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51

(4-Carboxamido)phenylalanine is a surrogate for tyrosine in opioid receptor peptide ligands

Roland E. Dolle, Mathieu Machaut, Blanca Martinez-Teipel, Serge Belanger, Joel A. Cassel, Gabriel J. Stabley, Thomas M. Graczyk, Robert N. DeHaven

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2004

Language:

english

File:

PDF, 266 KB

english, 2004

52

Potent and highly selective kappa opioid receptor agonists incorporating chroman- and 2,3-dihydrobenzofuran-based constraints

Guo-Hua Chu, Minghua Gu, Joel A. Cassel, Serge Belanger, Thomas M. Graczyk, Robert N. DeHaven, Nathalie Conway-James, Mike Koblish, Patrick J. Little, Diane L. DeHaven-Hudkins, Roland E. Dolle

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2005

Language:

english

File:

PDF, 166 KB

english, 2005

53

Novel phenylamino acetamide derivatives as potent and selective κ opioid receptor agonists

Guo-Hua Chu, Minghua Gu, Joel A. Cassel, Serge Belanger, Gabriel. J. Stabley, Robert N. DeHaven, Nathalie Conway-James, Mike Koblish, Patrick J. Little, Diane L. DeHaven-Hudkins, Roland E. Dolle

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2006

Language:

english

File:

PDF, 112 KB

english, 2006

54

Further studies of tyrosine surrogates in opioid receptor peptide ligands

Roland E. Dolle, Mathieu Michaut, Blanca Martinez-Teipel, Serge Belanger, Thomas M. Graczyk, Robert N. DeHaven

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2007

Language:

english

File:

PDF, 164 KB

english, 2007

55

Biaryl cannabinoid mimetics—Synthesis and structure–activity relationship

Karin Worm, Q. Jean Zhou, Gabriel J. Stabley, Robert N. DeHaven, Roland E. Dolle

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2007

Language:

english

File:

PDF, 183 KB

english, 2007

56

Discovery of a series of aminopiperidines as novel iNOS inhibitors

Bertrand Le Bourdonnec, Lara K. Leister, Christopher A. Ajello, Joel A. Cassel, Pamela R. Seida, Heather O’Hare, Minghua Gu, Guo-Hua Chu, Paul A. Tuthill, Robert N. DeHaven, Roland E. Dolle

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2008

Language:

english

File:

PDF, 294 KB

english, 2008

57

Nascent structure–activity relationship study of a diastereomeric series of kappa opioid receptor antagonists derived from CJ-15,208

Roland E. Dolle, Mathieu Michaut, Blanca Martinez-Teipel, Pamela R. Seida, Christopher W. Ajello, Alison L. Muller, Robert N. DeHaven, Patrick J. Carroll

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2009

Language:

english

File:

PDF, 296 KB

english, 2009

58

On the conundrum of deriving exact solutions from approximate master equations

Roland Doll, David Zueco, Martijn Wubs, Sigmund Kohler, Peter Hänggi

Journal:

Chemical Physics

Year:

2008

Language:

english

File:

PDF, 165 KB

english, 2008

59

High-performance liquid chromatographic enantioseparation of methanobenzazocines

William M. Barker, Karin Worm, Roland E. Dolle

Journal:

Journal of Chromatography A

Year:

2009

Language:

english

File:

PDF, 348 KB

english, 2009

60

General and efficient synthetic approach to novel tricyclic spiroketones

Guo-Hua Chu, Bertrand Le Bourdonnec, Minghua Gu, Christopher T. Saeui, Roland E. Dolle

Journal:

Year:

2009

Language:

english

File:

PDF, 266 KB

english, 2009

61

A facile synthesis of novel 2-amino-6-arylmethyl-7-carboxamido-7,8-dihydropyrimido[5,4-f][1,4]thiazepin-5-ones

Lan-Ying Qin, Andrew G. Cole, Axel Metzger, Marc-Raleigh Brescia, Kurt W. Saionz, Joan J. Zhang, Pascal Rigollier, James R. Wareing, Hubert Gstach, Juerg Zimmermann, Roland E. Dolle, John J. Baldwin,

Journal:

Tetrahedron Letters

Year:

2010

Language:

english

File:

PDF, 1.37 MB

english, 2010

62

9-(Sulfoximinoalkyl)guanine nucleosides as potential antiherpetic agents

Roland E. Dolle, David McNair

Journal:

Tetrahedron Letters

Year:

1993

Language:

english

File:

PDF, 273 KB

english, 1993

63

Regiocontrolled synthesis of the ergosterol B-isomers

Roland E. Dolle, Stanley J. Schmidt, Lawrence I. Kruse

Journal:

Tetrahedron Letters

Year:

1988

Language:

english

File:

PDF, 117 KB

english, 1988

64

Intramolecular [4+2] cycloaddition of α,β-unsaturated hydrazones as a route to annelated pyridines

Roland E. Dolle, W.Paul Armstrong, Antony N. Shaw, Riccardo Novelli

Journal:

Tetrahedron Letters

Year:

1988

Language:

english

File:

PDF, 205 KB

english, 1988

65

Enantioselective synthesis of (+)-pinidine

Roland E. Dolle, Kelly I. Osifo, Chun-Sing Li

Journal:

Tetrahedron Letters

Year:

1991

Language:

english

File:

PDF, 87 KB

english, 1991

66

Enantioselective synthesis of (+)-(2S,3s)-3-ethynyltyrosine

Antony N. Shaw, Roland E. Dolle, Lawrence I. Kruse

Journal:

Tetrahedron Letters

Year:

1990

Language:

english

File:

PDF, 212 KB

english, 1990

67

Solid-phase synthesis of α-hydroxy phosphonates and hydroxystatine amides. Transition-state isosteres derived from resin-bound amino acid aldehydes

Roland E Dolle, Timothy F Herpin, Yvonne Class Shimshock

Journal:

Tetrahedron Letters

Year:

2001

Language:

english

File:

PDF, 125 KB

english, 2001

68

Concomitant [2,3]-sigmatropic rearrangement of allylic sulfilimines and intramolecular N-alkylation. Synthesis of 2-vinyl substituted cyclic amines

Roland E. Dolle, Chun-Sing Li, Antony N. Shaw

Journal:

Tetrahedron Letters

Year:

1989

Language:

english

File:

PDF, 222 KB

english, 1989

69

Allylindium and allylboronic acid pinacolate: Mild reagents for the allylation of resin-bound aldehydes. Application to the solid-phase synthesis of hydroxypropylamines

Cullen L. Cavallaro, Timothy Herpin, Brian F. McGuinness, Yvonne Class Shimshock, Roland E. Dolle

Journal:

Tetrahedron Letters

Year:

1999

Language:

english

File:

PDF, 308 KB

english, 1999

70

Application of the intramolecular azomethine imine cycloaddition to the construction of a novel, orthogonally protected spirodiamino acid scaffold

Roland E Dolle, Michael C Barden, Paul E Brennan, Gulzar Ahmed, Vinh Tran, Douglas M Ho

Journal:

Tetrahedron Letters

Year:

1999

Language:

english

File:

PDF, 147 KB

english, 1999

71

Synthesis and evaluation of azapeptide-derived inhibitors of serine and cysteine proteases

Todd L. Graybill, Mitchell J. Ross, Bruce R. Gauvin, Jill S. Gregory, Alex L. Harris, Mark A. Ator, James M. Rinker, Roland E. Dolle

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1992

Language:

english

File:

PDF, 473 KB

english, 1992

72

α-((Tetronoyl)oxy)- and α-((tetramoyl)oxy)methyl ketone inhibitors of the interleukin-1β converting enzyme (ICE)

Todd L. Graybill, Catherine P. Prouty, Gary J. Speier, Denton Hoyer, Roland E. Dolle, Carla T. Helaszek, Mark A. Ator, Joanne Uhl, Joost Strastes

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1997

Language:

english

File:

PDF, 386 KB

english, 1997

73

3-chloro-4-carboxamido-6-arylpyridazines as a non-peptide class of interleukin-1β converting enzyme inhibitor

Roland E. Dolle, Denton Hoyer, James M. Rinker, Tina Morgan Ross, Stanley J. Schmidt, Carla T. Helaszek, Mark A. Ator

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1997

Language:

english

File:

PDF, 182 KB

english, 1997

74

Evaluation of a structure-based statine cyclic diamino amide encoded combinatorial library against plasmepsin II and cathepsin D

Carolyn DiIanni Carroll, Theodore O. Johnson, Shewei Tao, Giorgio Lauri, Marc Orlowski, Ilya Y. Gluzman, Daniel E. Goldberg, Roland E. Dolle

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1998

Language:

english

File:

PDF, 243 KB

english, 1998

75

Microwave-assisted Synthesis of Di- and trisubstituted Ureas from Thiophenoxy Carbamate Resins

Blanca Martinez-Teipel, Rosalyn C. Green, Roland E. Dolle

Journal:

Molecular Informatics

Year:

2004

Language:

english

File:

PDF, 79 KB

english, 2004

76

Discovery of enzyme inhibitors through combinatorial chemistry

Roland E. Dolle

Journal:

Molecular Diversity

Year:

1997

Language:

english

File:

PDF, 999 KB

english, 1997

77

PPARδ agonists suppress angiogenesis in a VEGFR2-dependent manner

Markus Meissner, Igor Hrgovic, Monika Doll, Roland Kaufmann

Journal:

Archives of Dermatological Research

Year:

2011

Language:

english

File:

PDF, 357 KB

english, 2011

78

Supporting large-scale hydrogeological monitoring and modelling by time-variable gravity data

Andreas Güntner, Roland Schmidt, Petra Döll

Journal:

Hydrogeology Journal

Year:

2007

Language:

english

File:

PDF, 727 KB

english, 2007

79

Impacts of Land Abandonment on Vegetation: Successional Pathways in European Habitats

Bernard Prévosto, Loek Kuiters, Markus Bernhardt-Römermann, Michaela Dölle, Wolfgang Schmidt, Maurice Hoffmann, Jan Van Uytvanck, Andreas Bohner, Daniel Kreiner, Jutta Stadler, Stephan Klotz, Roland B

Journal:

Folia Geobotanica

Year:

2011

Language:

english

File:

PDF, 419 KB

english, 2011

80

Ace inhibitors as a template for the design of bradykinin B2 receptor antagonists

Denton Hoyer, Mohamed M.A. Awad, Joseph M. Salvino, Peter R. Seoane, Roland E. Dolle, Wayne T. Houck, David G. Sawutz

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1995

Language:

english

File:

PDF, 207 KB

english, 1995

81

Synthesis of non-peptide bradykinin B2 receptor antagonists

Brent D. Douty, Joseph M. Salvino, Peter R. Seoane, Roland E. Dolle

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1995

Language:

english

File:

PDF, 187 KB

english, 1995

82

Characterization of a continuous fluorogenic assay for calpain I. Kinetic evaluation of peptide aldehydes, halomethyl ketones and (acyloxy)methyl ketones as inhibitors of the enzyme

Alex L. Harris, Jill S. Gregory, Alan L. Maycock, Todd L. Graybill, I.Kelly Osifo, Stanley J. Schmidt, Roland E. Dolle

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1995

Language:

english

File:

PDF, 431 KB

english, 1995

83

Structure activity relationships of non-peptide bradykinin B2 receptor antagonists

Joseph M. Salvino, Peter R. Seoane, Brent D. Douty, Mohamed A. Awad, Denton Hoyer, Tina Morgan Ross, Roland E. Dolle, Wayne T. Houck, David M. Faunce, David G. Sawutz

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1995

Language:

english

File:

PDF, 290 KB

english, 1995

84

Structural and stereochemical requirements of time-dependent inactivators of the interleukin-1β converting enzyme

C.V.C. Prasad, Catherine P. Prouty, Denton Hoyer, Tina M. Ross, Joseph M. Salvino, Mohamad Awad, Todd L. Graybill, Stanley J. Schmidt, I. Kelly Osifo, Roland E. Dolle, Carla T. Helaszek, Robert E. Mil

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1995

Language:

english

File:

PDF, 222 KB

english, 1995

85

Azepinone as a conformational constraint in the design of κ-opioid receptor agonists

Paul A. Tuthill, Pamela R. Seida, William Barker, Joel A. Cassel, Serge Belanger, Robert N. DeHaven, Michael Koblish, Susan L. Gottshall, Patrick J. Little, Diane L. DeHaven-Hudkins, Roland E. Dolle

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2004

Language:

english

File:

PDF, 371 KB

english, 2004

86

Arylacetamide κ opioid receptor agonists with reduced cytochrome P450 2D6 inhibitory activity

Bertrand Le Bourdonnec, Christopher W. Ajello, Pamela R. Seida, Roberta G. Susnow, Joel A. Cassel, Serge Belanger, Gabriel J. Stabley, Robert N. DeHaven, Diane L. DeHaven-Hudkins, Roland E. Dolle

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2005

Language:

english

File:

PDF, 182 KB

english, 2005

87

Combined solution-phase and solid-phase synthesis of 2-amino-7,8-dihydropteridin-6(5H)-ones

Axel Metzger, Lan-Ying Qin, Andrew G. Cole, Kurt W. Saionz, Marc-Raleigh Brescia, Hubert Gstach, James R. Wareing, Juerg Zimmermann, Wolfgang K-D. Brill, John J. Baldwin, Roland E. Dolle, Ian Henderso

Journal:

Tetrahedron Letters

Year:

2009

Language:

english

File:

PDF, 1.29 MB

english, 2009

88

EMERGENCY THORACIC SURGERY FOR PENETRATING, NON-MEDIASTINAL TRAUMA

Peter Loogna, Fabrizio Bonanno, Douglas M. Bowley, Dietrich Doll, Roland Girgensohn, Martin D. Smith, Miriam Glapa, Elias Degiannis

Journal:

ANZ Journal of Surgery

Year:

2007

Language:

english

File:

PDF, 59 KB

english, 2007

89

AP1-dependent repression of TGFα-mediated MMP9 upregulation by PPARδ agonists in keratinocytes

Markus Meissner, Barbara Berlinski, Monika Doll, Igor Hrgovic, Vesselina Laubach, Gabi Reichenbach, Stefan Kippenberger, Jens Gille, Roland Kaufmann

Journal:

Experimental Dermatology

Year:

2011

Language:

english

File:

PDF, 400 KB

english, 2011

90

Comprehensive survey of combinatorial libraries with undisclosed biological activity: 1992–1997

Roland E. Dolle

Journal:

Molecular Diversity

Year:

1998

Language:

english

File:

PDF, 624 KB

english, 1998

91

Comprehensive survey of chemical libraries yielding enzyme inhibitors, receptor agonists and antagonists, and other biologically active agents: 1992 through 1997

Roland E. Dolle

Journal:

Molecular Diversity

Year:

1997

Language:

english

File:

PDF, 687 KB

english, 1997

92

Analysis of libraries encoded with GC tags: Compound elution, tag decode analysis, and statistical sampling analysis

Roland E. Dolle, Joan Guo, Wenni Li, Ning Zhao, James A. Connelly

Journal:

Molecular Diversity

Year:

2000

Language:

english

File:

PDF, 240 KB

english, 2000

93

Annulation of Primary Amines to Piperazines and Diazaspirocycles Utilizing α-Methyl Benzyl Resin

Macleod, Calum, Martinez-Teipel, Blanca I., Barker, William M., Dolle, Roland E.

Journal:

Journal of Combinatorial Chemistry

Year:

2006

Language:

english

File:

PDF, 217 KB

english, 2006

94

Preparation and evaluation of peptidic aspartyl hemiacetals as reversible inhibitors of interleukin-l β converting enzyme (ICE)

TODD L. GRAYBILL, ROLAND E. DOLLE, CARLA T. HELASZEK, ROBERT E. MILLER, MARK A. ATOR

Journal:

Chemical Biology & Drug Design

Year:

1994

Language:

english

File:

PDF, 948 KB

english, 1994

95

Synthesis and evaluation of (+) and (−)-2,2-difluorocitrate as inhibitors of rat-liver ATP-citrate lyase and porcine-heart aconitase

Barbara A. SAXTY, Riccardo NOVELLI, Roland E. DOLLE, Lawrence I. KRUSE, David G. REID, Patrick CAMILLERI, Timothy N. C. WELLS

Journal:

Year:

1991

Language:

english

File:

PDF, 752 KB

english, 1991

96

Rescue of cytochrome P450 oxidoreductase (Por) mouse mutants reveals functions in vasculogenesis, brain and limb patterning linked to retinoic acid homeostasis

Vanessa Ribes, Diana M.E. Otto, Leslie Dickmann, Katy Schmidt, Brigitte Schuhbaur, Colin Henderson, Rune Blomhoff, C. Roland Wolf, Cheryll Tickle, Pascal Dollé

Journal:

Developmental Biology

Year:

2007

Language:

english

File:

PDF, 2.51 MB

english, 2007

97

Ligand activation of peroxisome proliferator-activated receptor delta suppresses cathepsin B expression in human endothelial cells in a posttranslational manner

Gabi Reichenbach, Anna Starzinski-Powitz, Monika Doll, Igor Hrgovic, Eva Maria Valesky, Stefan Kippenberger, August Bernd, Roland Kaufmann, Markus Meissner

Journal:

Experimental Dermatology

Year:

2012

Language:

english

File:

PDF, 435 KB

english, 2012

98

3-Aminopropylphosphinic acid—a potent, selective GABAB receptor agonist in the guinea-pig ileum and rat anococcygeus muscle

Judith M. Hills, Rhona A. Dingsdale, Michael E. Parsons, Roland E. Dolle, William Howson

Journal:

British Journal of Pharmacology

Year:

1989

Language:

english

File:

PDF, 791 KB

english, 1989

99

Comprehensive Survey of Combinatorial Library Synthesis: 2004

Dolle, Roland E.

Journal:

Journal of Combinatorial Chemistry

Year:

2005

Language:

english

File:

PDF, 15.59 MB

english, 2005

100

Comprehensive Survey of Combinatorial Library Synthesis: 1998

Dolle, Roland E., Nelson, Kingsley H.

Journal:

Journal of Combinatorial Chemistry

Year:

1999

Language:

english

File:

PDF, 2.01 MB

english, 1999