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1

Synthese von natürlich vorkommendem (−)-Calyculin A

Dr. Norihiko Tanimoto, Dr. Samuel W. Gerritz, Dr. Akiyoshi Sawabe, Dr. Takeshi Noda, Sandra A. Filla, Prof. Satoru Masamune

Journal:

Angewandte Chemie

Year:

1994

Language:

german

File:

PDF, 527 KB

german, 1994

2

The Synthesis of Naturally Occurring ()-Calyculin A

Dr. Norihiko Tánimoto, Dr. Samuel W. Gerritz, Dr. Akiyoshi Sawabe, Dr. Takeshi Noda, Sandra A. Filla, Prof. Satoru Masamune

Journal:

Angewandte Chemie International Edition

Year:

1994

Language:

english

File:

PDF, 355 KB

english, 1994

3

ChemInform Abstract: Two General Routes to 1,4-Disubstituted-2,3,4,5-tetrahydro-1H-3-benzazepines.

Samuel W. Gerritz, Jennifer S. Smith, Suganthini S. Nanthakumar, David E. Uehling, Jeffery E. Cobb

Journal:

Year:

2001

Language:

english

File:

PDF, 37 KB

english, 2001

4

ChemInform Abstract: A Facile One-Step Synthesis of 5-Chloro-imidazo[1-5-a]quinazoline by Microwave Irradiation.

Guo Li, Ramesh Kakarla, Samuel W. Gerritz, Annapurna Pendri, Baoqing Ma

Journal:

Year:

2010

File:

PDF, 41 KB

2010

5

ChemInform Abstract: An Efficient One-Pot Synthesis of 3-Aryl-5-methylisoxazoles from Aryl Aldehydes.

Shirong Zhu, Shuhao Shi, Samuel W. Gerritz

Journal:

Year:

2011

File:

PDF, 30 KB

2011

6

Discovery of pyrazine carboxamide CB1 antagonists: The introduction of a hydroxyl group improves the pharmaceutical properties and in vivo efficacy of the series

Bruce A. Ellsworth, Ying Wang, Yeheng Zhu, Annapurna Pendri, Samuel W. Gerritz, Chongqing Sun, Kenneth E. Carlson, Liya Kang, Rose A. Baska, Yifan Yang, Qi Huang, Neil T. Burford, Mary Jane Cullen, Su

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2007

Language:

english

File:

PDF, 239 KB

english, 2007

7

Solid-phase synthesis of a library based on biphenyl-containing trypsin-like serine protease inhibitors

Shuhao Shi, Shirong Zhu, Samuel W. Gerritz, Bogumila Rachwal, Zheming Ruan, Robert Hutchins, Ramesh Kakarla, Michael J. Sofia, James Sutton, Daniel Cheney

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2009

Language:

english

File:

PDF, 994 KB

english, 2009

8

Solid-phase synthesis and anti-infective activity of a combinatorial library based on the natural product anisomycin

Shuhao Shi, Shirong Zhu, Samuel W. Gerritz, Kim Esposito, Ramesh Padmanabha, Wenying Li, John J. Herbst, Henry Wong, Yue Zhong Shu, Kin S. Lam, Michael J. Sofia

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2005

Language:

english

File:

PDF, 579 KB

english, 2005

9

Discovery and optimization of (R)-prolinol-derived agonists of the Growth Hormone Secretagogue receptor (GHSR)

Weixu Zhai, Neil Flynn, Daniel A. Longhi, Joseph A. Tino, Brian J. Murphy, Dorothy Slusarchyk, David A. Gordon, Anna Pendri, Shuhao Shi, Robert Stoffel, Baoqing Ma, Michael J. Sofia, Samuel W. Gerritz

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2008

Language:

english

File:

PDF, 215 KB

english, 2008

10

A fast and efficient bromination of isoxazoles and pyrazoles by microwave irradiation

Guo Li, Ramesh Kakarla, Samuel W. Gerritz

Journal:

Tetrahedron Letters

Year:

2007

Language:

english

File:

PDF, 222 KB

english, 2007

11

An efficient one-pot synthesis of 3-aryl-5-methylisoxazoles from aryl aldehydes

Shirong Zhu, Shuhao Shi, Samuel W. Gerritz

Journal:

Tetrahedron Letters

Year:

2011

Language:

english

File:

PDF, 1.26 MB

english, 2011

12

Highly selective reducing agents. Reduction of nitrobenzene to aniline in the presence of aldehydes, alkyl halides, and acid halides.

P.L. Gaus, Samuel W. Gerritz, Patrick M. Jeffries

Journal:

Tetrahedron Letters

Year:

1988

Language:

english

File:

PDF, 199 KB

english, 1988

13

Solid-phase synthesis of trisubstituted guanidines

David H. Drewry, Samuel W. Gerritz, James A. Linn

Journal:

Tetrahedron Letters

Year:

1997

Language:

english

File:

PDF, 233 KB

english, 1997

14

Solid phase synthesis of 1,3,5-trisubstituted pyridin-2-ones

James A. Linn, Samuel W. Gerritz, Anthony L. Handlon, Clifton E. Hyman, Dennis Heyer

Journal:

Tetrahedron Letters

Year:

1999

Language:

english

File:

PDF, 283 KB

english, 1999

15

Quantitative techniques for the comparison of solid supports

Samuel W Gerritz

Journal:

Current Opinion in Chemical Biology

Year:

2001

Language:

english

File:

PDF, 69 KB

english, 2001

16

Combinatorial chemistry: Rumors of the demise of combinatorial chemistry are greatly exaggerated

Andrew T Merritt, Samuel W Gerritz

Journal:

Current Opinion in Chemical Biology

Year:

2003

Language:

english

File:

PDF, 49 KB

english, 2003

17

A facile one-step synthesis of 5-chloro-imidazo[1,5-a]quinazoline by microwave irradiation

Guo Li, Ramesh Kakarla, Samuel W. Gerritz, Annapurna Pendri, Baoqing Ma

Journal:

Tetrahedron Letters

Year:

2009

Language:

english

File:

PDF, 1.93 MB

english, 2009

18

Solid phase synthesis of 1,5-disubstituted pyrazole-4-hydroxamic acids and pyrazole-4-carboxamides via direct amidation of β-ketoesters

Weixu Zhai, Samuel W. Gerritz, Michael J. Sofia

Journal:

Tetrahedron Letters

Year:

2012

Language:

english

File:

PDF, 543 KB

english, 2012

19

Acyl Guanidine Inhibitors of β-Secretase (BACE-1): Optimization of a Micromolar Hit to a Nanomolar Lead via Iterative Solid- and Solution-Phase Library Synthesis

Gerritz, Samuel W., Zhai, Weixu, Shi, Shuhao, Zhu, Shirong, Toyn, Jeremy H., Meredith, Jere E., Iben, Lawrence G., Burton, Catherine R., Albright, Charles F., Good, Andrew C., Tebben, Andrew J., Mucke

Journal:

Journal of Medicinal Chemistry

Year:

2012

Language:

english

File:

PDF, 676 KB

english, 2012

20

Synthesis and Applications of a Novel Polymer-Supported EEDQ Reagent

Kakarla, Ramesh, Li, Guo, Gerritz, Samuel W.

Journal:

Journal of Combinatorial Chemistry

Year:

2008

File:

PDF, 16 KB

2008

21

Influenza Nucleoprotein: Promising Target for Antiviral Chemotherapy

Cianci, Christopher, Gerritz, Samuel W, Deminie, Carol, Krystal, Mark

Journal:

Antiviral Chemistry & Chemotherapy

Year:

2012

Language:

english

File:

PDF, 899 KB

english, 2012

22

Small-molecule pyrimidine inhibitors of the cdc2-like (Clk) and dual specificity tyrosine phosphorylation-regulated (Dyrk) kinases: Development of chemical probe ML315

Coombs, Thomas C., Tanega, Cordelle, Shen, Min, Wang, Jenna L., Auld, Douglas S., Gerritz, Samuel W., Schoenen, Frank J., Thomas, Craig J., Aubé, Jeffrey

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2013

Language:

english

File:

PDF, 6.18 MB

english, 2013

23

2,5-Dimethylfuran (DMFu): An Internal Standard for the “Traceless” Quantitation of Unknown Samples via 1 H NMR †

Gerritz, Samuel W., Sefler, Andrea M.

Journal:

Journal of Combinatorial Chemistry

Year:

2000

Language:

english

File:

PDF, 32 KB

english, 2000

24

Solid Phase Synthesis of 1,5-Diarylpyrazole-4-carboxamides: Discovery of Antagonists of the CB-1 Receptor

Pendri, Annapurna, Dodd, Dharmpal S., Chen, Jing, Cvijic, Mary Ellen, Kang, Liya, Baska, Rose A., Carlson, Kenneth E., Burford, Neil T., Sun, Chongqing, Ewing, William R., Gerritz, Samuel W.

Journal:

ACS Combinatorial Science

Year:

2012

Language:

english

File:

PDF, 938 KB

english, 2012

25

Using One- and Two-Dimensional NMR Techniques to Characterize Reaction Products Bound to Chiron SynPhase Crowns

Sefler, Andrea M., Gerritz, Samuel W.

Journal:

Journal of Combinatorial Chemistry

Year:

2000

Language:

english

File:

PDF, 157 KB

english, 2000

26

Solid Phase Synthesis of Novel Pyrrolidinedione Analogs as Potent HIV-1 Integrase Inhibitors

Pendri, Annapurna, Troyer, Timothy L., Sofia, Michael J., Walker, Michael A., Naidu, B. Narasimhulu, Banville, Jacques, Meanwell, Nicholas A., Dicker, Ira, Lin, Zeyu, Krystal, Mark, Gerritz, Samuel W.

Journal:

Journal of Combinatorial Chemistry

Year:

2010

Language:

english

File:

PDF, 1.88 MB

english, 2010

27

Probing the Reactivity of Solid Supports via Hammett Relationships

Gerritz, Samuel W., Trump, Ryan P., Zuercher, William J.

Journal:

Journal of the American Chemical Society

Year:

2000

Language:

english

File:

PDF, 175 KB

english, 2000

28

High-Throughput Manual Parallel Synthesis Using SynPhase Crowns and Lanterns

Gerritz, Samuel W., Norman, Mark H., Barger, Lee A., Berman, Judd, Bigham, Eric C., Bishop, Michael J., Drewry, David H., Garrison, Deanna T., Heyer, Dennis, Hodson, Stephen J., Kakel, Jennifer A., Li

Journal:

Journal of Combinatorial Chemistry

Year:

2003

Language:

english

File:

PDF, 1.09 MB

english, 2003

29

Two General Routes to 1,4-Disubstituted-2,3,4,5-tetrahydro- 1 H -3-benzazepines

Gerritz, Samuel W., Smith, Jennifer S., Nanthakumar, Suganthini S., Uehling, David E., Cobb, Jeffery E.

Journal:

Organic Letters

Year:

2000

Language:

english

File:

PDF, 62 KB

english, 2000

30

Synthesis and Applications of a Novel Polymer-Supported EEDQ Reagent

Kakarla, Ramesh, Li, Guo, Gerritz, Samuel W.

Journal:

Journal of Combinatorial Chemistry

Year:

2007

Language:

english

File:

PDF, 79 KB

english, 2007

31

Attachment of Unreactive Amines to the Solid Support: Synthesis of Phenyl-Substituted Anilines, 2-Aminopyridines, and 2-Aminopyrimidines

Zhu, Shirong, Shi, Shuhao, Gerritz, Samuel W., Sofia, Michael J.

Journal:

Journal of Combinatorial Chemistry

Year:

2003

Language:

english

File:

PDF, 37 KB

english, 2003

32

Ligand-Based Discovery of a New Scaffold for Allosteric Modulation of the μ-Opioid Receptor

Bisignano, Paola, Burford, Neil T., Shang, Yi, Marlow, Brennica, Livingston, Kathryn E., Fenton, Abigail M., Rockwell, Kristin, Budenholzer, Lauren, Traynor, John R., Gerritz, Samuel W., Alt, Andrew,

Journal:

Journal of Chemical Information and Modeling

Year:

2015

Language:

english

File:

PDF, 2.07 MB

english, 2015

33

Biochemical and Behavioral Effects of PDE10A inhibitors: Relationship to Target Site Occupancy

Li, Yu-Wen, Seager, Matthew A., Wojcik, Trevor, Heman, Karen, Molski, Thaddeus F., Fernandes, Alda, Langdon, Shaun, Pendri, Annapurna, Gerritz, Samuel, Tian, Yuan, Hong, Yang, Gallagher, Lizbeth, Merr

Journal:

Neuropharmacology

Year:

2015

Language:

english

File:

PDF, 11.28 MB

english, 2015

34

Macrocyclic prolinyl acyl guanidines as inhibitors of β-secretase (BACE)

Boy, Kenneth M., Guernon, Jason M., Wu, Yong-Jin, Zhang, Yunhui, Shi, Joe, Zhai, Weixu, Zhu, Shirong, Gerritz, Samuel W., Toyn, Jeremy H., Meredith, Jere E., Barten, Donna M., Burton, Catherine R., Al

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2015

Language:

english

File:

PDF, 2.97 MB

english, 2015

35

Inhibition of influenza virus replication via small molecules that induce the formation of higher-order nucleoprotein oligomers

Samuel W. Gerritz, Christopher Cianci, Sean Kim, Bradley C. Pearce, Carol Deminie, Linda Discotto, Brian McAuliffe, Beatrice F. Minassian, Shuhao Shi, Shirong Zhu, Weixu Zhai, Annapurna Pendri, Guo Li

Journal:

Proceedings of the National Academy of Sciences

Year:

2011

Language:

english

File:

PDF, 1.42 MB

english, 2011

36

Structure-Guided Discovery of Positive Allosteric Modulators of the Mu-Opioid Receptor

Bisignano, Paola, Burford, Neil T., Gerritz, Samuel W., Alt, Andrew, Filizola, Marta

Journal:

Biophysical Journal

Year:

2015

Language:

english

File:

PDF, 60 KB

english, 2015

37

Identification and biochemical analyses of selective CB2 agonists

Scott, Caitlin E., Tang, Yaliang, Alt, Andrew, Burford, Neil T., Gerritz, Samuel W., Ogawa, Lisa M., Zhang, Litao, Kendall, Debra A.

Journal:

European Journal of Pharmacology

Year:

2019

Language:

english

File:

PDF, 6.82 MB

english, 2019

38

Rapid Compound Integrity Assessment for High-Throughput Screening Hit Triaging

Shou, Wilson Z., Gerritz, Samuel W., Harden, David, Lawrence, R. Michael, Chase, Peter, Chin, Jefferson, Surti, Neha, Lippy, Jonathan S., Weller, Harold N., Nielsen, Julia, Weerakoon, Darshani

Journal:

Year:

2020

File:

PDF, 582 KB

2020