Acridone-Based Inhibitors of Inosine 5‘-Monophosphate Dehydrogenase: Discovery and SAR Leading to the Identification of N -(2-(6-(4-Ethylpiperazin-1-yl)pyridin-3-yl)propan-2-yl)-2- fluoro-9-oxo-9,10-dihydroacridine-3-carboxamide (BMS-566419)
Watterson, Scott H., Chen, Ping, Zhao, Yufen, Gu, Henry H., Dhar, T. G. Murali, Xiao, Zili, Ballentine, Shelley K., Shen, Zhongqi, Fleener, Catherine A., Rouleau, Katherine A., Obermeier, Mary, Yang,Volume:
50
Language:
english
Journal:
Journal of Medicinal Chemistry
DOI:
10.1021/jm070299x
Date:
July, 2007
File:
PDF, 206 KB
english, 2007