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51

Protease Inhibitors of the Sulfonamide Type: Anticancer, Antiinflammatory, and Antiviral Agents

Claudiu T. Supuran, Angela Casini, Andrea Scozzafava

Journal:

Year:

2003

File:

PDF, 67 KB

2003

52

Carbonic Anhydrase Inhibitors: The First Selective, Membrane-Impermeant Inhibitors Targeting the Tumor-Associated Isozyme IX.

Silvia Pastorekova, Angela Casini, Andrea Scozzafava, Daniela Vullo, Jaromir Pastorek, Claudiu T. Supuran

Journal:

Year:

2004

File:

PDF, 86 KB

2004

53

Carbonic Anhydrase Inhibitors: Inhibition of the Tumor-Associated Isozyme IX with Fluorine-Containing Sulfonamides. The First Subnanomolar CA IX Inhibitor Discovered.

Daniela Vullo, Andrea Scozzafava, Silvia Pastorekova, Jaromir Pastorek, Claudiu T. Supuran

Journal:

Year:

2004

File:

PDF, 83 KB

2004

54

Carbonic Anhydrase Inhibitors. Novel Sulfanilamide/Acetazolamide Derivatives Obtained by the Tail Approach and Their Interaction with the Cytosolic Isozymes I and II, and the Tumor-Associated Isozyme IX.

Hasan Turkmen, Mustafa Durgun, Serpil Yilmaztekin, Mahmut Emul, Alessio Innocenti, Daniela Vullo, Andrea Scozzafava, Claudiu T. Supuran

Journal:

Year:

2005

File:

PDF, 14 KB

2005

55

Carbonic Anhydrase Inhibitors: Synthesis and Inhibition of Cytosolic/Tumor-Associated Carbonic Anhydrase Isozymes I, II, and IX with Sulfonamides Incorporating Thioureido-Sulfanilyl Scaffolds.

Luca Puccetti, Giuseppe Fasolis, Alessendro Cecchi, Jean-Yves Winum, Alessandro Gamberi, Jean-Louis Montero, Andrea Scozzafava, Claudiu T. Supuran

Journal:

Year:

2005

File:

PDF, 23 KB

2005

56

Carbonic Anhydrase Inhibitors: Synthesis and Inhibition of Cytosolic/Tumor-Associated Carbonic Anhydrase Isozymes I, II, IX, and XII with N-Hydroxysulfamides — A New Zinc-Binding Function in the Design of Inhibitors.

Jean-Yves Winum, Alessio Innocenti, Jihane Nasr, Jean-Louis Montero, Andrea Scozzafava, Daniela Vullo, Claudiu T. Supuran

Journal:

Year:

2005

File:

PDF, 19 KB

2005

57

Carbonic Anhydrase Inhibitors: Design of Thioureido Sulfonamides with Potent Isozyme II and XII Inhibitory Properties and Intraocular Pressure Lowering Activity in a Rabbit Model of Glaucoma.

Francesco Mincione, Michele Starnotti, Emanuela Masini, Lucia Bacciottini, Chiara Scrivanti, Angela Casini, Daniela Vullo, Andrea Scozzafava, Claudiu T. Supuran

Journal:

Year:

2005

File:

PDF, 13 KB

2005

58

ChemInform Abstract: Synthesis of Rhodamine B-Benzenesulfonamide Conjugates and Their Inhibitory Activity Against Human α- and Bacterial/Fungal β-Carbonic Anhydrases.

Marouan Rami, Alessio Innocenti, Jean-Louis Montero, Andrea Scozzafava, Jean-Yves Winum, Claudiu T. Supuran

Journal:

Year:

2012

Language:

english

File:

PDF, 30 KB

english, 2012

59

ChemInform Abstract: An Inhibitor-Like Binding Mode of a Carbonic Anhydrase Activator within the Active Site of Isoform II.

Khyati Dave, Marc A. Ilies, Andrea Scozzafava, Claudia Temperini, Daniela Vullo, Claudiu T. Supuran

Journal:

Year:

2012

Language:

english

File:

PDF, 12 KB

english, 2012

60

Carbonic Anhydrase Inhibitors: Binding of Indanesulfonamides to the Human Isoform II

Katia D'Ambrosio, Bernard Masereel, Anne Thiry, Andrea Scozzafava, Claudiu T. Supuran, Giuseppina De Simone

Journal:

Year:

2008

Language:

english

File:

PDF, 378 KB

english, 2008

61

Carbonic Anhydrase Inhibitors: Design of Membrane-Impermeant Copper(II) Complexes of DTPA-, DOTA-, and TETA-Tailed Sulfonamides Targeting the Tumor-Associated Transmembrane Isoform IX

Marouan Rami, Alessandro Cecchi, Jean-Louis Montero, Alessio Innocenti, Daniela Vullo, Andrea Scozzafava, Jean-Yves Winum, Claudiu T. Supuran

Journal:

Year:

2008

Language:

english

File:

PDF, 263 KB

english, 2008

62

Functionalized Derivatives of Benzocrown Ethers, II. Supramolecular Complexes of L-Amino Acids as Efficient Activators of the Zinc Enzyme Carbonic Anhydrase

Mihai Barboiu, Claudiu T. Supuran, Andrea Scozzafava, Fabrizio Briganti, Constantin Luca, Georgeta Popescu, Louis Cot, Nadine Hovnanian

Journal:

European Journal of Organic Chemistry

Year:

1997

Language:

english

File:

PDF, 720 KB

english, 1997

63

Cyclodextrin complexes of sulfonamide carbonic anhydrase inhibitors as long-lasting topically acting antiglaucoma agents

Francesca Maestrelli, Paola Mura, Angela Casini, Francesco Mincione, Andrea Scozzafava, Claudiu T. Supuran

Journal:

Journal of Pharmaceutical Sciences

Year:

2002

Language:

english

File:

PDF, 119 KB

english, 2002

64

Bacterial protease inhibitors

Claudiu T. Supuran, Andrea Scozzafava, Brian W. Clare

Journal:

Medicinal Research Reviews

Year:

2002

Language:

english

File:

PDF, 361 KB

english, 2002

65

Carbonic anhydrase inhibitors

Claudiu T. Supuran, Andrea Scozzafava, Angela Casini

Journal:

Medicinal Research Reviews

Year:

2003

Language:

english

File:

PDF, 545 KB

english, 2003

66

Protease inhibitors of the sulfonamide type: Anticancer, antiinflammatory, and antiviral agents

Claudiu T. Supuran, Angela Casini, Andrea Scozzafava

Journal:

Medicinal Research Reviews

Year:

2003

Language:

english

File:

PDF, 303 KB

english, 2003

67

Sulfamates and their therapeutic potential

Jean-Yves Winum, Andrea Scozzafava, Jean-Louis Montero, Claudiu T. Supuran

Journal:

Medicinal Research Reviews

Year:

2005

Language:

english

File:

PDF, 627 KB

english, 2005

68

Therapeutic potential of sulfamides as enzyme inhibitors

Jean-Yves Winum, Andrea Scozzafava, Jean-Louis Montero, Claudiu T. Supuran

Journal:

Medicinal Research Reviews

Year:

2006

Language:

english

File:

PDF, 325 KB

english, 2006

69

Carbonic anhydrase IX: A new druggable target for the design of antitumor agents

Jean-Yves Winum, Marouan Rami, Andrea Scozzafava, Jean-Louis Montero, Claudiu Supuran

Journal:

Medicinal Research Reviews

Year:

2008

Language:

english

File:

PDF, 199 KB

english, 2008

70

Copper-cobalt superoxide dismutase: A re-examination of the 1H NMR spectrum through a novel selectively deuteriated derivative

Ivano Bertini, Mario Piccioli, Andrea Scozzafava, Maria Silvia Viezzoli

Journal:

Magnetic Resonance in Chemistry

Year:

1993

Language:

english

File:

PDF, 572 KB

english, 1993

71

Polymetallic macromolecules are potential contrast agents of improved efficiency

Frederich Cavagna, Claudio Luchinat, Professor Andrea Scozzafava, Zhicheng Xia

Journal:

Magnetic Resonance in Medicine

Year:

1994

Language:

english

File:

PDF, 285 KB

english, 1994

72

Inhibitor interactions with the active site of catechol 2,3 dioxygenase from pseudomonas putida MT2

Fabrizio Briganti, Andrea Scozzafava

Journal:

Journal of Inorganic Biochemistry

Year:

1993

Language:

english

File:

PDF, 72 KB

english, 1993

73

EXAFS studies on the catechol 2,3 dioxygenase from Pseudomonas putida MT2

Fabrizio Briganti, Stefano Mangani, Hans Nolting, Andrea Scozzafava

Journal:

Journal of Inorganic Biochemistry

Year:

1993

Language:

english

File:

PDF, 68 KB

english, 1993

74

Preliminary characterization of the terminal components of some bacterial hydroxylating dioxygenases

Fabrizio Briganti, Riccardo Macinai, Andrea Scozzafava

Journal:

Journal of Inorganic Biochemistry

Year:

1995

Language:

english

File:

PDF, 53 KB

english, 1995

75

Combined action of a bacterial monooxygenase and a fungal laccase for the biodegradation of mono- and poly-aromatic hydrocarbons

Antonella Gullotto, Sergio Branciamore, Ilaria Duchi, Maria Francisca Pareja Caño, Demetrio Randazzo, Silvia Tilli, Paola Giardina, Giovanni Sannia, Andrea Scozzafava, Fabrizio Briganti

Journal:

Bioresource Technology

Year:

2008

Language:

english

File:

PDF, 258 KB

english, 2008

76

Carbonic anhydrase inhibitors. Inhibition of Plasmodium falciparum carbonic anhydrase with aromatic sulfonamides: towards antimalarials with a novel mechanism of action?

Jerapan Krungkrai, Andrea Scozzafava, Sutarnthip Reungprapavut, Sudaratana R. Krungkrai, Roonglawan Rattanajak, Sumalee Kamchonwongpaisan, Claudiu T. Supuran

Journal:

Bioorganic & Medicinal Chemistry

Year:

2005

Language:

english

File:

PDF, 296 KB

english, 2005

77

Carbonic anhydrase inhibitors: Inhibition of the human transmembrane isozyme XIV with a library of aromatic/heterocyclic sulfonamides

Özen Özensoy, Isao Nishimori, Daniela Vullo, Luca Puccetti, Andrea Scozzafava, Claudiu T. Supuran

Journal:

Bioorganic & Medicinal Chemistry

Year:

2005

Language:

english

File:

PDF, 149 KB

english, 2005

78

Carbonic anhydrase inhibitors: Transepithelial transport of thioureido sulfonamide inhibitors of the cancer-associated isozyme IX is dependent on efflux transporters

Daniela Vullo, Bente Steffansen, Birger Brodin, Claudiu T. Supuran, Andrea Scozzafava, Carsten Uhd Nielsen

Journal:

Bioorganic & Medicinal Chemistry

Year:

2006

Language:

english

File:

PDF, 205 KB

english, 2006

79

Sulfonamides incorporating 1,3,5-triazine moieties selectively and potently inhibit carbonic anhydrase transmembrane isoforms IX, XII and XIV over cytosolic isoforms I and II: Solution and X-ray crystallographic studies

Fabrizio Carta, Vladimir Garaj, Alfonso Maresca, Jason Wagner, Balendu Sankara Avvaru, Arthur H. Robbins, Andrea Scozzafava, Robert McKenna, Claudiu T. Supuran

Journal:

Bioorganic & Medicinal Chemistry

Year:

2011

Language:

english

File:

PDF, 2.01 MB

english, 2011

80

Carbonic anhydrase inhibitors: synthesis and inhibition of cytosolic/tumor-associated carbonic anhydrase isozymes I, II, and IX with sulfonamides incorporating 1,2,4-triazine moieties

Vladimir Garaj, Luca Puccetti, Giuseppe Fasolis, Jean-Yves Winum, Jean-Louis Montero, Andrea Scozzafava, Daniela Vullo, Alessio Innocenti, Claudiu T. Supuran

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2004

Language:

english

File:

PDF, 291 KB

english, 2004

81

Carbonic anhydrase activators: The first X-ray crystallographic study of an adduct of isoform I

Claudia Temperini, Andrea Scozzafava, Claudiu T. Supuran

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2006

Language:

english

File:

PDF, 392 KB

english, 2006

82

Phosph(on)ate as a zinc-binding group in metalloenzyme inhibitors: X-ray crystal structure of the antiviral drug foscarnet complexed to human carbonic anhydrase I

Claudia Temperini, Alessio Innocenti, Annalisa Guerri, Andrea Scozzafava, Stefano Rusconi, Claudiu T. Supuran

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2007

Language:

english

File:

PDF, 288 KB

english, 2007

83

Carbonic anhydrase inhibitors: Inhibition of human, bacterial, and archaeal isozymes with benzene-1,3-disulfonamides—Solution and crystallographic studies

Vincenzo Alterio, Giuseppina De Simone, Simona Maria Monti, Andrea Scozzafava, Claudiu T. Supuran

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2007

Language:

english

File:

PDF, 756 KB

english, 2007

84

Carbonic anhydrase inhibitors: Selective inhibition of the extracellular, tumor-associated isoforms IX and XII over isozymes I and II with glycosyl-thioureido-sulfonamides

Fatma-Zohra Smaine, Jean-Yves Winum, Jean-Louis Montero, Zine Regainia, Daniela Vullo, Andrea Scozzafava, Claudiu T. Supuran

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2007

Language:

english

File:

PDF, 153 KB

english, 2007

85

Carbonic anhydrase inhibitors: Copper(II) complexes of polyamino-polycarboxylamido aromatic/heterocyclic sulfonamides are very potent inhibitors of the tumor-associated isoforms IX and XII

Marouan Rami, Jean-Yves Winum, Alessio Innocenti, Jean-Louis Montero, Andrea Scozzafava, Claudiu T. Supuran

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2008

Language:

english

File:

PDF, 150 KB

english, 2008

86

Carbonic anhydrase inhibitors: The X-ray crystal structure of ethoxzolamide complexed to human isoform II reveals the importance of thr200 and gln92 for obtaining tight-binding inhibitors

Anna Di Fiore, Carlo Pedone, Jochen Antel, Harald Waldeck, Andreas Witte, Michael Wurl, Andrea Scozzafava, Claudiu T. Supuran, Giuseppina De Simone

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2008

Language:

english

File:

PDF, 648 KB

english, 2008

87

Investigations of the esterase, phosphatase, and sulfatase activities of the cytosolic mammalian carbonic anhydrase isoforms I, II, and XIII with 4-nitrophenyl esters as substrates

Alessio Innocenti, Andrea Scozzafava, Seppo Parkkila, Luca Puccetti, Giuseppina De Simone, Claudiu T. Supuran

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2008

Language:

english

File:

PDF, 142 KB

english, 2008

88

Carbonic anhydrase inhibitors: Inhibition of the new membrane-associated isoform XV with phenols

Alessio Innocenti, Mika Hilvo, Andrea Scozzafava, Seppo Parkkila, Claudiu T. Supuran

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2008

Language:

english

File:

PDF, 193 KB

english, 2008

89

Carbonic anhydrase inhibitors: Design of spin-labeled sulfonamides incorporating TEMPO moieties as probes for cytosolic or transmembrane isozymes

Alessandro Cecchi, Laura Ciani, Jean-Yves Winum, Jean-Louis Montero, Andrea Scozzafava, Sandra Ristori, Claudiu T. Supuran

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2008

Language:

english

File:

PDF, 236 KB

english, 2008

90

Carbonic anhydrase inhibitors: Inhibition studies of a coral secretory isoform with inorganic anions

Anthony Bertucci, Alessio Innocenti, Didier Zoccola, Andrea Scozzafava, Denis Allemand, Sylvie Tambutté, Claudiu T. Supuran

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2009

Language:

english

File:

PDF, 324 KB

english, 2009

91

Carbonic anhydrase inhibitors. Synthesis of 2,4,6-trimethylpyridinium derivatives of 2-(hydrazinocarbonyl)-3-aryl-1H-indole-5-sulfonamides acting as potent inhibitors of the tumor-associated isoform IX and XII

Özlen Güzel, Alfonso Maresca, Andrea Scozzafava, Aydın Salman, Alexandru T. Balaban, Claudiu T. Supuran

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2009

Language:

english

File:

PDF, 221 KB

english, 2009

92

Carbonic anhydrase activators. Activation of the membrane-associated isoform XV with amino acids and amines

Alessio Innocenti, Mika Hilvo, Seppo Parkkila, Andrea Scozzafava, Claudiu T. Supuran

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2009

Language:

english

File:

PDF, 225 KB

english, 2009

93

Inhibition studies of a β-carbonic anhydrase from Brucella suis with a series of water soluble glycosyl sulfanilamides

Daniela Vullo, Isao Nishimori, Andrea Scozzafava, Stephan Köhler, Jean-Yves Winum, Claudiu T. Supuran

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2010

Language:

english

File:

PDF, 574 KB

english, 2010

94

Carbonic anhydrase inhibitors. The β-carbonic anhydrases from the fungal pathogens Cryptococcus neoformans and Candida albicans are strongly inhibited by substituted-phenyl-1H-indole-5-sulfonamides

Özlen Güzel, Alfonso Maresca, Rebecca A. Hall, Andrea Scozzafava, Antonio Mastrolorenzo, Fritz A. Mühlschlegel, Claudiu T. Supuran

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2010

Language:

english

File:

PDF, 201 KB

english, 2010

95

Crystal structure of the blue multicopper oxidase from the white-rot fungus Trametes trogii complexed with p-toluate

Irene Matera, Antonella Gullotto, Silvia Tilli, Marta Ferraroni, Andrea Scozzafava, Fabrizio Briganti

Journal:

Inorganica Chimica Acta

Year:

2008

Language:

english

File:

PDF, 1.44 MB

english, 2008

96

Role of surfactants in optimizing fluorene assimilation and intermediate formation by Rhodococcus rhodochrous VKM B-2469

Marina P. Kolomytseva, Dimetrio Randazzo, Boris P. Baskunov, Andrea Scozzafava, Fabrizio Briganti, Ludmila A. Golovleva

Journal:

Bioresource Technology

Year:

2009

Language:

english

File:

PDF, 364 KB

english, 2009

97

Carbonic anhydrase and matrix metalloproteinase inhibitors. Inhibition of human tumor-associated isozymes IX and cytosolic isozyme I and II with sulfonylated hydroxamates

Elisa Nuti, Elisabetta Orlandini, Susanna Nencetti, Armando Rossello, Alessio Innocenti, Andrea Scozzafava, Claudiu T. Supuran

Journal:

Bioorganic & Medicinal Chemistry

Year:

2007

Language:

english

File:

PDF, 476 KB

english, 2007

98

Carbonic anhydrase activators: The first activation study of the human secretory isoform VI with amino acids and amines

Isao Nishimori, Saburo Onishi, Daniela Vullo, Alessio Innocenti, Andrea Scozzafava, Claudiu T. Supuran

Journal:

Bioorganic & Medicinal Chemistry

Year:

2007

Language:

english

File:

PDF, 248 KB

english, 2007

99

Molecular modeling study for the binding of zonisamide and topiramate to the human mitochondrial carbonic anhydrase isoform VA

Rosa Maria Vitale, Carlo Pedone, Pietro Amodeo, Jochen Antel, Michael Wurl, Andrea Scozzafava, Claudiu T. Supuran, Giuseppina De Simone

Journal:

Bioorganic & Medicinal Chemistry

Year:

2007

Language:

english

File:

PDF, 676 KB

english, 2007

100

Carbonic anhydrase inhibitors: The inhibition profiles of the human mitochondrial isoforms VA and VB with anions are very different

Isao Nishimori, Alessio Innocenti, Daniela Vullo, Andrea Scozzafava, Claudiu T. Supuran

Journal:

Bioorganic & Medicinal Chemistry

Year:

2007

Language:

english

File:

PDF, 338 KB

english, 2007