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1

A new opioid designed multiple ligand derived from the μ opioid agonist endomorphin-2 and the δ opioid antagonist pharmacophore Dmt-Tic

Severo Salvadori, Claudio Trapella, Stella Fiorini, Lucia Negri, Roberta Lattanzi, Sharon D. Bryant, Yunden Jinsmaa, Lawrence H. Lazarus, Gianfranco Balboni

Journal:

Bioorganic & Medicinal Chemistry

Year:

2007

Language:

english

File:

PDF, 160 KB

english, 2007

2

Synthesis and activity of 3-pyridylamine ligands at central nicotinic receptors

Gianfranco Balboni, Mauro Marastoni, Stefania Merighi, Pier Andrea Borea, Roberto Tomatis

Journal:

European Journal of Medicinal Chemistry

Year:

2000

Language:

english

File:

PDF, 125 KB

english, 2000

3

New Opioid Designed Multiple Ligand from Dmt-Tic and Morphinan Pharmacophores

Neumeyer, John L., Peng, Xuemei, Knapp, Brian I., Bidlack, Jean M., Lazarus, Lawrence H., Salvadori, Severo, Trapella, Claudio, Balboni, Gianfranco

Journal:

Journal of Medicinal Chemistry

Year:

2006

Language:

english

File:

PDF, 69 KB

english, 2006

4

Further Studies on Lead Compounds Containing the Opioid Pharmacophore Dmt-Tic

Balboni, Gianfranco, Fiorini, Stella, Baldisserotto, Anna, Trapella, Claudio, Sasaki, Yusuke, Ambo, Akihiro, Marczak, Ewa D., Lazarus, Lawrence H., Salvadori, Severo

Journal:

Journal of Medicinal Chemistry

Year:

2008

Language:

english

File:

PDF, 484 KB

english, 2008

5

Benzofuran hydrazones as potential scaffold in the development of multifunctional drugs: Synthesis and evaluation of antioxidant, photoprotective and antiproliferative activity

Baldisserotto, Anna, Demurtas, Monica, Lampronti, Ilaria, Moi, Davide, Balboni, Gianfranco, Vertuani, Silvia, Manfredini, Stefano, Onnis, Valentina

Journal:

European Journal of Medicinal Chemistry

Year:

2018

Language:

english

File:

PDF, 800 KB

english, 2018

6

Indole derivatives as multifunctional drugs: Synthesis and evaluation of antioxidant, photoprotective and antiproliferative activity of indole hydrazones

Demurtas, Monica, Baldisserotto, Anna, Lampronti, Ilaria, Moi, Davide, Balboni, Gianfranco, Pacifico, Salvatore, Vertuani, Silvia, Manfredini, Stefano, Onnis, Valentina

Journal:

Bioorganic Chemistry

Year:

2019

Language:

english

File:

PDF, 896 KB

english, 2019

7

Effect of lysine residues on the deamidation reaction of asparagine side chains

Sante Capasso, Gianfranco Balboni, Paola Di Cerbo

Journal:

Year:

2000

Language:

english

File:

PDF, 98 KB

english, 2000

8

Nmr studies of a series of dehydrodermorphins

Maria A. Castiglione-Morelli, Gabriella Saviano, Piero A. Temussi, Gianfranco Balboni, Severo Salvadori, Roberto Tomatis

Journal:

Year:

1989

Language:

english

File:

PDF, 479 KB

english, 1989

9

δ-, but not µ-, opioid receptor stabilizes K+ homeostasis by reducing Ca2+ influx in the cortex during acute hypoxia

Dongman Chao, Alia Bazzy-Asaad, Gianfranco Balboni, Ying Xia

Journal:

Journal of Cellular Physiology

Year:

2007

Language:

english

File:

PDF, 325 KB

english, 2007

10

Opioid peptides. Synthesis and biological properties of dermorphin related hexapeptides

Severo Salvadori, Mauro Marastoni, Gianfranco Balboni, Pierandrea Borea, Roberto Tomatis

Journal:

European Journal of Medicinal Chemistry

Year:

1990

Language:

english

File:

PDF, 775 KB

english, 1990

11

Synthesis and opioid activity of N,N-Dimethyl-Dmt-Tic-NH-CH(R)-R′ analogues: acquisition of potent δ antagonism

Gianfranco Balboni, Severo Salvadori, Remo Guerrini, Lucia Negri, Elisa Giannini, Sharon D Bryant, Yunden Jinsmaa, Lawrence H Lazarus

Journal:

Bioorganic & Medicinal Chemistry

Year:

2003

Language:

english

File:

PDF, 251 KB

english, 2003

12

Further studies on the effect of lysine at the C-terminus of the Dmt-Tic opioid pharmacophore

Gianfranco Balboni, Valentina Onnis, Cenzo Congiu, Margherita Zotti, Yusuke Sasaki, Akihiro Ambo, Sharon D. Bryant, Yunden Jinsmaa, Lawrence H. Lazarus, Ilaria Lazzari, Claudio Trapella, Severo Salvad

Journal:

Bioorganic & Medicinal Chemistry

Year:

2007

Language:

english

File:

PDF, 216 KB

english, 2007

13

Role of benzimidazole (Bid) in the δ-opioid agonist pseudopeptide H-Dmt-Tic-NH-CH2-Bid (UFP-502)

Severo Salvadori, Stella Fiorini, Claudio Trapella, Frank Porreca, Peg Davis, Yusuke Sasaki, Akihiro Ambo, Ewa D. Marczak, Lawrence H. Lazarus, Gianfranco Balboni

Journal:

Bioorganic & Medicinal Chemistry

Year:

2008

Language:

english

File:

PDF, 172 KB

english, 2008

14

Novel multiple opioid ligands based on 4-aminobenzazepinone (Aba), azepinoindole (Aia) and tetrahydroisoquinoline (Tic) scaffolds

Steven Ballet, Ewa D. Marczak, Debby Feytens, Severo Salvadori, Yusuke Sasaki, Andrew D. Abell, Lawrence H. Lazarus, Gianfranco Balboni, Dirk Tourwé

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2010

Language:

english

File:

PDF, 357 KB

english, 2010

15

Opioid bifunctional ligands from morphine and the opioid pharmacophore Dmt-Tic

Gianfranco Balboni, Severo Salvadori, Ewa D. Marczak, Brian I. Knapp, Jean M. Bidlack, Lawrence H. Lazarus, Xuemei Peng, Yu Gui Si, John L. Neumeyer

Journal:

European Journal of Medicinal Chemistry

Year:

2011

Language:

english

File:

PDF, 234 KB

english, 2011

16

Assessment of substitution in the second pharmacophore of Dmt-Tic analogues

Vincenzo Santagada, Gianfranco Balboni, Giuseppe Caliendo, Remo Guerrini, Severo Salvadori, Clementina Bianchi, Sharon D Bryant, Lawrence H Lazarus

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2000

Language:

english

File:

PDF, 125 KB

english, 2000

17

δ-Opioid receptors protect from anoxic disruption of Na+homeostasis via Na+channel regulation

Xuezhi Kang, Dongman Chao, Quanbao Gu, Guanghong Ding, Yingwei Wang, Gianfranco Balboni, Lawrence H. Lazarus, Ying Xia

Journal:

Cellular and Molecular Life Sciences

Year:

2009

Language:

english

File:

PDF, 514 KB

english, 2009

18

Role of 2′,6′-dimethyl-l-tyrosine (Dmt) in some opioid lead compounds

Gianfranco Balboni, Erika Marzola, Yusuke Sasaki, Akihiro Ambo, Ewa D. Marczak, Lawrence H. Lazarus, Severo Salvadori

Journal:

Bioorganic & Medicinal Chemistry

Year:

2010

Language:

english

File:

PDF, 208 KB

english, 2010

19

Synthesis and activity profiles of new dermorphin-(1-4) peptide analogs

Marastoni, Mauro, Salvadori, Severo, Balboni, Gianfranco, Borea, Pier Andrea, Marzola, Giuliano, Tomatis, Roberto

Journal:

Journal of Medicinal Chemistry

Year:

1987

Language:

english

File:

PDF, 748 KB

english, 1987

20

Flavones and structurally related 4-chromenones inhibit carbonic anhydrases by a different mechanism of action compared to coumarins

Gianfranco Balboni, Cenzo Congiu, Valentina Onnis, Alfonso Maresca, Andrea Scozzafava, Jean-Yves Winum, Annalisa Maietti, Claudiu T. Supuran

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2012

Language:

english

File:

PDF, 277 KB

english, 2012

21

Peptidic delta opioid receptor agonists produce antidepressant-like effects in the forced swim test and regulate BDNF mRNA expression in rats

Mary M. Torregrossa, Emily M. Jutkiewicz, Henry I. Mosberg, Gianfranco Balboni, Stanley J. Watson, James H. Woods

Journal:

Year:

2006

Language:

english

File:

PDF, 603 KB

english, 2006

22

Orally administered H-Dmt-Tic-Lys-NH-CH2-Ph (MZ-2), a potent µ-/δ-opioid receptor antagonist, regulates obese-related factors in mice

Ewa D. Marczak, Yunden Jinsmaa, Page H. Myers, Terry Blankenship, Ralph Wilson, Gianfranco Balboni, Severo Salvadori, Lawrence H. Lazarus

Journal:

European Journal of Pharmacology

Year:

2009

Language:

english

File:

PDF, 676 KB

english, 2009

23

DOR activation inhibits anoxic/ischemic Na+ influx through Na+ channels via PKC mechanisms in the cortex

Dongman Chao, Xiaozhou He, Yilin Yang, Alia Bazzy-Asaad, Lawrence H. Lazarus, Gianfranco Balboni, Dong H. Kim, Ying Xia

Journal:

Experimental Neurology

Year:

2012

Language:

english

File:

PDF, 1.24 MB

english, 2012

24

Inhibition of the development of morphine tolerance by a potent dual μ-/δ-opioid antagonist, H-Dmt-Tic-Lys-NH-CH2-Ph

Yunden Jinsmaa, Ewa D. Marczak, Gianfranco Balboni, Severo Salvadori, Lawrence H. Lazarus

Journal:

Pharmacology Biochemistry and Behavior

Year:

2008

Language:

english

File:

PDF, 479 KB

english, 2008

25

Novel 2-amino-isoflavones exhibit aryl hydrocarbon receptor agonist or antagonist activity in a species/cell-specific context

Richard J. Wall, Guochun He, Michael S. Denison, Cenzo Congiu, Valentina Onnis, Alwyn Fernandes, David R. Bell, Martin Rose, J. Craig Rowlands, Gianfranco Balboni, Ian R. Mellor

Journal:

Year:

2012

Language:

english

File:

PDF, 468 KB

english, 2012

26

Inhibition of human multidrug resistance P-glycoprotein 1 by analogues of a potent δ-opioid antagonist

Tara Lovekamp, Peter S Cooper, Jenny Hardison, Sharon D Bryant, Remo Guerrini, Gianfranco Balboni, Severo Salvadori, Lawrence H Lazarus

Journal:

Year:

2001

Language:

english

File:

PDF, 82 KB

english, 2001

27

Inverse agonism by Dmt–Tic analogues and HS 378, a naltrindole analogue

Maryse Labarre, Joanne Butterworth, Stephane St-Onge, Kemal Payza, Helmut Schmidhammer, Severo Salvadori, Gianfranco Balboni, Remo Guerrini, Sharon D Bryant, Lawrence H Lazarus

Journal:

European Journal of Pharmacology

Year:

2000

Language:

english

File:

PDF, 77 KB

english, 2000

28

Design of δ-opioid peptide antagonists for emerging drug applications

Lawrence H Lazarus, Sharon D Bryant, Peter S Cooper, Remo Guerrini, Gianfranco Balboni, Severo Salvadori

Journal:

Drug Discovery Today

Year:

1998

Language:

english

File:

PDF, 424 KB

english, 1998

29

Synthesis and opioid activity of partial retro-inverso analogs of dermorphin

SEVERO SALVADORI, MAURO MARASTONI, GIANFRANCO BALBONI, GIANPIETRO SARTO, ROBERTO TOMATIS

Journal:

Chemical Biology & Drug Design

Year:

1985

Language:

english

File:

PDF, 509 KB

english, 1985

30

Dehydro-dermorphins : III. Circular dichroism investigation of conformation in solution

OSVALDO PIERONI, ADRIANO FISSI, SEVERO SALVADORI, GIANFRANCO BALBONI, ROBERTO TOMATIS

Journal:

Chemical Biology & Drug Design

Year:

1986

Language:

english

File:

PDF, 646 KB

english, 1986

31

Dehydro-dermorphins : II. Synthesis and biological activity of unsaturated dermorphin hexa and heptapeptides

SEVERO SALVADORI, MAURO MARASTONI, GIANFRANCO BALBONI, GIULIANO MARZOLA, ROBERTO TOMATIS

Journal:

Chemical Biology & Drug Design

Year:

1986

Language:

english

File:

PDF, 657 KB

english, 1986

32

Synthesis and biological activity of carboxyl terminally extended dermorphins

MAURO MARASTONI, SEVERO SALVADORI, GIANFRANCO BALBONI, GIULIANO MARZOLA, ETTORE CIRO DEGLIUBERTI, ROBERTO TOMATIS

Journal:

Chemical Biology & Drug Design

Year:

1986

Language:

english

File:

PDF, 555 KB

english, 1986

33

Dehydro-dermorphins : I. Influence of the stereo-orientation of aromatic groups in dermorphin-(1–5)-peptides to opioid activity

SEVERO SALVADORI, MAURO MARASTONI, GIANFRANCO BALBONI, GIULIANO MARZOLA, ROBERTO TOMATIS

Journal:

Chemical Biology & Drug Design

Year:

1986

Language:

english

File:

PDF, 566 KB

english, 1986

34

Opioid peptides Synthesis and binding properties of dermorphin related heptapeptides

SEVERO SALVADORI, MAURO MARASTONI, GIANFRANCO BALBONI, PIERANDREA BOREA, ROBERTO TOMATIS

Journal:

Chemical Biology & Drug Design

Year:

1989

Language:

english

File:

PDF, 611 KB

english, 1989

35

Synthesis, metabolic stability and chemotactic activity of peptide T and its analogues

MAURO MARASTONI, SEVERO SALVADORI, GIANFRANCO BALBONI, SUSANNA SPISANI, RICCARDO GAVIOLI, SERENA TRANIELLO, ROBERTO TOMATIS

Journal:

Chemical Biology & Drug Design

Year:

1990

Language:

english

File:

PDF, 618 KB

english, 1990

36

Acid catalysis in the formation of dioxopiperazines from peptides containing tetrahydroisoquinoline-3-carboxylic acid at position 2

SANTE CAPASSO, FILOMENA SICA, LELIO MAZZARELLA, GIANFRANCO BALBONI, REMO GUERRINI, SEVERO SALVADORI

Journal:

Chemical Biology & Drug Design

Year:

1995

Language:

english

File:

PDF, 577 KB

english, 1995

37

Design and Solution Structure of a Partially Rigid Opioid Antagonist Lacking the Basic Center — Models of Antagonism

Orlando Crescenzi, Franca Fraternali, Delia Picone, Teodorico Tancredi, Gianfranco Balboni, Remo Guerrini, Lawrence H. Lazarus, Severe Salvadori, Piero A. Temussi

Journal:

Year:

1997

Language:

english

File:

PDF, 978 KB

english, 1997

38

Alterations in vasoactive intestinal polypeptide-related peptides after pentylenetetrazole-induced seizures in rat brain

Patrizia Romualdi, Giovanni Lesa, Alessandra Donatini, Gianfranco Balboni, Roberto Tomatis, Sergio Ferri

Journal:

European Journal of Pharmacology

Year:

1992

Language:

english

File:

PDF, 469 KB

english, 1992

39

Dmt-Tic-OH, a highly selective and potent δ-opioid dipeptide receptor antagonist after systemic administration in the mouse

Anna Capasso, Remo Guerrini, Gianfranco Balboni, Ludovico Sorrentino, Pierandrea Temussi, Lawrence H. Lazarus, Sharon D. Bryant, Severo Salvadori

Journal:

Year:

1996

Language:

english

File:

PDF, 398 KB

english, 1996

40

Dmt-Tic-NH-CH2-Bid (UFP-502), a potent DOP receptor agonist: In vitro and in vivo studies

Raffaella Vergura, Elena Valenti, Christopher P. Hebbes, Elaine C. Gavioli, Barbara Spagnolo, John McDonald, David G. Lambert, Gianfranco Balboni, Severo Salvadori, Domenico Regoli, Girolamo Calo’

Journal:

Year:

2006

Language:

english

File:

PDF, 439 KB

english, 2006

41

Anxiolytic- and antidepressant-like activities of H-Dmt-Tic-NH-CH(CH2-COOH)-Bid (UFP-512), a novel selective delta opioid receptor agonist

Raffaella Vergura, Gianfranco Balboni, Barbara Spagnolo, Elaine Gavioli, David G. Lambert, John McDonald, Claudio Trapella, Lawrence H. Lazarus, Domenico Regoli, Remo Guerrini, Severo Salvadori, Girol

Journal:

Year:

2008

Language:

english

File:

PDF, 685 KB

english, 2008

42

Opioid pseudopeptides containing heteroaromatic or heteroaliphatic nuclei

Gianfranco Balboni, Severo Salvadori, Remo Guerrini, Clementina Bianchi, Vincenzo Santagada, Giuseppe Calliendo, Sharon D. Bryant, Lawrence H. Lazarus

Journal:

Year:

2000

Language:

english

File:

PDF, 216 KB

english, 2000

43

Synthesis and structure-activity relationships of deltorphins analogs

Salvadori, Severo, Marastoni, Mauro, Balboni, Gianfranco, Borea, Pier Andrea, Morari, Michele, Tomatis, Roberto

Journal:

Journal of Medicinal Chemistry

Year:

1991

Language:

english

File:

PDF, 802 KB

english, 1991

44

New 2‘,6‘-Dimethyl- l -tyrosine (Dmt) Opioid Peptidomimetics Based on the Aba-Gly Scaffold. Development of Unique μ-Opioid Receptor Ligands

Ballet, Steven, Salvadori, Severo, Trapella, Claudio, Bryant, Sharon D., Jinsmaa, Yunden, Lazarus, Lawrence H., Negri, Lucia, Giannini, Elisa, Lattanzi, Roberta, Tourwé, Dirk, Balboni, Gianfranco

Journal:

Journal of Medicinal Chemistry

Year:

2006

Language:

english

File:

PDF, 82 KB

english, 2006

45

Crystal Structures of Dipeptides Containing the Dmt-Tic Pharmacophore

Bryant, Sharon D., George, Clifford, Flippen-Anderson, Judith L., Deschamps, Jeffrey R., Salvadori, Severo, Balboni, Gianfranco, Guerrini, Remo, Lazarus, Lawrence H.

Journal:

Journal of Medicinal Chemistry

Year:

2002

Language:

english

File:

PDF, 226 KB

english, 2002

46

Further Studies on the Dmt-Tic Pharmacophore: Hydrophobic Substituents at the C-Terminus Endow δ Antagonists To Manifest μ Agonism or μ Antagonism

Salvadori, Severo, Guerrini, Remo, Balboni, Gianfranco, Bianchi, Clementina, Bryant, Sharon D., Cooper, Peter S., Lazarus, Lawrence H.

Journal:

Journal of Medicinal Chemistry

Year:

1999

Language:

english

File:

PDF, 126 KB

english, 1999

47

Base-promoted reactions of ?-halogeno-alkylanilides

Cavicchioni, Giorgio, Scrimin, Paolo, Veronese, Augusto C., Balboni, Gianfranco, D'Angeli, Ferruccio

Journal:

Journal of the Chemical Society Perkin Transactions 1

Year:

1982

Language:

english

File:

PDF, 535 KB

english, 1982

48

Ligand- and cell-dependent determinants of internalization and cAMP modulation by delta opioid receptor (DOR) agonists

Charfi, Iness, Nagi, Karim, Mnie-Filali, Ouissame, Thibault, Dominic, Balboni, Gianfranco, Schiller, Peter W., Trudeau, Louis-Eric, Pineyro, Graciela

Journal:

Cellular and Molecular Life Sciences

Year:

2014

Language:

english

File:

PDF, 937 KB

english, 2014

49

A new convenient synthetic method and preliminary pharmacological characterization of triazinediones as prokineticin receptor antagonists

Congiu, Cenzo, Onnis, Valentina, Deplano, Alessandro, Salvadori, Severo, Marconi, Veronica, Maftei, Daniela, Negri, Lucia, Lattanzi, Roberta, Balboni, Gianfranco

Journal:

European Journal of Medicinal Chemistry

Year:

2014

Language:

english

File:

PDF, 582 KB

english, 2014

50

Synthesis and carbonic anhydrase I, II, IX and XII inhibition studies of 4-N,N-disubstituted sulfanilamides incorporating 4,4,4-trifluoro-3-oxo-but-1-enyl, phenacylthiourea and imidazol-2(3H)-one/thione moieties

Congiu, Cenzo, Onnis, Valentina, Balboni, Gianfranco, Supuran, Claudiu T.

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2014

Language:

english

File:

PDF, 367 KB

english, 2014