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51

Synthesis and cyclooxygenase and 5-lipoxygenase inhibitory activity of some thiazolidene-4-one analogs of meclofenamic acid

Diane H. Boschelli, David T. Connor, Paul J. Kuipers, Clifford D. Wright

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1992

Language:

english

File:

PDF, 222 KB

english, 1992

52

Synthesis of reversed hydroxamic acids of indomethacin: dual inhibitors of cyclooxygenase and 5-lipoxygenase

James B. Kramer, Diane H. Boschelli, David T. Connor, Catherine R. Kostlan, Daniel L. Flynn, Richard D. Dyer, Dirk A. Bornemeier, John A. Kennedy, Clifford D. Wright, Paul J. Kuipers

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1992

Language:

english

File:

PDF, 364 KB

english, 1992

53

Conversion of NSAIDS into balanced dual inhibitors of cyclooxygenase and 5-lipoxygenase

Diane H. Boschelli, David T. Connor, Milton Hoefle, Dirk A. Bornemeier, Richard D. Dyer

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1992

Language:

english

File:

PDF, 227 KB

english, 1992

54

4-Anilino-3-cyanobenzo[g]quinolines as Kinase Inhibitors

Nan Zhang, Biqi Wu, Allan Wissner, Dennis W Powell, Sridhar K Rabindran, Constance Kohler, Frank Boschelli

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 108 KB

english, 2002

55

Cyclooxygenase and 5-lipoxygenase inhibitory activity of 2,6 di-t-butylphenols linked by a sulfur atom to 1,3,4-thiadiazoles and 1,3,4-oxadiazoles

James B. Kramer, Diane H. Boschelli, David T. Connor, Catherine R. Kostlan, Paul J. Kuipers, John A. Kennedy, Clifford D. Wright, Dirk A. Bornemeier, Richard D. Dyer

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1993

Language:

english

File:

PDF, 240 KB

english, 1993

56

Inhibition of Src kinase activity by 4-anilino-7-thienyl-3-quinolinecarbonitriles

Diane H. Boschelli, Daniel Y. Wang, Fei Ye, Ayako Yamashita, Nan Zhang, Dennis Powell, Jennifer Weber, Frank Boschelli

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 133 KB

english, 2002

57

8-Anilinoimidazo[4,5-g]quinoline-7-carbonitriles as Src Kinase Inhibitors

Dan Berger, Minu Dutia, Dennis Powell, Biqi Wu, Allan Wissner, Frenel DeMorin, Jennifer Weber, Frank Boschelli

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 139 KB

english, 2002

58

Substituted 4-anilino-7-phenyl-3-quinolinecarbonitriles as Src kinase inhibitors

Dan Berger, Minu Dutia, Dennis Powell, Allan Wissner, Frenel DeMorin, Yuri Raifeld, Jennifer Weber, Frank Boschelli

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 127 KB

english, 2002

59

Inhibition of Src kinase activity by 4-anilino-5,10-dihydro-pyrimido[4,5-b]quinolines

Diane H. Boschelli, Dennis Powell, Jennifer M. Golas, Frank Boschelli

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2003

Language:

english

File:

PDF, 172 KB

english, 2003

60

Synthesis and evaluation of 4-Anilino-6,7-dialkoxy-3-quinolinecarbonitriles as inhibitors of kinases of the Ras-MAPK signaling cascade

Dan Berger, Minu Dutia, Dennis Powell, Biqi Wu, Allan Wissner, Diane H. Boschelli, M.Brawner Floyd, Nan Zhang, Nancy Torres, Jeremy Levin, Xuemei Du, Donald Wojciechowicz, Carolyn Discafani, Constance

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2003

Language:

english

File:

PDF, 173 KB

english, 2003

61

Synergy between 5,10-dideaza-5,6,7,8-tetrahydrofolic acid and methotrexate in mice bearing L1210 tumors

K. Ferguson, D. Boschelli, P. Hoffman, A. Oronsky, J. Whiteley, S. Webber, J. Galivan, J. Freishiem, J. Hynes, S. S. Kerwar

Journal:

Cancer Chemotherapy and Pharmacology

Year:

1989

Language:

english

File:

PDF, 392 KB

english, 1989

62

Crystal and molecular structure of geiparvarin

Bruce H. Toder, Diane Boschelli, Amos B. Smith

Journal:

Journal of Chemical Crystallography

Year:

1979

Language:

english

File:

PDF, 437 KB

english, 1979

63

A cell-based screen for inhibitors of protein folding and degradation

Frank Boschelli, Jennifer M. Golas, Roseann Petersen, Vincent Lau, Lei Chen, Diane Tkach, Qiang Zhao, Dave S. Fruhling, Hao Liu, Chaneun Nam, Kim T. Arndt

Journal:

Cell Stress and Chaperones

Year:

2010

Language:

english

File:

PDF, 518 KB

english, 2010

64

Total synthesis of (±)-desepoxy-4,5-didehybromethylenomycin A

Diane Boschelli, Robert M. Scarborough Jr., Amos B. Smith III

Journal:

Tetrahedron Letters

Year:

1981

Language:

english

File:

PDF, 247 KB

english, 1981

65

Further studies on ethenyl and ethynyl-4-phenylamino-3-quinolinecarbonitriles: identification of a subnanomolar Src kinase inhibitor

Ana Carolina Barrios Sosa, Diane H. Boschelli, Biqi Wu, Yan Wang, Jennifer M. Golas

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2005

Language:

english

File:

PDF, 120 KB

english, 2005

66

A facile, scalable preparation of 4-oxo-4,7-dihydrothieno[2,3-b]pyridine-5-carbonitriles

L. Nathan Tumey, Niala Bhagirath, Biqi Wu, Diane H. Boschelli

Journal:

Tetrahedron Letters

Year:

2008

Language:

english

File:

PDF, 161 KB

english, 2008

67

Synergistic activity of the Src/Abl inhibitor bosutinib in combination with imatinib

Redaelli, S, Boschelli, F, Perini, P, Pirola, A, Viltadi, M, Gambacorti-Passerini, C

Journal:

Year:

2010

Language:

english

File:

PDF, 324 KB

english, 2010

68

ChemInform Abstract: Optimization of 7-Alkene-3-quinolinecarbonitriles as Src Kinase Inhibitors.

Diane H. Boschelli, Daniel Wang, Yan Wang, Biqi Wu, Erick E. Honores, Ana Carolina Barrios Sosa, Inder Chaudhary, Jennifer Golas, Judy Lucas, Frank Boschelli

Journal:

Year:

2010

File:

PDF, 20 KB

2010

69

2-Substituted Aminopyrido[2,3-d]pyrimidin-7(8H)-ones. Structure−Activity Relationships Against Selected Tyrosine Kinases and in Vitro and in Vivo Anticancer Activity

Klutchko, Sylvester R., Hamby, James M., Boschelli, Diane H., Wu, Zhipei, Kraker, Alan J., Amar, Aneesa M., Hartl, Brian G., Shen, Cynthia, Klohs, Wayne D., Steinkampf, Randall W.

Journal:

Journal of Medicinal Chemistry

Year:

1998

Language:

english

File:

PDF, 404 KB

english, 1998

70

ChemInform Abstract: Inhibition of E-Selectin-, ICAM-1, and VCAM-1-Mediated Cell Adhesion by Benzo(b)thiophene-, Benzofuran-, Indole-, and Naphthalene-2- carboxamides: Identification of PD 144795 as an Antiinflammatory Agent.

D. H. BOSCHELLI, J. B. KRAMER, S. S. KHATANA, R. J. SORENSON, D. T. CONNOR, M. A. FERIN, C. D. WRIGHT, M. E. LESCH, K. IMRE, G. C. OKONKWO, D. J. SCHRIER, M. C. CONROY, E. FERGUSON, J. WOELLE, U. SAXE

Journal:

Year:

1996

Language:

english

File:

PDF, 32 KB

english, 1996

71

Optimization of 4-Phenylamino-3-quinolinecarbonitriles as Potent Inhibitors of Src Kinase Activity

Boschelli, Diane H., Ye, Fei, Wang, Yanong D., Dutia, Minu, Johnson, Steve L., Wu, Biqi, Miller, Karen, Powell, Dennis W., Yaczko, Deanna, Young, Mairead

Journal:

Journal of Medicinal Chemistry

Year:

2001

Language:

english

File:

PDF, 245 KB

english, 2001

72

Synthesis and Tyrosine Kinase Inhibitory Activity of a Series of 2-Amino-8H-pyrido[2,3-d]pyrimidines: Identification of Potent, Selective Platelet-Derived Growth Factor Receptor Tyrosine Kinase Inhibitors

Boschelli, Diane H., Wu, Zhipei, Klutchko, Sylvester R., Showalter, H. D. Hollis, Hamby, James M., Lu, Gina H., Major, Terry C., Dahring, Tawny K., Batley, Brian, Panek, Robert L.

Journal:

Journal of Medicinal Chemistry

Year:

1998

Language:

english

File:

PDF, 219 KB

english, 1998

73

Preparation of Benzothieno[2,3-f]-1,4-oxazepin- and -thiazepin-5(2H)-ones and of Benzothieno[3,2-e]-1,4-diazepin-5-ones

Khatana, Sonya S., Boschelli, Diane H., Kramer, James B., Connor, David T., Barth, Hubert, Stoss, Peter

Journal:

Journal of Organic Chemistry

Year:

1996

Language:

english

File:

PDF, 156 KB

english, 1996

74

Inhibition of Tumor Necrosis Factor Induced Human Aortic Endothelial Cell Adhesion Molecule Gene Expression by an Alkoxybenzo[b]thiophene-2-carboxamide

J. Wolle, E. Ferguson, C. Keshava, L.J. Devall, D.H. Boschelli, R.S. Newton, U. Saxena

Journal:

Biochemical and Biophysical Research Communications

Year:

1995

File:

PDF, 253 KB

1995

75

Synthesis and biological properties of 5,10-dideaza-5,6,7,8-tetrahydrofolic acid

Diane H. Boschelli, Stephanie Webber, John M. Whiteley, Arnold L. Oronsky, S.S. Kerwar

Journal:

Archives of Biochemistry and Biophysics

Year:

1988

Language:

english

File:

PDF, 554 KB

english, 1988

76

Bosutinib: A review of preclinical studies in chronic myelogenous leukaemia

Frank Boschelli, Kim Arndt, Carlo Gambacorti-Passerini

Journal:

European Journal of Cancer

Year:

2010

Language:

english

File:

PDF, 282 KB

english, 2010

77

Structure−Activity Relationships for 1-Phenylbenzimidazoles as Selective ATP Site Inhibitors of the Platelet-Derived Growth Factor Receptor

Palmer, Brian D., Smaill, Jeff B., Boyd, Maruta, Boschelli, Diane H., Doherty, Annette M., Hamby, James M., Khatana, Sonya S., Kramer, James B., Kraker, Alan J., Panek, Robert L., Lu, Gina H., Dahring

Journal:

Journal of Medicinal Chemistry

Year:

1998

Language:

english

File:

PDF, 169 KB

english, 1998

78

Synthesis and Src Kinase Inhibitory Activity of 2-Phenyl- and 2-Thienyl-7-phenylaminothieno[3,2- b ]pyridine-6-carbonitriles

Boschelli, Diane H., Wu, Biqi, Barrios Sosa, Ana Carolina, Durutlic, Haris, Chen, Joan J., Wang, Yan, Golas, Jennifer M., Lucas, Judy, Boschelli, Frank

Journal:

Journal of Medicinal Chemistry

Year:

2005

Language:

english

File:

PDF, 197 KB

english, 2005

79

Pyrido[2,3- d ]pyrimidin-7-one Inhi-bitors of Cyclin-Dependent Kinases.

Barvian, Mark, Boschelli, Diane H., Cossrow, Jennifer, Dobrusin, Ellen, Fattaey, Ali, Fritsch, Alex, Fry, David, Harvey, Patricia, Keller, Paul, Garrett, Michelle, La, Frances, Leopold, Wilbur, McNama

Journal:

Journal of Medicinal Chemistry

Year:

2001

Language:

english

File:

PDF, 15 KB

english, 2001

80

118 Substituted 7-amino-4-anilino-6-alkoxy-3-quinolinecarbonitriles as Src kinase inhibitors

H. Tsou, E. Overbeek-Klumpers, W. Hallett, J. Golas, F. Boschelli

Journal:

European Journal of Cancer Supplements

Year:

2004

Language:

english

File:

PDF, 126 KB

english, 2004

81

Represser-operator interaction in the lac operon: II. Observations at the tyrosines and tryptophans

Harry Nick, Kim Arndt, Frank Boschelli, Mary Ann Jarema, Marcella Lillis, Hans Sommer, Ponzy Lu, John Sadler

Journal:

Journal of Molecular Biology

Year:

1982

Language:

english

File:

PDF, 1.58 MB

english, 1982

82

Repressor-operator interaction in the lac operon: III. Nuclear magnetic resonance observations with altered amino-terminal DNA binding domains

Kim Arndt, Harry Nick, Frank Boschelli, Ponzy Lu, John Sadler

Journal:

Journal of Molecular Biology

Year:

1982

Language:

english

File:

PDF, 1.21 MB

english, 1982

83

Lambda phage cro repressor: Non-specific DNA binding

Frank Boschelli

Journal:

Journal of Molecular Biology

Year:

1982

Language:

english

File:

PDF, 1.01 MB

english, 1982

84

Lambda phage cro repressor: DNA sequence-dependent interactions seen by tyrosine fluorescence

Frank Boschelli, Kim Arndt, Harry Nick, Qijiu Zhang, Ponzy Lu, Yoshinori Takeda

Journal:

Journal of Molecular Biology

Year:

1982

Language:

english

File:

PDF, 1.23 MB

english, 1982

85

4-Anilino-6,7-dialkoxyquinoline-3-carbonitrile Inhibitors of Epidermal Growth Factor Receptor Kinase and Their Bioisosteric Relationship to the 4-Anilino-6,7-dialkoxyquinazoline Inhibitors

Wissner, Allan, Berger, Dan M., Boschelli, Diane H., Floyd, M. Brawner, Greenberger, Lee M., Gruber, Brian C., Johnson, Bernard D., Mamuya, Nellie, Nilakantan, Ramaswamy, Reich, Marvin F., Shen, Ru, T

Journal:

Journal of Medicinal Chemistry

Year:

2000

Language:

english

File:

PDF, 384 KB

english, 2000

86

1,3,4-Oxadiazole, 1,3,4-thiadiazole, and 1,2,4-triazole analogs of the fenamates: in vitro inhibition of cyclooxygenase and 5-lipoxygenase activities

Boschelli, Diane H., Connor, David T., Bornemeier, Dirk A., Dyer, Richard D., Kennedy, John A., Kuipers, Paul J., Okonkwo, Godwin C., Schrier, Denis J., Wright, Clifford D.

Journal:

Journal of Medicinal Chemistry

Year:

1993

Language:

english

File:

PDF, 1.07 MB

english, 1993

87

Identification of 7-Phenylaminothieno- [3,2- b ]pyridine-6-carbonitriles as a New Class of Src Kinase Inhibitors

Boschelli, Diane H., Wu, Biqi, Barrios Sosa, Ana Carolina, Durutlic, Haris, Ye, Fei, Raifeld, Yuri, Golas, Jennifer M., Boschelli, Frank

Journal:

Journal of Medicinal Chemistry

Year:

2004

Language:

english

File:

PDF, 182 KB

english, 2004

88

Discovery of Dibenzo[ c , f ][2,7]naphthyridines as Potent and Selective 3-Phosphoinositide-Dependent Kinase-1 Inhibitors

Gopalsamy, Ariamala, Shi, Mengxiao, Boschelli, Diane H., Williamson, Robert, Olland, Andrea, Hu, Yongbo, Krishnamurthy, Girija, Han, Xin, Arndt, Kim, Guo, Bing

Journal:

Journal of Medicinal Chemistry

Year:

2007

Language:

english

File:

PDF, 170 KB

english, 2007

89

Pyrido[2,3- d ]pyrimidin-7-one Inhibitors of Cyclin-Dependent Kinases

Barvian, Mark, Boschelli, Diane H., Cossrow, Jennifer, Dobrusin, Ellen, Fattaey, Ali, Fritsch, Alex, Fry, David, Harvey, Patricia, Keller, Paul, Garrett, Michelle, La, Frances, Leopold, Wilbur, McNama

Journal:

Journal of Medicinal Chemistry

Year:

2000

Language:

english

File:

PDF, 228 KB

english, 2000

90

Inhibition of E-Selectin-, ICAM-1-, and VCAM-1-Mediated Cell Adhesion by Benzo[b]thiophene-, Benzofuran-, Indole-, and Naphthalene-2-carboxamides: Identification of PD 144795 as an Antiinflammatory Agent

Boschelli, Diane H., Kramer, James B., Khatana, Sonya S., Sorenson, Roderick J., Connor, David T., Ferin, Mark A., Wright, Clifford D., Lesch, Mark E., Imre, Kathleen

Journal:

Journal of Medicinal Chemistry

Year:

1995

Language:

english

File:

PDF, 2.55 MB

english, 1995

91

7-Alkoxy-4-phenylamino-3-quinolinecar-bonitriles as Dual Inhibitors of Src and Abl Kinases

Boschelli, Diane H., Wang, Yanong D., Johnson, Steve, Wu, Biqi, Ye, Fei, Barrios Sosa, Ana Carolina, Golas, Jennifer M., Boschelli, Frank

Journal:

Journal of Medicinal Chemistry

Year:

2004

Language:

english

File:

PDF, 53 KB

english, 2004

92

[Part 1: Biological Sciences] || lac Repressor--lac Operator Interaction: NMR Observations

Harry Nick, Kim Arndt, Frank Boschelli, Mary Ann C. Jarema, Marcella Lillis, John Sadler, Marvin Caruthers and Ponzy Lu

Journal:

Proceedings of the National Academy of Sciences

Year:

1982

Language:

english

File:

PDF, 1.44 MB

english, 1982

93

Benzylidene-thiolactone rearrangement: synthesis and rearrangement of 5-substituted-3-benzylidene-4-thiolen-2-ones

Heindel, Ned D., Conley, Richard A., Minatelli, John A., Boschelli, Diane Harris

Journal:

Journal of Organic Chemistry

Year:

1983

Language:

english

File:

PDF, 390 KB

english, 1983

94

3-Alkoxybenzo[b]thiophene-2-carboxamides as Inhibitors of Neutrophil-Endothelial Cell Adhesion

Boschelli, Diane H., Kramer, James B., Connor, David T., Lesch, Mark E., Schrier, Denis J., Ferin, Mark A., Wright, Clifford D.

Journal:

Journal of Medicinal Chemistry

Year:

1994

Language:

english

File:

PDF, 256 KB

english, 1994

95

Lac Repressor: a proton magnetic resonance look at the deoxyribonucleic acid binding fragment

Arndt, Kim T., Boschelli, Frank, Lu, Ponzy, Miller, Jeffrey H.

Journal:

Year:

1981

Language:

english

File:

PDF, 1.20 MB

english, 1981

96

Synthesis and Src Kinase Inhibitory Activity of a Series of 4-[(2,4-Dichloro-5-methoxyphenyl)amino]-7-furyl-3-quinolinecarbonitriles

Boschelli, Diane H., Wu, Biqi, Ye, Fei, Wang, Yan, Golas, Jennifer M., Lucas, Judy, Boschelli, Frank

Journal:

Journal of Medicinal Chemistry

Year:

2006

Language:

english

File:

PDF, 142 KB

english, 2006

97

Stereocontrolled total synthesis of (.+-.)-xanthocidin, two diastereomers, (.+-.)-epixanthocidin and (.+-.)-.beta.-isoxanthocidin, and (.+-.)-dedihydroxy-4,5-didehydroxanthocidin, a likely biosynthetic precursor

Smith, Amos B., Boschelli, Diane

Journal:

Journal of Organic Chemistry

Year:

1983

Language:

english

File:

PDF, 1.42 MB

english, 1983

98

Synthesis and Src Kinase Inhibitory Activity of a Series of 4-Phenylamino-3-quinolinecarbonitriles

Boschelli, Diane H., Wang, Yanong D., Ye, Fei, Wu, Biqi, Zhang, Nan, Dutia, Minu, Powell, Dennis W., Wissner, Allan, Arndt, Kim, Weber, Jennifer M., Boschelli, Frank

Journal:

Journal of Medicinal Chemistry

Year:

2001

Language:

english

File:

PDF, 162 KB

english, 2001

99

4-Anilino-7,8-dialkoxybenzo[ g ]quinoline-3-carbonitriles as Potent Src Kinase Inhibitors

Berger, Dan M., Dutia, Minu, Birnberg, Gary, Powell, Dennis, Boschelli, Diane H., Wang, Yanong D., Ravi, Malini, Yaczko, Deanna, Golas, Jennifer, Lucas, Judy, Boschelli, Frank

Journal:

Journal of Medicinal Chemistry

Year:

2005

Language:

english

File:

PDF, 576 KB

english, 2005

100

Identification of a Conserved Sequence Motif That Promotes Cdc37 and Cyclin D1 Binding to Cdk4

Zhao, Q., Boschelli, F., Caplan, A. J., Arndt, K. T.

Journal:

Journal of Biological Chemistry

Year:

2004

Language:

english

File:

PDF, 207 KB

english, 2004