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1

Blockade of NMDA receptors 2A subunit in the dorsal striatum impairs the learning of a complex motor skill.

Lemay-Clermont, Julie, Robitaille, Christine, Auberson, Yves P., Bureau, Geneviève, Cyr, Michel

Journal:

Behavioral Neuroscience

Year:

2011

Language:

english

File:

PDF, 7.85 MB

english, 2011

2

ABP688, a novel selective and high affinity ligand for the labeling of mGlu5 receptors: Identification, in vitro pharmacology, pharmacokinetic and biodistribution studies

Samuel Hintermann, Ivo Vranesic, Hans Allgeier, Armin Brülisauer, Daniel Hoyer, Michel Lemaire, Thomas Moenius, Stephan Urwyler, Steven Whitebread, Fabrizio Gasparini, Yves P. Auberson

Journal:

Bioorganic & Medicinal Chemistry

Year:

2007

Language:

english

File:

PDF, 481 KB

english, 2007

3

Substituent effects on the regioselectivity of one-carbon ring expansions of 7-oxabicyclo[2.2.1]heptan-2-one derivatives with diazomethane

Yves Auberson, R.Mampuya Bimwala, Pierre Vogel

Journal:

Tetrahedron Letters

Year:

1991

Language:

english

File:

PDF, 403 KB

english, 1991

4

From Ergolines to Indoles: Improved Inhibitors of the Human H3 Receptor for the Treatment of Narcolepsy

Auberson, Yves P., Troxler, Thomas, Zhang, Xuechun, Yang, Charles R., Feuerbach, Dominik, Liu, Yu-Chih, Lagu, Bharat, Perrone, Mark, Lei, Lijun, Shen, Xiaoxia, Zhang, Dushan, Wang, Chunxiu, Wang, Tie-

Journal:

Year:

2015

Language:

english

File:

PDF, 553 KB

english, 2015

5

Prolongation of levodopa responses by glycineB antagonists in parkinsonian primates

Stella M. Papa, Yves P. Auberson, J. Timothy Greenamyre

Journal:

Annals of Neurology

Year:

2004

Language:

english

File:

PDF, 163 KB

english, 2004

6

Totalsynthese von Allonojirimycin (5-Amino-5-desoxy-D-allopyranose)

Yves Auberson, Prof. Pierre Vogel

Journal:

Angewandte Chemie

Year:

1989

File:

PDF, 261 KB

1989

7

Total Synthesis of Allonojirimycin (5-Amino-5-deoxy-D-allopyranose)

Yves Auberson, Prof. Pierre Vogel

Journal:

Angewandte Chemie International Edition

Year:

1989

Language:

english

File:

PDF, 264 KB

english, 1989

8

ChemInform Abstract: N-Phosphonoalkyl-5-aminomethylquinoxaline-2,3-diones: In vivo Active AMPA and NMDA (Glycine) Antagonists.

Yves P. Auberson, Pierre Acklin, Serge Bischoff, Robert Moretti, Silvio Ofner, Markus Schmutz, Siem J. Veenstra

Journal:

Year:

1999

File:

PDF, 33 KB

1999

9

ChemInform Abstract: 5-Phosphonomethylquinoxalinediones as Competitive NMDA Receptor Antagonists with a Preference for the Human 1A/2A, Rather than 1A/2B Receptor Composition.

Yves P. Auberson, Hans Allgeier, Serge Bischoff, Kurt Lingenhoehl, Robert Moretti, Markus Schmutz

Journal:

Year:

2002

File:

PDF, 27 KB

2002

10

BZM055, an Iodinated Radiotracer Candidate for PET and SPECT Imaging of Myelin and FTY720 Brain Distribution

Dr. Emmanuelle Briard, Dr. David Orain, Dr. Christian Beerli, Dr. Andreas Billich, Dr. Markus Streiff, Dr. Marc Bigaud, Dr. Yves P. Auberson

Journal:

Year:

2011

Language:

english

File:

PDF, 452 KB

english, 2011

11

Cover Picture: BZM055, an Iodinated Radiotracer Candidate for PET and SPECT Imaging of Myelin and FTY720 Brain Distribution (ChemMedChem 4/2011)

Dr. Emmanuelle Briard, Dr. David Orain, Dr. Christian Beerli, Dr. Andreas Billich, Dr. Markus Streiff, Dr. Marc Bigaud, Dr. Yves P. Auberson

Journal:

Year:

2011

Language:

english

File:

PDF, 1.27 MB

english, 2011

12

Total Synthesis of L-Allose, L-Talose, and derivatives.

Yves Auberson, Pierre Vogel

Journal:

Helvetica Chimica Acta

Year:

1989

Language:

english

File:

PDF, 637 KB

english, 1989

13

Quinazolinedione sulfonamides: A novel class of competitive AMPA receptor antagonists with oral activity

Manuel Koller, Kurt Lingenhoehl, Markus Schmutz, Ivan-Toma Vranesic, Joerg Kallen, Yves P. Auberson, David A. Carcache, Henri Mattes, Silvio Ofner, David Orain, Stephan Urwyler

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2011

Language:

english

File:

PDF, 546 KB

english, 2011

14

Diastereoselectivity in the alkylation of 4-fluoroproline methyl esters

Rosanna Filosa, Claude Holder, Yves P. Auberson

Journal:

Tetrahedron Letters

Year:

2006

Language:

english

File:

PDF, 227 KB

english, 2006

15

Total asymmetric synthesis of deoxypolyoxin C

Yves Auberson, Pierre Vogel

Journal:

Year:

1990

Language:

english

File:

PDF, 1012 KB

english, 1990

16

5-Phosphonomethylquinoxalinediones as competitive NMDA receptor antagonists with a preference for the human 1A/2A, rather than 1A/2B receptor composition

Yves P Auberson, Hans Allgeier, Serge Bischoff, Kurt Lingenhoehl, Robert Moretti, Markus Schmutz

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 135 KB

english, 2002

17

5-aminomethylquinoxaline-2,3-diones. Part II: N-aryl derivatives as novel NMDA/glycine and AMPA antagonists

Yves P Auberson, Pierre Acklin, Hans Allgeier, Michel Biollaz, Serge Bischoff, Silvio Ofner, Siem J Veenstra

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1998

Language:

english

File:

PDF, 214 KB

english, 1998

18

5-aminomethylquinoxaline-2,3-diones. Part I: A novel class of AMPA receptor antagonists

Yves P Auberson, Serge Bischoff, Robert Moretti, Markus Schmutz, Siem J Veenstra

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1998

Language:

english

File:

PDF, 251 KB

english, 1998

19

5-aminomethylquinoxaline-2,3-diones, Part III: Arylamide derivatives as highly potent and selective glycine-site NMDA receptor antagonists

Pierre Acklin, Hans Allgeier, Yves P. Auberson, Serge Bischoff, Silvio Ofner, Dirk Sauer, Markus Schmutz

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1998

Language:

english

File:

PDF, 332 KB

english, 1998

20

N-Phosphonoalkyl-5-aminomethylquinoxaline-2,3-diones: In vivo active AMPA and NMDA(glycine) antagonists

Yves P. Auberson, Pierre Acklin, Serge Bischoff, Robert Moretti, Silvio Ofner, Markus Schmutz, Siem J. Veenstra

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1999

Language:

english

File:

PDF, 340 KB

english, 1999

21

Synthesis, radiolabelling and biological characterization of (d)-7-iodo-N-(1-phosphonoethyl)-5-aminomethylquinoxaline-2,3-dione, a glycine-binding site antagonist of NMDA receptors

Simon M. Ametamey, Marco Kokic, Nathalie Carrey-Rémy, Peter Bläuenstein, Martine Willmann, Serge Bischoff, Markus Schmutz, Pius A. Schubiger, Yves P. Auberson

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2000

Language:

english

File:

PDF, 122 KB

english, 2000

22

Selective subunit antagonists suggest an inhibitory relationship between NR2B and NR2A-subunit containingN-methyl-d-aspartate receptors in hippocampal slices

Andrew P. Mallon, Yves P. Auberson, Trevor W. Stone

Journal:

Experimental Brain Research

Year:

2005

Language:

english

File:

PDF, 279 KB

english, 2005

23

NR2A and NR2B subunit containing NMDA receptors differentially regulate striatal output pathways

Martina Fantin, Matteo Marti, Yves P. Auberson, Michele Morari

Journal:

Journal of Neurochemistry

Year:

2007

Language:

english

File:

PDF, 428 KB

english, 2007

24

Differential effect of NR2A and NR2B subunit selective NMDA receptor antagonists on striato-pallidal neurons: relationship to motor response in the 6-hydroxydopamine model of parkinsonism

Martina Fantin, Yves P. Auberson, Michele Morari

Journal:

Journal of Neurochemistry

Year:

2008

Language:

english

File:

PDF, 471 KB

english, 2008

25

The xenon-mediated antagonism against the NMDA receptor is non-selective for receptors containing either NR2A or NR2B subunits in the mouse amygdala

Rainer Haseneder, Stephan Kratzer, Eberhard Kochs, Daniela Höfelmann, Yves Auberson, Matthias Eder, Gerhard Rammes

Journal:

European Journal of Pharmacology

Year:

2009

Language:

english

File:

PDF, 228 KB

english, 2009

26

Reduced spatial learning in mice treated with NVP-AAM077 through down-regulating neurogenesis

Mei Hu, Yong-Jun Sun, Qi-Gang Zhou, Yves P. Auberson, Ling Chen, Yao Hu, Chun-Xia Luo, Jia-Yi Wu, Dong-Ya Zhu, Li-Xin Li

Journal:

European Journal of Pharmacology

Year:

2009

Language:

english

File:

PDF, 700 KB

english, 2009

27

Traumatic mechanical injury to the hippocampus in vitro causes regional caspase-3 and calpain activation that is influenced by NMDA receptor subunit composition

Michael N. DeRidder, Melissa J. Simon, Robert Siman, Yves P. Auberson, Ramesh Raghupathi, David F. Meaney

Journal:

Neurobiology of Disease

Year:

2006

Language:

english

File:

PDF, 890 KB

english, 2006

28

Endoplasmic reticulum stress occurs downstream of GluN2B subunit of N-methyl-d-aspartate receptor in mature hippocampal cultures treated with amyloid-β oligomers

Rui O. Costa, Pascale N. Lacor, Ildete L. Ferreira, Rosa Resende, Yves P. Auberson, William L. Klein, Catarina R. Oliveira, Ana C. Rego, Cláudia M. F. Pereira

Journal:

Year:

2012

Language:

english

File:

PDF, 7.38 MB

english, 2012

29

Rap2-JNK Removes Synaptic AMPA Receptors during Depotentiation

Yinghua Zhu, Daniel Pak, Yi Qin, Stefanie G. McCormack, Myung J. Kim, Joel P. Baumgart, Vanisree Velamoor, Yves P. Auberson, Pavel Osten, Linda van Aelst, Morgan Sheng, J. Julius Zhu

Journal:

Year:

2005

Language:

english

File:

PDF, 563 KB

english, 2005

30

Rap2-JNK Removes Synaptic AMPA Receptors during Depotentiation

Yinghua Zhu, Daniel Pak, Yi Qin, Stefanie G. McCormack, Myung J. Kim, Joel P. Baumgart, Vanisree Velamoor, Yves P. Auberson, Pavel Osten, Linda van Aelst, Morgan Sheng, J. Julius Zhu

Journal:

Year:

2005

Language:

english

File:

PDF, 45 KB

english, 2005

31

P2-382

Streffer, Johannes R., Treyer, Valerie, Schmidt, Mark E., Blagoev, Milen, Hintermann, Samuel, Auberson, Yves, Nitsch, Roger M., Ametamey, Simon M., Buck, Alfred, Hock, Christoph

Journal:

Alzheimer's & Dementia

Year:

2006

Language:

english

File:

PDF, 55 KB

english, 2006

32

The Role of GluN2A and GluN2B Subunits on the Effects of NMDA Receptor Antagonists in Modeling Schizophrenia and Treating Refractory Depression

Jiménez-Sánchez, Laura, Campa, Leticia, Auberson, Yves P, Adell, Albert

Journal:

Neuropsychopharmacology

Year:

2014

Language:

english

File:

PDF, 953 KB

english, 2014

33

GluN2A and GluN2B NMDA Receptor Subunits Differentially Modulate Striatal Output Pathways and Contribute to Levodopa-Induced Abnormal Involuntary Movements in Dyskinetic Rats

Mabrouk, Omar S., Mela, Flora, Calcagno, Mariangela, Budri, Mirco, Viaro, Riccardo, Dekundy, Andrzej, Parsons, Christopher G., Auberson, Yves P., Morari, Michele

Journal:

ACS Chemical Neuroscience

Year:

2013

Language:

english

File:

PDF, 1.33 MB

english, 2013

34

Cover Picture: Ergoline-Derived Inverse Agonists of the Human H3 Receptor for the Treatment of Narcolepsy (ChemMedChem 8/2014)

Auberson, Yves P., Troxler, Thomas, Zhang, Xuechun, Yang, Charles R., Fendt, Markus, Feuerbach, Dominik, Liu, Yu-Chih, Lagu, Bharat, Lerchner, Andreas, Perrone, Mark, Lei, Lijun, Zhang, Chao, Wang, Ch

Journal:

Year:

2014

Language:

english

File:

PDF, 603 KB

english, 2014

35

Ergoline-Derived Inverse Agonists of the Human H3 Receptor for the Treatment of Narcolepsy

Auberson, Yves P., Troxler, Thomas, Zhang, Xuechun, Yang, Charles R., Fendt, Markus, Feuerbach, Dominik, Liu, Yu-Chih, Lagu, Bharat, Lerchner, Andreas, Perrone, Mark, Lei, Lijun, Zhang, Chao, Wang, Ch

Journal:

Year:

2014

Language:

english

File:

PDF, 509 KB

english, 2014

36

Ligand-Biased and Probe-Dependent Modulation of Chemokine Receptor CXCR3 Signaling by Negative Allosteric Modulators

Bernat, Viachaslau, Brox, Regine, Heinrich, Markus R., Auberson, Yves P., Tschammer, Nuska

Journal:

Year:

2015

Language:

english

File:

PDF, 770 KB

english, 2015

37

Preclinical evaluation and test–retest studies of [18F]PSS232, a novel radioligand for targeting metabotropic glutamate receptor 5 (mGlu5)

Sephton, Selena Milicevic, Herde, Adrienne Müller, Mu, Linjing, Keller, Claudia, Rüdisühli, Sonja, Auberson, Yves, Schibli, Roger, Krämer, Stefanie D., Ametamey, Simon M.

Journal:

European Journal of Nuclear Medicine and Molecular Imaging

Year:

2015

Language:

english

File:

PDF, 2.00 MB

english, 2015

38

Blockade of NR2A-Containing NMDA Receptors Induces Tau Phosphorylation in Rat Hippocampal Slices

Allyson, Julie, Dontigny, Eve, Auberson, Yves, Cyr, Michel, Massicotte, Guy

Journal:

Neural Plasticity

Year:

2010

Language:

english

File:

PDF, 1003 KB

english, 2010

39

Reduced Metabotropic Glutamate Receptor 5 Density in Major Depression Determined by [ 11 C]ABP688 PET and Postmortem Study

Deschwanden, Alexandra, Karolewicz, Beata, Feyissa, Anteneh M., Treyer, Valerie, Ametamey, Simon M., Johayem, Anass, Burger, Cyrill, Auberson, Yves P., Sovago, Judit, Stockmeier, Craig A., Buck, Alfre

Journal:

American Journal of Psychiatry

Year:

2011

Language:

english

File:

PDF, 6.71 MB

english, 2011

40

Benzazepinediones by the Reaction of Anthranilides under Vilsmeier-Haack Conditions: A Reinvestigation

Auberson, Yves P., Winkler, Tammo

Journal:

Year:

1994

File:

PDF, 50 KB

1994

41

AMPA Receptor Antagonists: Potential Therapeutic Applications

Mattes, Henri, Lingenhoehl, Kurt, Kalkman, Hans, Auberson, Yves, Renaud, Johanne, Schmutz, Markus, Orain, David

Journal:

Recent Patents on CNS Drug Discovery

Year:

2006

Language:

english

File:

PDF, 84 KB

english, 2006

42

Ligand Specific Efficiency (LSE) Index for PET Tracer Optimization

Auberson, Yves P., Briard, Emmanuelle, Sykes, David, Reilly, John, Healy, Mark

Journal:

Year:

2016

Language:

english

File:

PDF, 763 KB

english, 2016

43

MS565: A SPECT Tracer for Evaluating the Brain Penetration of BAF312 (Siponimod)

Briard, Emmanuelle, Rudolph, Bettina, Desrayaud, Sandrine, Krauser, Joel A., Auberson, Yves P.

Journal:

Year:

2015

Language:

english

File:

PDF, 652 KB

english, 2015

44

Improving Nonspecific Binding and Solubility: Bicycloalkyl Groups and Cubanes as para -Phenyl Bioisosteres

Auberson, Yves P., Brocklehurst, Cara, Furegati, Markus, Fessard, Thomas C., Koch, Guido, Decker, Andrea, La Vecchia, Luigi, Briard, Emmanuelle

Journal:

Year:

2017

Language:

english

File:

PDF, 1.65 MB

english, 2017

45

Cover Picture: Ligand Specific Efficiency (LSE) Index for PET Tracer Optimization (ChemMedChem 13/2016)

Auberson, Yves P., Briard, Emmanuelle, Sykes, David, Reilly, John, Healy, Mark

Journal:

Year:

2016

File:

PDF, 356 KB

2016

46

Joining Forces: The Chemical Biology–Medicinal Chemistry Continuum

Plowright, Alleyn T., Ottmann, Christian, Arkin, Michelle, Auberson, Yves P., Timmerman, Henk, Waldmann, Herbert

Journal:

Cell Chemical Biology

Year:

2017

Language:

english

File:

PDF, 1.13 MB

english, 2017

47

Synthesis and Biological Evaluation of Quinoxaline Derivatives for PET Imaging of the NMDA Receptor

Sephton, Selena Milicevic, Vetterli, Peter T., Pedani, Valentina, Cermak, Stjepko, Chiotellis, Aristeidis, Roscales, Sylvia, Herde, Adrienne Müller, Schibli, Roger, Auberson, Yves P., Ametamey, Simon

Journal:

Helvetica Chimica Acta

Year:

2017

Language:

english

File:

PDF, 449 KB

english, 2017

48

In vivo molecular imaging tools facilitate drug discovery

Auberson, Yves P.

Journal:

Drug Discovery Today: Technologies

Year:

2017

Language:

english

File:

PDF, 189 KB

english, 2017

49

Signaling pathways responsible for the rapid antidepressant-like effects of a GluN2A-preferring NMDA receptor antagonist

Gordillo-Salas, Marta, Pilar-Cuéllar, Fuencisla, Auberson, Yves P., Adell, Albert

Journal:

Translational Psychiatry

Year:

2018

Language:

english

File:

PDF, 1.47 MB

english, 2018

50

PET imaging of T cells: Target identification and feasibility assessment

Auberson, Yves P., Briard, Emmanuelle, Rudolph, Bettina, Kaupmann, Klemen, Smith, Paul, Oberhauser, Berndt

Journal:

Year:

2018

Language:

english

File:

PDF, 1.72 MB

english, 2018