Studies on Neurokinin Antagonists. 4. Synthesis and Structure-Activity Relationships of Novel Dipeptide Substance P Antagonists: N2-[(4R)-4-Hydroxy-1-[(1-methyl-1H-indol-3-yl)carbonyl]-L-prolyl]-N-methyl-N-(phenylmethyl)-3-(2-naphthyl)-L-alaninamide and Its Related Compounds
Hagiwara, Daijiro, Miyake, Hiroshi, Igari, Norihiro, Karino, Masako, Maeda, Yasue, Fujii, Takashi, Matsuo, MasaakiVolume:
37
Language:
english
Journal:
Journal of Medicinal Chemistry
DOI:
10.1021/jm00039a022
Date:
June, 1994
File:
PDF, 1.42 MB
english, 1994