monique S. Martin, François Martin

Journal:

International Journal of Immunopharmacology

Year:

1984

Language:

english

File:

PDF, 469 KB

english, 1984

95

Synthesis and cytotoxicity of artemisinin derivatives containing cyanoarylmethyl group

Jin-Ming Wu, Feng Shan, Guang-Shao Wu, Ying Li, Jian Ding, Dong Xiao, Jia-Xian Han, Ghanem Atassi, Stéphane Leonce, Daniel-Henri Caignard, Pierre Renard

Journal:

European Journal of Medicinal Chemistry

Year:

2001

Language:

english

File:

PDF, 147 KB

english, 2001

96

Synthesis and structure-activity relationships of novel 2-amino alkyl chromones and related derivatives as a site-selective ligands

Geneviève Baziard-Mouysset, Salouma Younes, Youssef Labssita, Marc Payard, Daniel-Henri Caignard, Marie-Claire Rettori, Pierre Renard, Bruno Pfeiffer, Béatrice Guardiola-Lemaitre

Journal:

European Journal of Medicinal Chemistry

Year:

1998

Language:

english

File:

PDF, 837 KB

english, 1998

97

Activated K-ras in Tumorigenic and Non-tumorigenic Cell Variants from a Rat Colon Adenocarcinoma, Induced by Dimethylhydrazine

Anne Caignard, Yoshinori Kitagawa, Shigeaki Sato, Minako Nagao

Journal:

Year:

1988

File:

PDF, 293 KB

1988

98

Effects of cimetidine and indomethacin on the growth of dimethylhydrazine-induced or transplanted intestinal cancers in the rat

Caignard, A, Martin, M, Reisser, D, Thomas, B, Martin, F

Journal:

British Journal of Cancer

Year:

1984

Language:

english

File:

PDF, 693 KB

english, 1984

99

Plasminogen receptors on rat colon carcinoma cells

Durliat, M, Komano, O, Correc, P, Bertrand, O, Cochet, S, Caignard, A, Martin, F, Burtin, P

Journal:

British Journal of Cancer

Year:

1992

Language:

english

File:

PDF, 1.39 MB

english, 1992

100

Mutations of the von Hippel–Lindau gene confer increased susceptibility to natural killer cells of clear-cell renal cell carcinoma

Perier, A, Fregni, G, Wittnebel, S, Gad, S, Allard, M, Gervois, N, Escudier, B, Azzarone, B, Caignard, A

Journal:

Year:

2011

Language:

english

File:

PDF, 855 KB

english, 2011