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51

Correction to Targeting the Binding Function 3 (BF3) Site of the Human Androgen Receptor through Virtual Screening

Lack, Nathan A., Axerio-Cilies, Peter, Tavassoli, Peyman, Han, Frank Q., Chan, Ka Hong, Feau, Clementine, LeBlanc, Eric, Guns, Emma Tomlinson, Guy, R. Kiplin, Rennie, Paul S., Cherkasov, Artem

Journal:

Journal of Medicinal Chemistry

Year:

2012

Language:

english

File:

PDF, 113 KB

english, 2012

52

Synthesis and Evaluation of 7-Substituted 4-Aminoquinoline Analogues for Antimalarial Activity

Hwang, Jong Yeon, Kawasuji, Takashi, Lowes, David J., Clark, Julie A., Connelly, Michele C., Zhu, Fangyi, Guiguemde, W. Armand, Sigal, Martina S., Wilson, Emily B., DeRisi, Joseph L., Guy, R. Kiplin

Journal:

Journal of Medicinal Chemistry

Year:

2011

Language:

english

File:

PDF, 3.56 MB

english, 2011

53

Discovery of the First Irreversible Small Molecule Inhibitors of the Interaction between the Vitamin D Receptor and Coactivators

Nandhikonda, Premchendar, Lynt, Wen Z., McCallum, Megan M., Ara, Tahniyath, Baranowski, Athena M., Yuan, Nina Y., Pearson, Dana, Bikle, Daniel D., Guy, R. Kiplin, Arnold, Leggy A.

Journal:

Journal of Medicinal Chemistry

Year:

2012

Language:

english

File:

PDF, 1.25 MB

english, 2012

54

Antimalarial activity of 10-alkyl/aryl esters and -aminoethylethers of artemisinin

Cloete, Theunis T., Krebs, Henk J., Clark, Julie A., Connelly, Michele C., Orcutt, Amy, Sigal, Martina S., Kiplin Guy, R., N’Da, David D.

Journal:

Bioorganic Chemistry

Year:

2013

Language:

english

File:

PDF, 310 KB

english, 2013

55

Discovery of Novel Antimalarial Compounds Enabled by QSAR-Based Virtual Screening

Zhang, Liying, Fourches, Denis, Sedykh, Alexander, Zhu, Hao, Golbraikh, Alexander, Ekins, Sean, Clark, Julie, Connelly, Michele C., Sigal, Martina, Hodges, Dena, Guiguemde, Armand, Guy, R. Kiplin, Tro

Journal:

Journal of Chemical Information and Modeling

Year:

2013

Language:

english

File:

PDF, 997 KB

english, 2013

56

Optimization of Propafenone Analogues as Antimalarial Leads

Lowes, David J., Guiguemde, W. Armand, Connelly, Michele C., Zhu, Fangyi, Sigal, Martina S., Clark, Julie A., Lemoff, Andrew S., Derisi, Joseph L., Wilson, Emily B., Guy, R. Kiplin

Journal:

Journal of Medicinal Chemistry

Year:

2011

Language:

english

File:

PDF, 1.17 MB

english, 2011

57

Copper-Mediated Cross-Coupling of Aryl Boronic Acids and Alkyl Thiols

Herradura, Prudencio S., Pendola, Kathleen A., Guy, R. Kiplin

Journal:

Organic Letters

Year:

2000

Language:

english

File:

PDF, 116 KB

english, 2000

58

A Solid-Phase Approach to the Phallotoxins: Total Synthesis of [Ala 7 ]-Phalloidin

Anderson, Marc O., Shelat, Anang A., Guy, R. Kiplin

Journal:

Journal of Organic Chemistry

Year:

2005

Language:

english

File:

PDF, 265 KB

english, 2005

59

Synthesis and evaluation of methylsulfonylnitrobenzamides (MSNBAs) as inhibitors of the thyroid hormone receptor–coactivator interaction

Hwang, Jong Yeon, Attia, Ramy R., Carrillo, Angela K., Connelly, Michele C., Guy, R. Kiplin

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2013

Language:

english

File:

PDF, 872 KB

english, 2013

60

Optimization of Chloronitrobenzamides (CNBs) as Therapeutic Leads for Human African Trypanosomiasis (HAT)

Hwang, Jong Yeon, Smithson, David, Zhu, Fangyi, Holbrook, Gloria, Connelly, Michele C., Kaiser, Marcel, Brun, Reto, Guy, R. Kiplin

Journal:

Journal of Medicinal Chemistry

Year:

2013

Language:

english

File:

PDF, 1.23 MB

english, 2013

61

Optimization of the electrophile of chloronitrobenzamide leads active against Trypanosoma brucei

Hwang, Jong Yeon, Smithson, David C., Holbrook, Gloria, Zhu, Fangyi, Connelly, Michele C., Kaiser, Marcel, Brun, Reto, Kiplin Guy, R.

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2013

Language:

english

File:

PDF, 1.98 MB

english, 2013

62

Similarities and Differences between Two Modes of Antagonism of the Thyroid Hormone Receptor

Sadana, Prabodh, Hwang, Jong Yeon, Attia, Ramy R., Arnold, Leggy A., Neale, Geoffrey, Guy, R. Kiplin

Journal:

ACS Chemical Biology

Year:

2011

Language:

english

File:

PDF, 3.86 MB

english, 2011

63

Pharmacokinetics and Efficacy of the Spleen Tyrosine Kinase Inhibitor R406 after Ocular Delivery for Retinoblastoma

Pritchard, Eleanor M., Stewart, Elizabeth, Zhu, Fangyi, Bradley, Cori, Griffiths, Lyra, Yang, Lei, Suryadevara, Praveen Kumar, Zhang, Jiakun, Freeman, Burgess B., Guy, R. Kiplin, Dyer, Michael A.

Journal:

Pharmaceutical Research

Year:

2014

Language:

english

File:

PDF, 993 KB

english, 2014

64

Organocatalytic, Diastereo- and Enantioselective Synthesis of Nonsymmetric cis -Stilbene Diamines: A Platform for the Preparation of Single-Enantiomer cis -Imidazolines for Protein–Protein Inhibition

Vara, Brandon A., Mayasundari, Anand, Tellis, John C., Danneman, Michael W., Arredondo, Vanessa, Davis, Tyler A., Min, Jaeki, Finch, Kristin, Guy, R. Kiplin, Johnston, Jeffrey N.

Journal:

Journal of Organic Chemistry

Year:

2014

Language:

english

File:

PDF, 2.67 MB

english, 2014

65

Structure-Guided Development of Selective TbcatB Inhibitors

Mallari, Jeremy P., Shelat, Anang A., Kosinski, Aaron, Caffrey, Conor R., Connelly, Michele, Zhu, Fangyi, McKerrow, James H., Guy, R. Kiplin

Journal:

Journal of Medicinal Chemistry

Year:

2009

Language:

english

File:

PDF, 3.39 MB

english, 2009

66

Improvement of Pharmacological Properties of Irreversible Thyroid Receptor Coactivator Binding Inhibitors

Hwang, Jong Yeon, Arnold, Leggy A., Zhu, Fangyi, Kosinski, Aaron, Mangano, Thomas J., Setola, Vincent, Roth, Bryan L., Guy, R. Kiplin

Journal:

Journal of Medicinal Chemistry

Year:

2009

Language:

english

File:

PDF, 1.41 MB

english, 2009

67

Parallel Synthesis and Antimalarial Screening of a 4-Aminoquinoline Library

Madrid, Peter B., Wilson, Nathan T., DeRisi, Joseph L., Guy, R. Kiplin

Journal:

Journal of Combinatorial Chemistry

Year:

2004

Language:

english

File:

PDF, 86 KB

english, 2004

68

Novel Flufenamic Acid Analogues as Inhibitors of Androgen Receptor Mediated Transcription

Féau, Clémentine, Arnold, Leggy A., Kosinski, Aaron, Zhu, Fangyi, Connelly, Michele, Guy, R. Kiplin

Journal:

ACS Chemical Biology

Year:

2009

Language:

english

File:

PDF, 1.73 MB

english, 2009

69

Synthesis of Medium Ring Heterocycles Using an Intramolecular Heck Reaction

Arnold, Leggy A., Luo, Wenchen, Guy, R. Kiplin

Journal:

Organic Letters

Year:

2004

Language:

english

File:

PDF, 53 KB

english, 2004

70

Novel Selective Inhibitors of the Interaction of Individual Nuclear Hormone Receptors with a Mutually Shared Steroid Receptor Coactivator 2

Geistlinger, Timothy R., Guy, R. Kiplin

Journal:

Journal of the American Chemical Society

Year:

2003

Language:

english

File:

PDF, 83 KB

english, 2003

71

An α-Helical Peptidomimetic Inhibitor of the HIV-1 Rev−RRE Interaction

Mills, Nicholas L., Daugherty, Matthew D., Frankel, Alan D., Guy, R. Kiplin

Journal:

Journal of the American Chemical Society

Year:

2006

Language:

english

File:

PDF, 127 KB

english, 2006

72

Quantification of the Vitamin D Receptor−Coregulator Interaction †

Teichert, Arnaud, Arnold, Leggy A., Otieno, Steve, Oda, Yuko, Augustinaite, Indre, Geistlinger, Tim R., Kriwacki, Richard W., Guy, R. Kiplin, Bikle, Daniel D.

Journal:

Year:

2009

Language:

english

File:

PDF, 4.08 MB

english, 2009

73

Incorporation of an Intramolecular Hydrogen-Bonding Motif in the Side Chain of 4-Aminoquinolines Enhances Activity against Drug-Resistant P. falciparum

Madrid, Peter B., Liou, Ally P., DeRisi, Joseph L., Guy, R. Kiplin

Journal:

Journal of Medicinal Chemistry

Year:

2008

Language:

english

File:

PDF, 29 KB

english, 2008

74

An Inhibitor of the Interaction of Thyroid Hormone Receptor β and Glucocorticoid Interacting Protein 1

Geistlinger, Timothy R., Guy, R. Kiplin

Journal:

Journal of the American Chemical Society

Year:

2001

Language:

english

File:

PDF, 53 KB

english, 2001

75

Development of a New Generation of 4-Aminoquinoline Antimalarial Compounds Using Predictive Pharmacokinetic and Toxicology Models

Ray, Sunetra, Madrid, Peter B., Catz, Paul, LeValley, Susanna E., Furniss, Michael J., Rausch, Linda L., Guy, R. Kiplin, DeRisi, Joseph L., Iyer, Lalitha V., Green, Carol E., Mirsalis, Jon C.

Journal:

Journal of Medicinal Chemistry

Year:

2010

Language:

english

File:

PDF, 1.20 MB

english, 2010

76

Incorporation of an Intramolecular Hydrogen-Bonding Motif in the Side Chain of 4-Aminoquinolines Enhances Activity against Drug-Resistant P. f alciparum

Madrid, Peter B., Liou, Ally P., DeRisi, Joseph L., Guy, R. Kiplin

Journal:

Journal of Medicinal Chemistry

Year:

2006

Language:

english

File:

PDF, 180 KB

english, 2006

77

Role of Electrostatic Interactions in PDZ Domain Ligand Recognition †

Harris, Baruch Z., Lau, Francis W., Fujii, Naoaki, Guy, R. Kiplin, Lim, Wendell A.

Journal:

Year:

2003

Language:

english

File:

PDF, 348 KB

english, 2003

78

A Novel 2‘-( N -Methylpyridinium Acetate) Prodrug of Paclitaxel Induces Superior Antitumor Responses in Preclinical Cancer Models

Wrasidlo, Wolfgang, Gaedicke, Gerhard, Guy, Rodney Kiplin, Renaud, Johanne, Pitsinos, Emmanuel, Nicolaou, Kyriaco C., Reisfeld, Ralph A., Lode, Holger N.

Journal:

Bioconjugate Chemistry

Year:

2002

Language:

english

File:

PDF, 133 KB

english, 2002

79

Synthesis and Evaluation of Sulfonylnitrophenylthiazoles (SNPTs) as Thyroid Hormone Receptor–Coactivator Interaction Inhibitors

Hwang, Jong Yeon, Attia, Ramy R., Zhu, Fangyi, Yang, Lei, Lemoff, Andrew, Jeffries, Cynthia, Connelly, Michele C., Guy, R. Kiplin

Journal:

Journal of Medicinal Chemistry

Year:

2012

Language:

english

File:

PDF, 1.91 MB

english, 2012

80

Development of Potent Purine-Derived Nitrile Inhibitors of the Trypanosomal Protease TbcatB

Mallari, Jeremy P., Shelat, Anang A., Obrien, Terri, Caffrey, Conor R., Kosinski, Aaron, Connelly, Michele, Harbut, Michael, Greenbaum, Doron, McKerrow, James H., Guy, R. Kiplin

Journal:

Journal of Medicinal Chemistry

Year:

2008

Language:

english

File:

PDF, 1.79 MB

english, 2008

81

Partial Acetylation of Lysine Residues Improves Intraprotein Cross-Linking

Guo, Xin, Bandyopadhyay, Pradipta, Schilling, Birgit, Young, Malin M., Fujii, Naoaki, Aynechi, Tiba, Guy, R. Kiplin, Kuntz, Irwin D., Gibson, Bradford W.

Journal:

Analytical Chemistry

Year:

2008

Language:

english

File:

PDF, 330 KB

english, 2008

82

Antimalarials in Development in 2014

Barnett, David S., Guy, R. Kiplin

Journal:

Chemical Reviews

Year:

2014

Language:

english

File:

PDF, 2.07 MB

english, 2014

83

Optimization of a Non-Radioactive High-Throughput Assay for Decarboxylase Enzymes

Smithson, David C., Shelat, Anang A., Baldwin, Jeffrey, Phillips, Margaret A., Guy, R. Kiplin

Journal:

Assay and Drug Development Technologies

Year:

2010

Language:

english

File:

PDF, 2.38 MB

english, 2010

84

A Facile One-Pot Synthesis of Symmetrical and Unsymmetrical Acetaldehyde Acetals from Primary Alcohols

Guy, Rodney Kiplin, DiPietro, Richard Anthony

Journal:

Synthetic Communications

Year:

1992

Language:

english

File:

PDF, 189 KB

english, 1992

85

Interrogating alkyl and arylalkylpolyamino (bis)urea and (bis)thiourea isosteres as potent antimalarial chemotypes against multiple lifecycle forms of Plasmodium falciparum parasites

Verlinden, Bianca K., de Beer, Marna, Pachaiyappan, Boobalan, Besaans, Ethan, Andayi, Warren A., Reader, Janette, Niemand, Jandeli, van Biljon, Riette, Guy, Kiplin, Egan, Timothy, Woster, Patrick M.,

Journal:

Bioorganic & Medicinal Chemistry

Year:

2015

Language:

english

File:

PDF, 1.47 MB

english, 2015

86

Evaluation of histone deacetylase inhibitors (HDACi) as therapeutic leads for human African trypanosomiasis (HAT)

Carrillo, Angela K., Guiguemde, W. Armand, Guy, R. Kiplin

Journal:

Bioorganic & Medicinal Chemistry

Year:

2015

Language:

english

File:

PDF, 999 KB

english, 2015

87

Potent Plasmodium falciparum Gametocytocidal Activity of Diaminonaphthoquinones, Lead Antimalarial Chemotypes Identified in an Antimalarial Compound Screen

Tanaka, Takeshi Q, Guiguemde, W. Armand, Barnett, David S., Maron, Maxim I., Min, Jaeki, Connelly, Michele C., Suryadevara, Praveen Kumar, Guy, R. Kiplin, Williamson, Kim C.

Journal:

Antimicrobial Agents and Chemotherapy

Year:

2015

Language:

english

File:

PDF, 2.14 MB

english, 2015

88

Anticancer Properties of Distinct Antimalarial Drug Classes

Hooft van Huijsduijnen, Rob, Guy, R. Kiplin, Chibale, Kelly, Haynes, Richard K., Peitz, Ingmar, Kelter, Gerhard, Phillips, Margaret A., Vennerstrom, Jonathan L., Yuthavong, Yongyuth, Wells, Timothy N.

Journal:

Year:

2013

Language:

english

File:

PDF, 3.51 MB

english, 2013

89

LC-MS- and 1 H NMR Spectroscopy-Guided Identification of Antifungal Diterpenoids from Sagittaria latifolia

Ravu, Ranga Rao, Jacob, Melissa R., Jeffries, Cynthia, Tu, Ying, Khan, Shabana I., Agarwal, Ameeta K., Guy, R. Kiplin, Walker, Larry A., Clark, Alice M., Li, Xing-Cong

Journal:

Journal of Natural Products

Year:

2015

Language:

english

File:

PDF, 752 KB

english, 2015

90

A Convenient Procedure for Parallel Ester Hydrolysis

Anderson, Marc O., Moser, Jamie, Sherrill, John, Guy, R. Kiplin

Journal:

Year:

2004

Language:

english

File:

PDF, 94 KB

english, 2004

91

Structural Insight into the Mode of Action of a Direct Inhibitor of Coregulator Binding to the Thyroid Hormone Receptor

Estébanez-Perpiñá, Eva, Arnold, Leggy A., Jouravel, Natalia, Togashi, Marie, Blethrow, Justin, Mar, Ellena, Nguyen, Phuong, Phillips, Kevin J., Baxter, John D., Webb, Paul, Guy, R. Kiplin, Fletterick,

Journal:

Molecular Endocrinology

Year:

2007

Language:

english

File:

PDF, 479 KB

english, 2007

92

Pentacyclic nitrofurans that rapidly kill nifurtimox-resistant trypanosomes

Bruhn, David F., Wyllie, Susan, Rodríguez-Cortés, Adaris, Carrillo, Angela K., Rakesh,, Guy, Kiplin, Fairlam, Alan H., Lee, Richard E.

Journal:

Journal of Antimicrobial Chemotherapy

Year:

2015

Language:

english

File:

PDF, 464 KB

english, 2015

93

Monitoring ligand-induced protein ordering in drug discovery

Grace, Christy R., Ban, David, Min, Jaeki, Mayasundari, Anand, Min, Lie, Finch, Kristin E., Griffiths, Lyra, Bharatham, Nagakumar, Bashford, Donald, Kiplin Guy, R., Dyer, Michael A., Kriwacki, Richard

Journal:

Journal of Molecular Biology

Year:

2016

Language:

english

File:

PDF, 834 KB

english, 2016

94

Current and emerging therapy for improving outcomes in patients with intraocular retinoblastoma

Brennan, Rachel C, Pritchard, Eleanor M, Guy, R Kiplin, Dyer, Michael A, Wilson, Matthew W

Journal:

Expert Opinion on Orphan Drugs

Year:

2015

Language:

english

File:

PDF, 836 KB

english, 2015

95

Evaluation of artemisinins for the treatment of acute myeloid leukemia

Drenberg, Christina D., Buaboonnam, Jassada, Orwick, Shelley J., Hu, Shuiying, Li, Lie, Fan, Yiping, Shelat, Anang A., Guy, R. Kiplin, Rubnitz, Jeffrey, Baker, Sharyn D.

Journal:

Cancer Chemotherapy and Pharmacology

Year:

2016

Language:

english

File:

PDF, 4.29 MB

english, 2016

96

ChemInform Abstract: Organocatalytic, Diastereo- and Enantioselective Synthesis of Nonsymmetric cis-Stilbene Diamines: A Platform for the Preparation of Single-Enantiomer cis-Imidazolines for Protein-Protein Inhibition.

Vara, Brandon A., Mayasundari, Anand, Tellis, John C., Danneman, Michael W., Arredondo, Vanessa, Davis, Tyler A., Min, Jaeki, Finch, Kristin, Guy, R. Kiplin, Johnston, Jeffrey N.

Journal:

Year:

2015

Language:

english

File:

PDF, 32 KB

english, 2015

97

Flexibility is important for inhibition of the MDM2/p53 protein–protein interaction by cyclic β-hairpins

Danelius, Emma, Pettersson, Mariell, Bred, Matilda, Min, Jaeki, Waddell, M. Brett, Guy, R. Kiplin, Grøtli, Morten, Erdelyi, Mate

Journal:

Organic & Biomolecular Chemistry

Year:

2016

Language:

english

File:

PDF, 908 KB

english, 2016

98

Performance of a docking/molecular dynamics protocol for virtual screening of nutlin-class inhibitors of Mdmx

Bharatham, Nagakumar, Finch, Kristin E., Min, Jaeki, Mayasundari, Anand, Dyer, Michael A., Guy, R. Kiplin, Bashford, Donald

Journal:

Journal of Molecular Graphics and Modelling

Year:

2017

Language:

english

File:

PDF, 457 KB

english, 2017

99

Shared Consensus Machine Learning Models for Predicting Blood Stage Malaria Inhibition

Verras, Andreas, Waller, Chris L., Gedeck, Peter, Green, Darren V. S., Kogej, Thierry, Raichurkar, Anandkumar, Panda, Manoranjan, Shelat, Anang A., Clark, Julie, Guy, R. Kiplin, Papadatos, George, Bur

Journal:

Journal of Chemical Information and Modeling

Year:

2017

Language:

english

File:

PDF, 1.34 MB

english, 2017

100

Seeking the Elusive Long-Acting Ozonide: Discovery of Artefenomel (OZ439)

Kim, Ho Shin, Hammill, Jared T., Guy, R. Kiplin

Journal:

Journal of Medicinal Chemistry

Year:

2017

Language:

english

File:

PDF, 643 KB

english, 2017

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