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51

First Synthesis of Arylpyrrolo- and Pyrazolopyrrolizinones as Useful Agents with Potential Biological Interest.

Christophe Rochais, Vincent Lisowski, Patrick Dallemagne, Sylvain Rault

Journal:

Year:

2004

File:

PDF, 17 KB

2004

52

Synthesis of ortho-Substituted Cyanopyridines Through Lithio Intermediate Trapping.

Thomas Cailly, Frederic Fabis, Stephane Lemaitre, Alexandre Bouillon, Sylvain Rault

Journal:

Year:

2005

File:

PDF, 26 KB

2005

53

Efficient Synthesis of Halohydroxypyridines by Hydroxydeboronation.

Anne Sophie Voisin, Alexandre Bouillon, Jean-Charles Lancelot, Sylvain Rault

Journal:

Year:

2005

File:

PDF, 28 KB

2005

54

Solution-Phase Parallel Synthesis of a 1140-Member Ureidothiophene Carboxylic Acid Library.

Francois-Xavier Le Foulon, Emmanuelle Braud, Frederic Fabis, Jean-Charles Lancelot, Sylvain Rault

Journal:

Year:

2005

File:

PDF, 17 KB

2005

55

3D-QSAR and Docking Studies of Selective GSK-3β Inhibitors. Comparison with a Thieno[2,3-b]pyrrolizinone Derivative, a New Potential Lead for GSK-3β Ligands.

Elodie Lescot, Ronan Bureau, Jana Sopkova-de Oliveira Santos, Christophe Rochais, Vincent Lisowski, Jean-Charles Lancelot, Sylvain Rault

Journal:

Year:

2005

File:

PDF, 9 KB

2005

56

Sequential Sonogashira and Suzuki Cross-Coupling Reactions in the Indole and Indazole Series.

Bernhard Witulski, Javier Ramon Azcon, Carole Alayrac, Anca Arnautu, Valerie Collot, Sylvain Rault

Journal:

Year:

2005

File:

PDF, 33 KB

2005

57

Molecular Modeling Studies Focused on 5-HT7 versus 5-HT1A Selectivity. Discovery of Novel Phenylpyrrole Derivatives with High Affinity for 5-HT7 Receptors.

Alban Lepailleur, Ronan Bureau, Magalie Paillet-Loilier, Frederic Fabis, Nicolas Saettel, Stephane Lemaitre, Francois Dauphin, Aurelien Lesnard, Jean-Charles Lancelot, Sylvain Rault

Journal:

Year:

2005

File:

PDF, 8 KB

2005

58

Direct Synthesis of New Arylanthranilic Acids via a Suzuki Cross-Coupling Reaction from Iodoisatins.

Anne-Laure Gerard, Vincent Lisowski, Sylvain Rault

Journal:

Year:

2005

File:

PDF, 25 KB

2005

59

Phenylpyrroles, a New Chemolibrary Virtual Screening Class of 5-HT7 Receptor Ligands.

Magalie Paillet-Loilier, Frederic Fabis, Alban Lepailleur, Ronan Bureau, Sabrina Butt-Gueulle, Francois Dauphin, Catherine Delarue, Hubert Vaudry, Sylvain Rault

Journal:

Year:

2006

File:

PDF, 12 KB

2006

60

ChemInform Abstract: Protected Indazole Boronic Acid Pinacolyl Esters: Facile Syntheses and Studies of Reactivities in Suzuki—Miyaura Cross-Coupling and Hydroxydeboronation Reactions.

Francois Cresty, Elodie Lohou, Silvia Stiebing, Valerie Collot, Sylvain Rault

Journal:

Year:

2009

File:

PDF, 27 KB

2009

61

ChemInform Abstract: Synthesis of New Dipyrrolo- and Furopyrrolopyrazinones Related to Tripentones and Their Biological Evaluation as Potential Kinases (CDKs1—5, GSK-3) Inhibitors.

Christophe Rochais, Nghie Vu Duc, Elodie Lescot, Jana Sopkova-de Oliveira Santos, Ronan Bureau, Laurent Meijer, Patrick Dallemagne, Sylvain Rault

Journal:

Year:

2009

File:

PDF, 31 KB

2009

62

ChemInform Abstract: Synthesis of Dihalo Bi- and Terpyridines by Regioselective Suzuki—Miyaura Cross-Coupling Reactions.

Gregory Burzicki, Anne Sophie Voisin-Chiret, Jana Sopkova-de Oliveira Santos, Sylvain Rault

Journal:

Year:

2009

File:

PDF, 32 KB

2009

63

ChemInform Abstract: Synthesis of 5-Arylthiazoles. Comparative Study Between Suzuki Cross-Coupling Reaction and Direct Arylation.

Nicolas Primas, Alexandre Bouillon, Jean-Charles Lancelot, Hussein El-Kashef, Sylvain Rault

Journal:

Year:

2009

File:

PDF, 33 KB

2009

64

ChemInform Abstract: Synthesis of 2-TIPS-Oxazol-5-ylboronic Acid Pinacol Ester: Efficient Route to 5-(Het)aryloxazoles via Suzuki Cross-Coupling Reaction.

Nicolas Primas, Alexandre Bouillon, Jean-Charles Lancelot, Sylvain Rault

Journal:

Year:

2009

File:

PDF, 45 KB

2009

65

ChemInform Abstract: An Expedient One-Pot Synthesis of Novel 10-Substituted 9-Aminophenanthrenes.

Christophe Rochais, Rodrigue Yougnia, Patrick Dallemagne, Sylvain Rault

Journal:

Year:

2010

File:

PDF, 31 KB

2010

66

ChemInform Abstract: An Efficient Microwave-Promoted Route to (Z)-Stilbenes from trans-Cinnamic Acids: Synthesis of Combretastatin A-4 and Analogues.

Marc-Antoine Bazin, Marie Jouanne, Hussein El-Kashef, Sylvain Rault

Journal:

Year:

2010

File:

PDF, 39 KB

2010

67

ChemInform Abstract: A Rapid and Versatile Synthesis of Novel Pyrimido[5,4-b]carbazoles.

Anna Caruso, Jean-Charles Lancelot, Hussein El-Kashef, Maria Stefania Sinicropi, Remi Legay, Aurelien Lesnard, Sylvain Rault

Journal:

Year:

2010

File:

PDF, 38 KB

2010

68

ChemInform Abstract: Synthesis of 6-Aryl-Substituted Cholesterol Derivatives from 3β-Acetoxy-6-iodocholest-5-ene and Arylboronic Acids Promoted by Palladium-Catalyzed Cross-Coupling.

Dominique Brossard, Laila El Kihel, Mohamed Khalid, Sylvain Rault

Journal:

Year:

2010

File:

PDF, 45 KB

2010

69

ChemInform Abstract: Hydrogenative Desulfurization of Thienopyrrolizinones: An Easy and Selective Access to (Z)-Phenethylidenepyrrolizinones with in vitro Cytotoxic Activity.

Vittoria Perri, Christophe Rochais, Jana Sopkova-de Oliveira Santos, Remi Legay, Thierry Cresteil, Patrick Dallemagne, Sylvain Rault

Journal:

Year:

2010

File:

PDF, 22 KB

2010

70

ChemInform Abstract: One-Pot Synthesis of Novel Poly-Substituted Phenanthrenes.

Rodrigue Yougnia, Christophe Rochais, Jana Sopkova-de Oliveira Santos, Patrick Dallemagne, Sylvain Rault

Journal:

Year:

2010

File:

PDF, 34 KB

2010

71

ChemInform Abstract: Two-Step Synthesis of Substituted 3-Aminoindazoles from 2-Bromobenzonitriles.

Valerie Lefebvre, Thomas Cailly, Frederic Fabis, Sylvain Rault

Journal:

Year:

2010

File:

PDF, 23 KB

2010

72

ChemInform Abstract: General Method for the Synthesis of Substituted Phenanthridin-6(5H)-ones Using a KOH-Mediated Anionic Ring Closure as the Key Step.

Emmanuelle Dubost, Rosa Magnelli, Thomas Cailly, Remi Legay, Frederic Fabis, Sylvain Rault

Journal:

Year:

2010

File:

PDF, 41 KB

2010

73

ChemInform Abstract: Recent Progress in the Synthesis of Five-Membered Heterocycles Boronic Acids and Esters

Nicolas Primas, Alexandre Bouillon, Sylvain Rault

Journal:

Year:

2011

File:

PDF, 20 KB

2011

74

ChemInform Abstract: Synthesis of New Phenylpyridyl Scaffolds Using the Garlanding Approach.

Anne Sophie Voisin-Chiret, Marilena Muraglia, Gregory Burzicki, Serge Perato, Filomena Corbo, Jana Sopkova-de Oliveira Santos, Carlo Franchini, Sylvain Rault

Journal:

Year:

2011

File:

PDF, 37 KB

2011

75

ChemInform Abstract: Intramolecular Cyclization of β-Aryl-β-amino Acids in the Design of Novel Heterocyclic Systems with Therapeutic Interest: An Unfailing Source of Diversity

Christophe Rochais, Sylvain Rault, Patrick Dallemagne

Journal:

Year:

2011

File:

PDF, 19 KB

2011

76

ChemInform Abstract: First and Mild Synthesis of Fluorene-9-malonic Acid and Some Substituted Derivatives (IV), (VII)/(VIII) via the Intramolecular Hydroarylation of 2-Phenylbenzylidenemalonic Acids.

Elizabeth Chosson, Christophe Rochais, Remi Legay, Jana Sopkova de Oliveira Santos, Sylvain Rault, Patrick Dallemagne

Journal:

Year:

2011

File:

PDF, 39 KB

2011

77

ChemInform Abstract: Efficient Room-Temperature One-Pot Synthesis of 2-Amino-3-alkyl(3-aryl)-quinazolin-4(3H)-ones.

Cedric Lecoutey, Christine Fossey, Sylvain Rault, Frederic Fabis

Journal:

Year:

2011

File:

PDF, 43 KB

2011

78

ChemInform Abstract: Selective ortho-Bromination of Substituted Benzaldoximes Using Pd-Catalyzed C—H Activation: Application to the Synthesis of Substituted 2-Bromobenzaldehydes.

Emmanuelle Dubost, Christine Fossey, Thomas Cailly, Sylvain Rault, Frederic Fabis

Journal:

Year:

2011

File:

PDF, 33 KB

2011

79

ChemInform Abstract: One-Pot Synthesis of New Aza- and Diaza-Aminophenanthrenes.

Christophe Rochais, Rodrigue Yougnia, Thomas Cailly, Jana Sopkova-de Oliveira Santos, Sylvain Rault, Patrick Dallemagne

Journal:

Year:

2011

File:

PDF, 29 KB

2011

80

ChemInform Abstract: Direct Access to 3-Aminoindazoles by Buchwald—Hartwig C—N Coupling Reaction.

Elodie Lohou, Valerie Collot, Silvia Stiebing, Sylvain Rault

Journal:

Year:

2011

File:

PDF, 34 KB

2011

81

ChemInform Abstract: Design and Synthesis of Thienylpyridyl Garlands as Non-Peptidic Alpha Helix Mimetics and Potential Protein—Protein Interactions Disruptors.

Marcella De Giorgi, Anne Sophie Voisin-Chiret, Jana Sopkova-de Oliveira Santos, Filomena Corbo, Carlo Franchini, Sylvain Rault

Journal:

Year:

2011

File:

PDF, 28 KB

2011

82

Efficient Room-Temperature One-Pot Synthesis of 2-Amino-3-alkyl(3-aryl)quinazolin-4(3H)-ones

Cédric Lecoutey, Christine Fossey, Sylvain Rault, Frédéric Fabis

Journal:

European Journal of Organic Chemistry

Year:

2011

Language:

english

File:

PDF, 442 KB

english, 2011

83

Pyrrolo[2,1-c][1,4]benzodiazepines. Synthesis of new cyclic amidines and fused[a]triazolo, tetrazolo and oxadiazolo derivatives

Alain-Claude Gillard, Marie-Paule Foloppe, Sylvain Rault

Journal:

Journal of Heterocyclic Chemistry

Year:

1997

File:

PDF, 582 KB

1997

84

2-Azidopyrrolo[2,1-c][1,4]benzodiazepines. Synthesis of the first cyclic amidine derivatives

Alain-Claude Gillard, Sylvain Rault

Journal:

Journal of Heterocyclic Chemistry

Year:

1997

File:

PDF, 384 KB

1997

85

Pyrrolothieno[1,4]diazepines. Part V. Study of their chemical reactivity and first synthesis of oxazino[4,3-c]pyrrolo[1,2-a]thieno[2,3-f] [1,4]diazepines

Michel Boulouard, Patrick Dallemagne, Sylvain Rault

Journal:

Journal of Heterocyclic Chemistry

Year:

1997

File:

PDF, 524 KB

1997

86

Synthesis of new 6-(4-chlorophenyl)perhydro-1,3-diazepine-2,4-diones via ureidobutyric acids

Jean Guillon, Pascal Sonnet, Patrick Dallemagne, Hugues Miel, Sylvain Rault, Martine Daoust, Michel Boulouard

Journal:

Journal of Heterocyclic Chemistry

Year:

1998

File:

PDF, 371 KB

1998

87

First synthesis of 5,6-dihydro-4H-furo[3,2-f]pyrrolo- [1,2-a][1,4]diazepines

Xiao Feng, Jean-Charles Lancelot, Alain-Claude Gillard, Henriette Landelle, Sylvain Rault

Journal:

Journal of Heterocyclic Chemistry

Year:

1998

File:

PDF, 310 KB

1998

88

Synthesis of novel pyrazolopyrrolopyrazines, potential analogs of sildenafil

Marina Kopp, Jean-Charles Lancelot, Patrick Dallemagne, Sylvain Rault

Journal:

Journal of Heterocyclic Chemistry

Year:

2001

Language:

english

File:

PDF, 62 KB

english, 2001

89

A versatile synthesis of 2-amino-4H-pyrido[1,2-a][1,3,5]triazin-4-ones from 2-aminopyridines

Marina Kopp, Jean-Charles Lancelot, Saïd Dagdag, Hugues Miel, Sylvain Rault

Journal:

Journal of Heterocyclic Chemistry

Year:

2002

Language:

english

File:

PDF, 52 KB

english, 2002

90

Synthesis of novel benzo[h] [1,6]naphthyridines via a rearrangement of hexahydro-5H-pyrrolo [2,1 -c] [1,4]benzodiazepines

Antoine Hinschberger, Frédéric Fabis, Jana Sopkova-De Oliveira Santos, Sylvain Rault

Journal:

Journal of Heterocyclic Chemistry

Year:

2003

Language:

english

File:

PDF, 117 KB

english, 2003

91

Consensus QSAR Related to Global or MOA Models: Application to Acute Toxicity for Fish

Sylvain Lozano, Marie-Pierre Halm-Lemeille, Alban Lepailleur, Sylvain Rault, Ronan Bureau

Journal:

Molecular Informatics

Year:

2010

Language:

english

File:

PDF, 384 KB

english, 2010

92

One-pot cyclization of alkoxy-3-aminoindan-1-ones.

Patrick Dallemagne, Sylvain Rault, Juan Carlos Pilo, Marie Paule Foloppe, Max Robba

Journal:

Tetrahedron Letters

Year:

1991

Language:

english

File:

PDF, 106 KB

english, 1991

93

Original and quick access to 4-phenyl-6H-pyrrolo[1,2-a]thieno [3,2-f][1,4]diazepines

Marie Paule Foloppe, Pascal Sonnet, Sylvain Rault, Max Robba

Journal:

Tetrahedron Letters

Year:

1995

Language:

english

File:

PDF, 95 KB

english, 1995

94

A new rearrangement under microwave heating conditions: synthesis of cyclopenta[b][1,4]benzodiazepines and tetrahydrodibenzo[b,fl[1,4]diazepines.

Sylvain Rault, Alain-Claude Gillard, Marie-Paule Foloppe, Max Robba

Journal:

Tetrahedron Letters

Year:

1995

Language:

english

File:

PDF, 254 KB

english, 1995

95

Etude de la cytotoxicitéin vitro de dérivés du carbazole I. Nitro et amino-9H-carbazoles

Thabet Tabka, Jean-François Héron, Pascal Gauduchon, Jean-Yves Le Talaer, Jean-Charles Lancelot, Sylvain Rault, Max Robba

Journal:

European Journal of Medicinal Chemistry

Year:

1988

File:

PDF, 674 KB

1988

96

Etude de la cytotoxicité in vitro de dérivés du carbazole II. Nitro et amino halogéno-6 diméthyl-1,4 9H-carbazoles

Thabet Tabka, Bertrand Letois, Jean-Charles Lancelot, Pascal Gauduchon, Jean-François Heron, Jean-Yves Le Talaer, Sylvain Rault, Max Robba

Journal:

European Journal of Medicinal Chemistry

Year:

1989

File:

PDF, 662 KB

1989

97

First synthesis of 7α- and 7β-amino-DHEA, dehydroepiandrosterone (DHEA) analogues and preliminary evaluation of their cytotoxicity on Leydig cells and TM4 Sertoli cells

Marc-Antoine Bazin, Carine Travert, Serge Carreau, Sylvain Rault, Laïla El Kihel

Journal:

Bioorganic & Medicinal Chemistry

Year:

2007

Language:

english

File:

PDF, 206 KB

english, 2007

98

New lithocholic and chenodeoxycholic piperazinylcarboxamides with antiproliferative and pro-apoptotic effects on human cancer cell lines

Laïla El Kihel, Monique Clément, Marc-Antoine Bazin, Géraldine Descamps, Mohamed Khalid, Sylvain Rault

Journal:

Bioorganic & Medicinal Chemistry

Year:

2008

Language:

english

File:

PDF, 570 KB

english, 2008

99

Synthesis and in vitro antiplasmodial evaluation of 4-anilino-2-trichloromethylquinazolines

Pierre Verhaeghe, Nadine Azas, Sébastien Hutter, Caroline Castera-Ducros, Michèle Laget, Aurélien Dumètre, Monique Gasquet, Jean-Pierre Reboul, Sylvain Rault, Pascal Rathelot, Patrice Vanelle

Journal:

Bioorganic & Medicinal Chemistry

Year:

2009

Language:

english

File:

PDF, 325 KB

english, 2009

100

Synthesis, reactivity and biological evaluation of novel halogenated tripentones

Vittoria Perri, Christophe Rochais, Thierry Cresteil, Patrick Dallemagne, Sylvain Rault

Journal:

Bioorganic & Medicinal Chemistry

Year:

2009

Language:

english

File:

PDF, 557 KB

english, 2009