A-995662 [(R)-8-(4-methyl-5-(4-(trifluoromethyl)phenyl)oxazol-2-ylamino)-1,2,3,4-tetrahydronaphthalen-2-ol], a novel, selective TRPV1 receptor antagonist, reduces spinal release of glutamate and CGRP in a rat knee joint pain model
Pamela S. Puttfarcken, Ping Han, Shailen K. Joshi, Torben R. Neelands, Donna M. Gauvin, Scott J. Baker, La Geisha R. Lewis, Bruce R. Bianchi, Joseph P. Mikusa, John R. Koenig, Richard J. Perner, MichaVolume:
150
Year:
2010
Language:
english
Pages:
8
DOI:
10.1016/j.pain.2010.05.015
File:
PDF, 526 KB
english, 2010