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From Fragment Screening to In Vivo Efficacy: Optimization of a Series of 2-Aminoquinolines as Potent Inhibitors of Beta-Site Amyloid Precursor Protein Cleaving Enzyme 1 (BACE1)
Cheng, Yuan, Judd, Ted C., Bartberger, Michael D., Brown, James, Chen, Kui, Fremeau, Robert T., Hickman, Dean, Hitchcock, Stephen A., Jordan, Brad, Li, VivianVolume:
54
Year:
2011
Language:
english
Pages:
22
DOI:
10.1021/jm200544q
File:
PDF, 3.27 MB
english, 2011