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P2-Substituted N -Acylprolylpyrrolidine Inhibitors of Prolyl Oligopeptidase: Biochemical Evaluation, Binding Mode Determination, and Assessment in a Cellular Model of Synucleinopathy
Van der Veken, Pieter, Fülöp, Vilmos, Rea, Dean, Gerard, Melanie, Van Elzen, Roos, Joossens, Jurgen, Cheng, Jonathan D., Baekelandt, Veerle, De Meester, Ingrid, Lambeir, Anne-Marie, Augustyns, KoenVolume:
55
Language:
english
Journal:
Journal of Medicinal Chemistry
DOI:
10.1021/jm301060g
Date:
November, 2012
File:
PDF, 2.37 MB
english, 2012