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1

PDE5 inhibitors: An original access to novel potent arylated analogues of tadalafil

Terence Beghyn, Candide Hounsou, Benoit P. Deprez

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2007

Language:

english

File:

PDF, 150 KB

english, 2007

2

Racemic and diastereoselective construction of indole alkaloids under solvent- and catalyst-free microwave-assisted Pictet–Spengler condensation

Jida, Mouhamad, Soueidan, Olivier-Mohamad, Deprez, Benoit, Laconde, Guillaume, Deprez-Poulain, Rebecca

Journal:

Green Chemistry

Year:

2012

Language:

english

File:

PDF, 543 KB

english, 2012

3

Identification of novel TACE inhibitors compatible with topical application

Ouvry, Gilles, Berton, Yaël, Bhurruth-Alcor, Yushma, Bonnary, Laetitia, Bouix-Peter, Claire, Bouquet, Karine, Bourotte, Marilyne, Chambon, Sandrine, Comino, Catherine, Deprez, Benoît, Duvert, Denis, D

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2017

Language:

english

File:

PDF, 638 KB

english, 2017

4

The use or generation of biomedical data and existing medicines to discover and establish new treatments for patients with rare diseases – recommendations of the IRDiRC Data Mining and Repurposing Task Force

Southall, Noel T, Natarajan, Madhusudan, Lau, Lilian Pek Lian, Jonker, Anneliene Hechtelt, Deprez, Benoît, Guilliams, Tim, Hunter, Lawrence, Rademaker, Carin MA, Hivert, Virginie, Ardigò, Diego

Journal:

Orphanet Journal of Rare Diseases

Year:

2019

File:

PDF, 569 KB

2019

5

Kinetic Target-Guided Synthesis: reaching the age of maturity.

Bosc, Damien, Camberlein, Virgyl, Gealageas, Ronan, Castillo-Aguilera, Omar, Deprez, Benoit, Deprez-Poulain, Rebecca

Journal:

Journal of Medicinal Chemistry

Year:

2019

File:

PDF, 2.06 MB

2019

6

ChemInform Abstract: Combinatorial Chemistry: A Rational Access to Molecular Diversity

Patricia Melnyk, Line Bourel, Xavier Williard, Iuliana Pop, Dragos Horvath, Benoit Deprez, Andre Tartar

Journal:

Year:

1999

File:

PDF, 25 KB

1999

7

ChemInform Abstract: Automated Parallel Synthesis of a Tetrahydroisoquinolin-Based Library: Potential Prolyl Endopeptidase Inhibitors.

Sandrine Vendeville, Line Bourel, Elisabeth Davioud-Charvet, Philippe Grellier, Benoit Deprez, Christian Sergheraert

Journal:

Year:

1999

File:

PDF, 29 KB

1999

8

ChemInform Abstract: Parallel Synthesis of 1,2,4-Oxadiazoles from Carboxylic Acids Using an Improved, Uronium-Based, Activation.

Rebecca F. Poulain, Andre L. Tartar, Benoit P. Deprez

Journal:

Year:

2001

File:

PDF, 28 KB

2001

9

Efficient, Protection-Free Suzuki—Miyaura Synthesis of ortho-Biphenyltetrazoles.

Nicolas Cousaert, Patrick Toto, Nicolas Willand, Benoit Deprez

Journal:

Year:

2005

File:

PDF, 18 KB

2005

10

ChemInform Abstract: Solvent-Free Microwave-Assisted Meyers′ Lactamization.

Mouhamad Jida, Rebecca Deprez-Poulain, Sandra Malaquin, Pascal Roussel, Francine Agbossou-Niedercorn, Benoit Deprez, Guillaume Laconde

Journal:

Year:

2010

File:

PDF, 44 KB

2010

11

ChemInform Abstract: Synthesis of Five- and Six-Membered Lactams via Solvent-Free Microwave Ugi Reaction.

Mouhamad Jida, Sandra Malaquin, Rebecca Deprez-Poulain, Guillaume Laconde, Benoit Deprez

Journal:

Year:

2011

File:

PDF, 30 KB

2011

12

ChemInform Abstract: A Facile and Rapid Synthesis of N-Benzyl-2-substituted Piperazines.

Mouhamad Jida, Mohamad Soueidan, Nicolas Willand, Francine Agbossou-Niedercorn, Lydie Pelinski, Guillaume Laconde, Rebecca Deprez-Poulain, Benoit Deprez

Journal:

Year:

2011

File:

PDF, 27 KB

2011

13

ChemInform Abstract: Application of Ullmann and Ullmann—Finkelstein Reactions for the Synthesis of N-Aryl-N-(1H-pyrazol-3-yl)acetamide or N-(1-Aryl-1H-pyrazol-3-yl)acetamide Derivatives and Pharmacological Evaluation.

Rebecca Deprez-Poulain, Nicolas Cousaert, Patrick Toto, Nicolas Willand, Benoit Deprez

Journal:

Year:

2012

File:

PDF, 45 KB

2012

14

A library of novel hydroxamic acids targeting the metallo-protease family: Design, parallel synthesis and screening

Marion Flipo, Terence Beghyn, Julie Charton, Virginie A. Leroux, Benoit P. Deprez, Rebecca F. Deprez-Poulain

Journal:

Bioorganic & Medicinal Chemistry

Year:

2007

Language:

english

File:

PDF, 281 KB

english, 2007

15

Synthesis of a 200-member library of squaric acid N-hydroxylamide amides

Julie Charton, Benoît P. Déprez, Rébecca F. Déprez-Poulain

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2008

Language:

english

File:

PDF, 274 KB

english, 2008

16

Corrigendum to “Synthesis of a 200-member library of squaric acid N-hydroxylamide amides” [Bioorg. Med. Chem. Lett. 18 (2008) 4968–4971]

Julie Charton, Florence Leroux, Sylvain Delaroche, Valérie Landry, Benoît P. Déprez, Rébecca F. Déprez-Poulain

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2009

Language:

english

File:

PDF, 103 KB

english, 2009

17

Novel non-carboxylic acid retinoids: 1,2,4-Oxadiazol-5-one derivatives

Julie Charton, Rebecca Deprez-Poulain, Nathalie Hennuyer, Anne Tailleux, Bart Staels, Benoit Deprez

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2009

Language:

english

File:

PDF, 182 KB

english, 2009

18

New non-hydroxamic ADAMTS-5 inhibitors based on the 1,2,4-triazole-3-thiol scaffold

Lucie Maingot, Florence Leroux, Valérie Landry, Julie Dumont, Hideaki Nagase, Bruno Villoutreix, Olivier Sperandio, Rebecca Deprez-Poulain, Benoit Deprez

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2010

Language:

english

File:

PDF, 550 KB

english, 2010

19

Synthesis and structural studies of a novel scaffold for drug discovery: a 4,5-dihydro-3H-spiro[1,5-benzoxazepine-2,4′-piperidine]

Nicolas Willand, Terence Beghyn, Guy Nowogrocki, Jean-Claude Gesquiere, Benoit Deprez

Journal:

Tetrahedron Letters

Year:

2004

Language:

english

File:

PDF, 257 KB

english, 2004

20

A simple reaction to produce small structurally complex and diverse molecules

Rebecca Deprez-Poulain, Nicolas Willand, Christophe Boutillon, Guy Nowogrocki, Nathalie Azaroual, Benoit Deprez

Journal:

Tetrahedron Letters

Year:

2004

Language:

english

File:

PDF, 264 KB

english, 2004

21

Efficient, protection-free Suzuki–Miyaura synthesis of ortho-biphenyltetrazoles

Nicolas Cousaert, Patrick Toto, Nicolas Willand, Benoît Deprez

Journal:

Tetrahedron Letters

Year:

2005

Language:

english

File:

PDF, 121 KB

english, 2005

22

Synthesis of N-(iodophenyl)-amides via an unprecedented Ullmann–Finkelstein tandem reaction

Patrick Toto, Jean-Claude Gesquière, Benoit Deprez, Nicolas Willand

Journal:

Tetrahedron Letters

Year:

2006

Language:

english

File:

PDF, 136 KB

english, 2006

23

UFU (‘Ullmann–Finkelstein–Ullmann’): a new multicomponent reaction

Patrick Toto, Jean-Claude Gesquière, Nicolas Cousaert, Benoit Deprez, Nicolas Willand

Journal:

Tetrahedron Letters

Year:

2006

Language:

english

File:

PDF, 146 KB

english, 2006

24

A versatile solid-phase synthesis of 3-aryl-1,2,4-oxadiazolones and analogues

Julie Charton, Nicolas Cousaert, Christophe Bochu, Nicolas Willand, Benoît Déprez, Rébecca Déprez-Poulain

Journal:

Tetrahedron Letters

Year:

2007

Language:

english

File:

PDF, 149 KB

english, 2007

25

Efficient, two-step synthesis of N-substituted nortropinone derivatives

Nicolas Willand, Benoit Folléas, Christophe Boutillon, Liesbeth Verbraeken, Jean-Claude Gesquière, André Tartar, Benoit Deprez

Journal:

Tetrahedron Letters

Year:

2007

Language:

english

File:

PDF, 207 KB

english, 2007

26

Convenient synthesis of 4H-1,2,4-triazole-3-thiols using di-2-pyridylthionocarbonate

Rebecca F. Deprez-Poulain, Julie Charton, Virginie Leroux, Benoit P. Deprez

Journal:

Tetrahedron Letters

Year:

2007

Language:

english

File:

PDF, 162 KB

english, 2007

27

Original loading and Suzuki conditions for the solid-phase synthesis of biphenyltetrazoles. Application to the first solid-phase synthesis of irbesartan

Nicolas Cousaert, Nicolas Willand, Jean-Claude Gesquière, André Tartar, Benoît Déprez, Rebecca Deprez-Poulain

Journal:

Tetrahedron Letters

Year:

2008

Language:

english

File:

PDF, 132 KB

english, 2008

28

Ugi reaction for the synthesis of 4-aminopiperidine-4-carboxylic acid derivatives. Application to the synthesis of carfentanil and remifentanil

Sandra Malaquin, Mouhamad Jida, Jean-Claude Gesquiere, Rebecca Deprez-Poulain, Benoit Deprez, Guillaume Laconde

Journal:

Tetrahedron Letters

Year:

2010

Language:

english

File:

PDF, 429 KB

english, 2010

29

Synthesis of five- and six-membered lactams via solvent-free microwave Ugi reaction

Mouhamad Jida, Sandra Malaquin, Rebecca Deprez-Poulain, Guillaume Laconde, Benoit Deprez

Journal:

Tetrahedron Letters

Year:

2010

Language:

english

File:

PDF, 285 KB

english, 2010

30

A facile and rapid synthesis of N-benzyl-2-substituted piperazines

Mouhamad Jida, Mohamad Soueidan, Nicolas Willand, Francine Agbossou-Niedercorn, Lydie Pelinski, Guillaume Laconde, Rebecca Deprez-Poulain, Benoit Deprez

Journal:

Tetrahedron Letters

Year:

2011

Language:

english

File:

PDF, 1.12 MB

english, 2011

31

Lewis acid-induced reaction of homophthalic anhydride with imines: a convenient synthesis of trans-isoquinolonic acids

Niefang Yu, Line Bourel, Benoit Deprez, Jean-Claude Gesquiere

Journal:

Tetrahedron Letters

Year:

1998

Language:

english

File:

PDF, 215 KB

english, 1998

32

Discovery of Thioazepinone Ligands for Src SH2: From Non-specific to Specific Binding

Dominique Lesuisse, Pierre Deprez, Eva Albert, Tran Thien Duc, Benoit Sortais, Dominique Gofflo, Véronique Jean-Baptiste, Jean-Pierre Marquette, Bernard Schoot, Edoardo Sarubbi, Gudrun Lange, Pierre B

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 465 KB

english, 2001

33

Automated parallel synthesis of a tetrahydroisoquinolin-based library: Potential prolyl endopeptidase inhibitors

Sandrine Vendeville, Line Bourel, Elisabeth Davioud-Charvet, Philippe Grellier, Benoît Deprez, Christian Sergheraert

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1999

Language:

english

File:

PDF, 375 KB

english, 1999

34

Loss of Left Ventricular Epicardial Lead Capture Due to Pneumothorax

DOMINIQUE BLOMMAERT, FRÉDÉRIC DEPREZ, PHILIPPE EUCHER, ISABELLE MANCINI, JOSEPH MUCUMBITSI, BENOÎT COLLET, LUC DE ROY

Journal:

Pacing and Clinical Electrophysiology

Year:

2002

Language:

english

File:

PDF, 162 KB

english, 2002

35

A 36-year-old man with sudden severe headache

Paolo Simoni, Benoît Meunier, Manuel Deprez, Tudor Racaru, Didier Martin

Journal:

Skeletal Radiology

Year:

2011

Language:

english

File:

PDF, 131 KB

english, 2011

36

36-year-old man with sudden severe headache

Paolo Simoni, Benoît Meunier, Manuel Deprez, Tudor Racaru, Didier Martin

Journal:

Skeletal Radiology

Year:

2011

Language:

english

File:

PDF, 164 KB

english, 2011

37

Monitoring of a three-step solid phase synthesis involving a Heck reaction using magic angle spinning NMR spectroscopy

Iuliana E. Pop, Christophe F. Dhalluin, Benoît P. Déprez, Patricia C. Melnyk, Guy M. Lippens, AndréL. Tartar

Journal:

Year:

1996

Language:

english

File:

PDF, 620 KB

english, 1996

38

Parallel synthesis of polysubstituted tetrahydroquinolines

Romuald Baudelle, Patricia Melnyk, Benoît Déprez, André Tartar

Journal:

Year:

1998

Language:

english

File:

PDF, 641 KB

english, 1998

39

Expression of Hoxa2 in cells entering chondrogenesis impairs overall cartilage development

Laurent Massip, Fabien Ectors, Pierre Deprez, Mehdi Maleki, Catherine Behets, Benoît Lengelé, Philippe Delahaut, Jacques Picard, René Rezsöhazy

Journal:

Differentiation

Year:

2007

Language:

english

File:

PDF, 2.68 MB

english, 2007

40

Natural Compounds: Leads or Ideas? Bioinspired Molecules for Drug Discovery

Terence Beghyn, Rebecca Deprez-Poulain, Nicolas Willand, Benoit Folleas, Benoit Deprez

Journal:

Chemical Biology & Drug Design

Year:

2008

Language:

english

File:

PDF, 1.07 MB

english, 2008

41

Friedländer synthesis of polysubstituted quinolines and naphthyridines promoted by propylphosphonic anhydride (T3P®) under mild conditions

Jida, Mouhamad, Deprez, Benoit

Journal:

New Journal of Chemistry

Year:

2012

Language:

english

File:

PDF, 817 KB

english, 2012

42

Drug-to-Genome-to-Drug, Step 2: Reversing Selectivity in a Series of Antiplasmodial Compounds

Beghyn, Terence B., Charton, Julie, Leroux, Florence, Henninot, Antoine, Reboule, Irena, Cos, Paul, Maes, Louis, Deprez, Benoit

Journal:

Journal of Medicinal Chemistry

Year:

2012

Language:

english

File:

PDF, 682 KB

english, 2012

43

Versatile Acylation of N-Nucleophiles Using a New Polymer-Supported 1-Hydroxybenzotriazole Derivative

Pop, Iuliana E., Déprez, Benoît P., Tartar, André L.

Journal:

Journal of Organic Chemistry

Year:

1997

Language:

english

File:

PDF, 346 KB

english, 1997

44

ChemInform Abstract: Squaric Acid Is a Suitable Building-Block in 4C-Ugi Reaction: Access to Original Bivalent Compounds.

Karen Aknin, Marion Gauriot, Jane Totobenazara, Noemie Deguine, Rebecca Deprez-Poulain, Benoit Deprez, Julie Charton

Journal:

Year:

2012

File:

PDF, 30 KB

2012

45

ChemInform Abstract: Racemic and Diastereoselective Construction of Indole Alkaloids under Solvent- and Catalyst-Free Microwave-Assisted Pictet—Spengler Condensation

Mouhamad Jida, Olivier-Mohamad Soueidan, Benoit Deprez, Guillaume Laconde, Rebecca Deprez-Poulain

Journal:

Year:

2012

File:

PDF, 44 KB

2012

46

ChemInform Abstract: Efficient Propylphosphonic Anhydride (®T3P) Mediated Synthesis of Benzothiazoles, Benzoxazoles and Benzimidazoles.

Xiaoan Wen, Jamal El Bakali, Rebecca Deprez-Poulain, Benoit Deprez

Journal:

Year:

2012

File:

PDF, 40 KB

2012

47

Subclassification of diffuse glioma tumours based on gene expression and allele copy number variation

Christophe Poulet, Benoit Hennuy, Pierre Robe, Manuel Deprez, Christian Herens, Vincent Bours

Journal:

Cancer Genetics and Cytogenetics

Year:

2010

Language:

english

File:

PDF, 36 KB

english, 2010

48

Application of Ullmann and Ullmann–Finkelstein reactions for the synthesis of N-aryl-N-(1H-pyrazol-3-yl) acetamide or N-(1-aryl-1H-pyrazol-3-yl) acetamide derivatives and pharmacological evaluation

Rebecca Deprez-Poulain, Nicolas Cousaert, Patrick Toto, Nicolas Willand, Benoit Deprez

Journal:

European Journal of Medicinal Chemistry

Year:

2011

Language:

english

File:

PDF, 566 KB

english, 2011

49

Tuberculosis: The drug development pipeline at a glance

Baptiste Villemagne, Céline Crauste, Marion Flipo, Alain R. Baulard, Benoit Déprez, Nicolas Willand

Journal:

European Journal of Medicinal Chemistry

Year:

2012

Language:

english

File:

PDF, 1.30 MB

english, 2012

50

Squaric acid is a suitable building-block in 4C-Ugi reaction: access to original bivalent compounds

Karen Aknin, Marion Gauriot, Jane Totobenazara, Noemie Deguine, Rebecca Deprez-Poulain, Benoit Deprez, Julie Charton

Journal:

Tetrahedron Letters

Year:

2012

Language:

english

File:

PDF, 1.93 MB

english, 2012