Substrate-Induced Stable Enzyme–Inhibitor Complex Formation Allows Tight Binding of Novel 2-Aminopyrimidin-4(3H)-ones to Drug-Resistant HIV-1 Reverse Transcriptase Mutants
Alberta Samuele, Marcella Facchini, Dante Rotili, Antonello Mai, Marino Artico, Mercedes Armand-Ugón, José A. Esté, Giovanni MagaVolume:
3
Year:
2008
Language:
english
Pages:
7
DOI:
10.1002/cmdc.200800051
File:
PDF, 425 KB
english, 2008