Discovery of 1-(3‘-Aminobenzisoxazol-5‘-yl)-3-trifluoromethyl-N-[2-fluoro-4- [(2‘-dimethylaminomethyl)imidazol-1-yl]phenyl]-1H-pyrazole-5-carboxyamide Hydrochloride (Razaxaban), a Highly Potent, Selective, and Orally Bioavailable Factor Xa Inhibitor
Quan, Mimi L., Lam, Patrick Y. S., Han, Qi, Pinto, Donald J. P., He, Ming Y., Li, Renhua, Ellis, Christopher D., Clark, Charles G., Teleha, Christopher A., Sun, Jung-HuiVolume:
48
Year:
2005
Language:
english
Pages:
16
DOI:
10.1021/jm0497949
File:
PDF, 319 KB
english, 2005