Identification, Synthesis, and Biological Evaluation of 6-[(6 R )-2-(4-Fluorophenyl)-6-(hydroxymethyl)-4,5,6,7-tetrahydropyrazolo[1,5- a ]pyrimidin-3-yl]-2-(2-methylphenyl)pyridazin-3(2 H )-one (AS1940477), a Potent p38 MAP Kinase Inhibitor
Asano, Toru, Yamazaki, Hitoshi, Kasahara, Chiyoshi, Kubota, Hirokazu, Kontani, Toru, Harayama, Yu, Ohno, Kazuki, Mizuhara, Hidekazu, Yokomoto, Masaharu, Misumi, Keiji, Kinoshita, Tomohiko, Ohta, MitsuVolume:
55
Language:
english
Pages:
14
Journal:
Journal of Medicinal Chemistry
DOI:
10.1021/jm3008008
Date:
September, 2012
File:
PDF, 906 KB
english, 2012