Discovery and Optimization of 1,3,4-Trisubstituted-pyrazolone Derivatives as Novel, Potent, and Nonsteroidal Farnesoid X Receptor (FXR) Selective Antagonists
Huang, Huang, Yu, Ying, Gao, Zhenting, Zhang, Yong, Li, Chenjing, Xu, Xing, Jin, Hui, Yan, Wenzhong, Ma, Ruoqun, Zhu, Jin, Shen, Xu, Jiang, Hualiang, Chen, Lili, Li, JianVolume:
55
Language:
english
Journal:
Journal of Medicinal Chemistry
DOI:
10.1021/jm3002718
Date:
August, 2012
File:
PDF, 2.80 MB
english, 2012