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51

Synthesis of [3H](4-fluorobutyl)propyl[2,5,6-trimethyl-7-(2,4,6-trimethylphenyl)pyrrolo[2,3-d]pyrimidin-4-yl]amine: a potent radioligand for corticotropin-releasing hormone type 1 receptor

Ling-Wei Hsin, Elizabeth L. Webster, George P. Chrousos, Philip W. Gold, William C. Eckelman, Carlo Contoreggi, Kenner C. Rice

Journal:

Journal of Labelled Compounds and Radiopharmaceuticals

Year:

2000

File:

PDF, 413 KB

2000

52

ChemInform Abstract: L-Selectride as a Convenient Reagent for the Selective Cleavage of Carbamates.

Andrew Coop, Kenner C. Rice

Journal:

Year:

1999

File:

PDF, 28 KB

1999

53

ChemInform Abstract: A Novel Synthesis of Thebaine from Codeine.

Andrew Coop, Kenner C. Rice

Journal:

Year:

1999

File:

PDF, 25 KB

1999

54

ChemInform Abstract: Direct Oxidation of Codeinone to 14-Hydroxycodeinone

Andrew Coop, Kenner C. Rice

Journal:

Year:

2000

File:

PDF, 26 KB

2000

55

ChemInform Abstract: Probes for Narcotic Receptor Mediated Phenomena. Part 26. Synthesis and Biological Evaluation of Diarylmethylpiperazines and Diarylmethylpiperidines as Novel, Nonpeptidic δ Opioid Receptor Ligands.

Kenner C. Rice, et al. et al.

Journal:

Year:

2000

File:

PDF, 32 KB

2000

56

ChemInform Abstract: Delta Opioid Binding Selectivity of 3-Ether Analogues of Naltrindole.

Andrew Coop, Julia Pinto, Lijuan Wang, Karen McCullough, Richard B. Rothman, Christine Dersch, Arthur E. Jacobsen, Kenner C. Rice

Journal:

Year:

2000

File:

PDF, 33 KB

2000

57

ChemInform Abstract: Synthesis and Biological Activity of Fluoro-Substituted Pyrrolo[2,3-d]pyrimidines. The Development of Potential Positron Emission Tomography Imaging Agents for the Corticotropin-Releasing Hormone Type 1 Receptor.

Ling-Wei Hsin, Elizabeth L. Webster, George P. Chrousos, Philip W. Gold, William C. Eckelman, Carlo Contoreggi, Kenner C. Rice

Journal:

Year:

2000

File:

PDF, 33 KB

2000

58

ChemInform Abstract: Design, Synthesis, and Monoamine Transporter Binding Site Affinities of Methoxy Derivatives of Indatraline.

Xiao-Hui Gu, Han Yu, Arthur E. Jacobson, Richard B. Rothman, Christina M. Dersch, Clifford George, Judith L. Flippen-Anderson, Kenner C. Rice

Journal:

Year:

2001

File:

PDF, 30 KB

2001

59

ChemInform Abstract: Synthesis and Transporter Binding Properties of Bridged Piperazine Analogues of 1-{2-[Bis(4-fluorophenyl)methoxy]ethyl}-4-(3-phenylpropyl)piperazine (GBR 12909).

Ying Zhang, Richard B. Rothman, Christina M. Dersch, Brian R. de Costa, Arthur E. Jacobson, Kenner C. Rice

Journal:

Year:

2001

File:

PDF, 36 KB

2001

60

ChemInform Abstract: The Development of a Potential Single Photon Emission Computed Tomography (SPECT) Imaging Agent for the Corticotropin-Releasing Hormone Receptor Type 1

Kenner C. Rice, et al. et al.

Journal:

Year:

2001

File:

PDF, 28 KB

2001

61

ChemInform Abstract: Derivatives of 17-(2-Methylallyl)-substituted Noroxymorphone: Variation of the Delta Address and Its Effects on Affinity and Selectivity for the Delta Opioid Receptor.

Thomas Ullrich, Christina M. Dersch, Richard B. Rothman, Arthur E. Jacobson, Kenner C. Rice

Journal:

Year:

2002

File:

PDF, 37 KB

2002

62

ChemInform Abstract: CRHR1 Receptor Binding and Lipophilicity of Pyrrolopyrimidines, Potential Nonpeptide Corticotropin-Releasing Hormone Type 1 Receptor Antagonists.

Kenner C. Rice, et al. et al.

Journal:

Year:

2002

File:

PDF, 29 KB

2002

63

Synthesis and Dopamine Transporter Affinity of Chiral 1-[2-[Bis(4-fluorophenyl)methoxy]ethyl]-4-(2-hydroxypropyl)piperazines as Potential Cocaine Abuse Therapeutic Agents.

Ling-Wei Hsin, Thomas Prisinzano, Chavon R. Wilkerson, Christina M. Dersch, Robert Horel, Arthur E. Jacobson, Richard B. Rothman, Kenner C. Rice

Journal:

Year:

2003

File:

PDF, 115 KB

2003

64

1-(Phenyl)isoquinoline Carboxamides: A Novel Class of Subtype Selective Inhibitors of Thyrotropin-Releasing Hormone (TRH) Receptors.

Jian-kang Jiang, Craig J. Thomas, Susanne Neumann, Xinping Lu, Kenner C. Rice, Marvin C. Gershengorn

Journal:

Year:

2005

File:

PDF, 19 KB

2005

65

ChemInform Abstract: Probes for Narcotic Receptor Mediated Phenomena. Part 38. An Expeditious Synthesis of rac-cis-4a-Ethyl-2-methyl-1,2,3,4,4a,9a-hexahydrobenzofuro [2,3-c]pyridin-6-ol and rac-cis-2-Methyl-4a-phenethyl-1,2,3,4,4a,9a-hexahydrobenzofuro [2,3-c]pyridin-6-ol.

Malliga R. Iyer, Jeffrey R. Deschamps, Arthur E. Jacobson, Kenner C. Rice

Journal:

Year:

2009

File:

PDF, 34 KB

2009

66

Distribution of opiate receptor subtypes and enkephalin and dynorphin immunoreactivity in the hippocampus of squirrel, guinea pig, rat, and hamster

Stafford McLean, Richard B. Rothman, Arthur E. Jacobson, Kenner C. Rice, Miles Herkenham

Journal:

The Journal of Comparative Neurology

Year:

1987

Language:

english

File:

PDF, 2.02 MB

english, 1987

67

The Oxidation of Thebaine with m-Chloroperbenzoic Acid. Studies in the (+)-Morphinan Series. III

Ikuo Iijima, Kenner C. Rice, Arnold Brossi

Journal:

Helvetica Chimica Acta

Year:

1977

Language:

english

File:

PDF, 160 KB

english, 1977

68

Structure Determination of Brominated Morphinan-6-ones by 13C-NMR. Spectroscopy: A novel closure of the oxygen bridge using 4-acetoxymorphinan-6-ones

Arnold Brossi, Fu-Lian Hsu, Kenner C. Rice, Maria D. Rozwadowska, Helmut Schmidhammer, Charles D. Hufford, Chian Chian Chiang, Isabella L. Karle

Journal:

Helvetica Chimica Acta

Year:

1981

Language:

english

File:

PDF, 612 KB

english, 1981

69

Probes for Narcotic Receptor Mediated Phenomena : Synthesis of rac-(3R,6aS,11aR)-1,3,4,5,6,11a-Hexahydro-2-methyl-2H-3,6a-methanobenzofuro[2,3-c]azocin-8-ol, an Epoxy Isomer of 5-Phenylmorphan

Joannes T. M. Linders, Seid Mirsadeghi, Judith L. Flippen-Anderson, Clifford George, Arthur E. Jacobson, Kenner C. Rice

Journal:

Helvetica Chimica Acta

Year:

2003

Language:

english

File:

PDF, 162 KB

english, 2003

70

The high specific activity tritium labeling of the ganglion-blocking nicotinic antagonist chlorisondamine

Josef Zezula, Hay-Yan J. Wang, Amina S. Woods, Roy A. Wise, Arthur E. Jacobson, Kenner C. Rice

Journal:

Journal of Labelled Compounds and Radiopharmaceuticals

Year:

2006

Language:

english

File:

PDF, 111 KB

english, 2006

71

Synthesis of [3H]-labelled 4-[Ethyl[2,5,6-trimethyl-7-(2,4,6-trimethylphenyl)pyrrolo[2,3-d]pyrimidin-4-yl]amino]-2,3-[3H]-butan-1-ol: a high affinity radioligand for the corticotropin-releasing hormone type 1 receptor

Anne-Cécile Hiebel, John S. Partilla, Richard B. Rothman, Arthur E. Jacobson, Kenner C. Rice

Journal:

Journal of Labelled Compounds and Radiopharmaceuticals

Year:

2006

Language:

english

File:

PDF, 117 KB

english, 2006

72

Probes for narcotic receptor mediated phenomena 8. Tritiation of irreversible mu or delta specific opioid receptor affinity ligands to high specific activity

Terrence R. Burke Jr., Kenner C. Rice, Arthur E. Jacobson, William F. Simonds, Werner A. Klee

Journal:

Journal of Labelled Compounds and Radiopharmaceuticals

Year:

1984

Language:

english

File:

PDF, 381 KB

english, 1984

73

Synthesis of carbon-14 labeled (±)-2-methyl-3,3-diphenyl-3-propanolamine (2-MDP)

Brian De Costa, Andrew Thurkauf, Arthur E. Jacobson, Kenner C. Rice

Journal:

Journal of Labelled Compounds and Radiopharmaceuticals

Year:

1988

Language:

english

File:

PDF, 150 KB

english, 1988

74

Radiochemical synthesis of [18F]fluorothienyl cyclohexylpiperidine [18F]FTCP

Dale O. Kiesewetter, Kenner C. Rice, Marlena V. Mattson, Ronald D. Finn

Journal:

Journal of Labelled Compounds and Radiopharmaceuticals

Year:

1989

Language:

english

File:

PDF, 81 KB

english, 1989

75

Radiochemical synthesis of [18F]-fluorothienylcyclohexylpiperidine ([18F]FTCP)

Dale O. Kiesewetter, Kenner C. Rice, Mariena V. Matson, Ronald D. Finn

Journal:

Journal of Labelled Compounds and Radiopharmaceuticals

Year:

1989

Language:

english

File:

PDF, 393 KB

english, 1989

76

Synthesis of tritium labelled (–)–U50,488, a selective kappa opioid agonist

Andrew Thurkauf, Brian De Gosta, Kenner C. Rice

Journal:

Journal of Labelled Compounds and Radiopharmaceuticals

Year:

1989

Language:

english

File:

PDF, 227 KB

english, 1989

77

Synthesis of tritium labelled 4-fluoro-1-[1–(2-thienyl)]cyclohexylpiperidine ([3H]-FTCP); a tool for autoradiographic study of the phencyclidine binding site

Andrew Thurkauf, Brian R. De Costa, Dale O. Kiesewetter, Arthur E. Jacobson, Kenner C. Rice

Journal:

Journal of Labelled Compounds and Radiopharmaceuticals

Year:

1989

Language:

english

File:

PDF, 270 KB

english, 1989

78

Synthesis of high specific activity tritium labelled 1S,2S-(-)-trans-2-isothiocyanato-N-methyl-N-[2-(1-pyrrolidinyl)-cyclohexyl]benzeneacetamide, a specific irreversible ligand for kappa opioid receptors

Brian R. De Costa, Andew Thurkauf, Richard R. Rothman, Arthur E. Jacobson, Kenner C. Rice

Journal:

Journal of Labelled Compounds and Radiopharmaceuticals

Year:

1990

Language:

english

File:

PDF, 383 KB

english, 1990

79

An expedient synthesis of high specific activity tritium labelled 4-fluoro-1-[1-(2-thienyl)]cyclohexylpiperidine ([3H]FTCP), a ligand for further characterization of the phencyclidine/NMDA receptor complex

Neile A. Grayson, Brian R. de Costa, Joannes T. M. Linders, Kenner C. Rice

Journal:

Journal of Labelled Compounds and Radiopharmaceuticals

Year:

1991

Language:

english

File:

PDF, 319 KB

english, 1991

80

Synthesis of unlabelled and tritium labelled 4-isothiocyanato-1-(1-phenylcyclohexyl)piperidine (fourphit), tools for the study of the dopamine reuptake complex.

Joannes T. M. Linders, Brian R. de Costa, Neile A. Grayson, Kenner C. Rice

Journal:

Journal of Labelled Compounds and Radiopharmaceuticals

Year:

1992

Language:

english

File:

PDF, 656 KB

english, 1992

81

Synthesis of [3H]tert-butyl 8-chloro-5,6-dihydro-5-methyl-6-oxo-4h-imidazo[1,5-a][1,4]benzodiazepine 3-carboxylate, a selective, high affinity ligand for the diazepam insensitive (DI) subtype of the benzodiazepine receptor

Zi-Qiang Gu, Brian R. de Costa, Garry Wong, Kenner C. Rice, Phil Skolnick

Journal:

Journal of Labelled Compounds and Radiopharmaceuticals

Year:

1992

Language:

english

File:

PDF, 388 KB

english, 1992

82

Synthesis of [123I]tert-butyl 8-iodo-5,6-dihydro-5-methyl-6-oxo-4H-imidazo[1,5-a][1,4]benzodiazepine 3-carboxylate, a potential SPECT imaging agent for diazepam-insensitive (DI) benzodiazepine receptors

Xiao-Shu He, Dorota Matecka, Kan Sam Lee, Zi-Qiang Gu, Kenner C. Rice, Garry Wong, Phil Skolnick, Brian R. De Costa

Journal:

Journal of Labelled Compounds and Radiopharmaceuticals

Year:

1994

Language:

english

File:

PDF, 355 KB

english, 1994

83

2,5-dimethyl-2′-hydroxy-9α- and 9β-(3-methylbutyl)-6,7-benzomorphans and n-substituted compounds in the 9α-(3-methylbutyl) series: Chemistry, pharmacology, and biochemistry

Arthur E. Jacobson, Kenner C. Rice, Terrence R. Burke Jr., Lillian Lupinacci, Mariena V. Mattson, Mario D. Aceto, Louis S. Harris

Journal:

Journal of Pharmaceutical Sciences

Year:

1987

Language:

english

File:

PDF, 560 KB

english, 1987

84

Carbon-13 n.m.r. studies of some saturated 1,2-oxazepine derivatives

Kenner C. Rice, Roderick E. Wasylishen

Journal:

Magnetic Resonance in Chemistry

Year:

1976

Language:

english

File:

PDF, 475 KB

english, 1976

85

Radiosynthesis of [18F]3-acetylcyclofoxy: a high affinity opiate antagonist

Michael A. Channing, William C. Eckelman, Jean M. Bennett, Terrence R. Burke Jr., Kenner C. Rice

Journal:

The International Journal of Applied Radiation and Isotopes

Year:

1985

Language:

english

File:

PDF, 439 KB

english, 1985

86

A novel and facile preparation of bremazocine enantiomers through optically pure N-norbremazocines

Elisabeth Greiner, John E Folk, Arthur E Jacobson, Kenner C Rice

Journal:

Bioorganic & Medicinal Chemistry

Year:

2004

Language:

english

File:

PDF, 197 KB

english, 2004

87

A critical structural determinant of opioid receptor interaction with phenolic 5-phenylmorphans

In Jong Kim, Christina M Dersch, Richard B Rothman, Arthur E Jacobson, Kenner C Rice

Journal:

Bioorganic & Medicinal Chemistry

Year:

2004

Language:

english

File:

PDF, 338 KB

english, 2004

88

Structure–activity relationships of substituted N-benzyl piperidines in the GBR series: Synthesis of 4-(2-(bis(4-fluorophenyl)methoxy)ethyl)-1-(2-trifluoromethylbenzyl)piperidine, an allosteric modulator of the serotonin transporter

Terrence L. Boos, Elisabeth Greiner, W. Jason Calhoun, Thomas E. Prisinzano, Barbara Nightingale, Christina M. Dersch, Richard B. Rothman, Arthur E. Jacobson, Kenner C. Rice

Journal:

Bioorganic & Medicinal Chemistry

Year:

2006

Language:

english

File:

PDF, 181 KB

english, 2006

89

Probes for narcotic receptor mediated phenomena. Part 42: Synthesis and in vitro pharmacological characterization of the N-methyl and N-phenethyl analogues of the racemic ortho-c and para-c oxide-bridged phenylmorphans

Jin-Hee Kim, Jeffrey R. Deschamps, Richard B. Rothman, Christina M. Dersch, John E. Folk, Kejun Cheng, Arthur E. Jacobson, Kenner C. Rice

Journal:

Bioorganic & Medicinal Chemistry

Year:

2011

Language:

english

File:

PDF, 697 KB

english, 2011

90

PET imaging of opiate receptor binding in human epilepsy using [18F]cyclofoxy

William H. Theodore, Richard E. Carson, Paul Andreasen, Allan Zametkin, Ron Blasberg, Deborah B. Leiderman, Kenner Rice, Amy Newman, Michael Channing, Bonnie Dunn, Norman Simpson, Peter Herscovitch

Journal:

Epilepsy Research

Year:

1992

Language:

english

File:

PDF, 947 KB

english, 1992

91

DAT/SERT selectivity of flexible GBR 12909 analogs modeled using 3D-QSAR methods

Kathleen M. Gilbert, Terrence L. Boos, Christina M. Dersch, Elisabeth Greiner, Arthur E. Jacobson, David Lewis, Dorota Matecka, Thomas E. Prisinzano, Ying Zhang, Richard B. Rothman, Kenner C. Rice, Ca

Journal:

Bioorganic & Medicinal Chemistry

Year:

2007

Language:

english

File:

PDF, 586 KB

english, 2007

92

Probes for narcotic receptor mediated phenomena. 40. N-Substituted cis-4a-ethyl-1,2,3,4,4a,9a-hexahydrobenzofuro[2,3-c]pyridin-8-ols

Malliga R. Iyer, Yong Sok Lee, Jeffrey R. Deschamps, Richard B. Rothman, Christina M. Dersch, Arthur E. Jacobson, Kenner C. Rice

Journal:

Bioorganic & Medicinal Chemistry

Year:

2010

Language:

english

File:

PDF, 673 KB

english, 2010

93

1-(Phenyl)isoquinoline carboxamides: a novel class of subtype selective inhibitors of thyrotropin-releasing hormone (TRH) receptors

Jian-kang Jiang, Craig J. Thomas, Susanne Neumann, Xinping Lu, Kenner C. Rice, Marvin C. Gershengorn

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2005

Language:

english

File:

PDF, 280 KB

english, 2005

94

A concise synthesis of (S)-(+)-1-(4-{2-[bis-(4-fluorophenyl)methoxy]-ethyl}piperazin-1-yl)-2-phenylpropan-2-ol dimaleate

Thomas Prisinzano, Ling-Wei Hsin, John E. Folk, Judith L. Flippen-Anderson, Clifford George, Arthur E. Jacobson, Kenner C. Rice

Journal:

Tetrahedron: Asymmetry

Year:

2003

Language:

english

File:

PDF, 289 KB

english, 2003

95

Probes for narcotic receptor mediated phenomena. Part 31: Synthesis of rac-(3R,6aS,11aS)-2-methyl-1,3,4,5,6,11a-hexahydro-2H-3,6a-methanobenzofuro[2,3-c]azocine-10-ol, and azocine-8-ol, the ortho-c and the para-c oxide-bridged phenylmorphan isomers

Dragana Tadic, Joannes T.M Linders, Judith L Flippen-Anderson, Arthur E Jacobson, Kenner C Rice

Journal:

Year:

2003

Language:

english

File:

PDF, 495 KB

english, 2003

96

The reaction of dimethyl β-ketoglutarate with 1,2-dicarbonyl compounds. III. Exo-tetracyclo[5.5.1.02,6.010,13]tridecane-4,8,12-trione

Kenner C. Rice, Norman E. Sharpless, Ulrich Weiss, Robert J. Highet

Journal:

Tetrahedron Letters

Year:

1975

Language:

english

File:

PDF, 182 KB

english, 1975

97

Identification of the so-called triacetonehydroxylamine as hexahydro-3,3,7,7-tetramethyl-1,2-oxazepine-5-one.

Kenner C. Rice, Ulrich Weiss

Journal:

Tetrahedron Letters

Year:

1973

Language:

english

File:

PDF, 176 KB

english, 1973

98

Palladium-catalyzed cyanation of hindered, electron-rich aryl triflates by zinc cyanide

Hitoshi Kubota, Kenner C. Rice

Journal:

Tetrahedron Letters

Year:

1998

Language:

english

File:

PDF, 186 KB

english, 1998

99

L-Selectride as a convenient reagent for the selective cleavage of carbamates

Andrew Coop, Kenner C. Rice

Journal:

Tetrahedron Letters

Year:

1998

Language:

english

File:

PDF, 135 KB

english, 1998

100

An expedient synthesis of 9-keto-2-methyl-5-(dimethoxyphenyl)morphans

Joannes T.M Linders, Judith L Flippen-Anderson, Clifford F George, Kenner C Rice

Journal:

Tetrahedron Letters

Year:

1999

Language:

english

File:

PDF, 199 KB

english, 1999