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Benzoylalanine-Derived Ketoamides Carrying Vinylbenzyl Amino Residues: Discovery of Potent Water-Soluble Calpain Inhibitors with Oral Bioavailability
Lubisch, Wilfried, Beckenbach, Edith, Bopp, Sabina, Hofmann, Hans-Peter, Kartal, Arzu, Kästel, Claudia, Lindner, Tanja, Metz-Garrecht, Marion, Reeb, Jutta, Regner, Ferdinand, Vierling, Michael, MöllerVolume:
46
Language:
english
Journal:
Journal of Medicinal Chemistry
DOI:
10.1021/jm0210717
Date:
June, 2003
File:
PDF, 131 KB
english, 2003