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A series of potent HIV-1 protease inhibitors containing a hydroxyethyl secondary amine transition state isostere: synthesis, enzyme inhibition, and antiviral activity
Tucker, Thomas J., Lumma, William C., Payne, Linda S., Wai, Jenny M., De Solms, S. Jane, Giuliani, Elizabeth A., Darke, Paul L., Heimbach, Jill C., Zugay, Joan A.Volume:
35
Language:
english
Journal:
Journal of Medicinal Chemistry
DOI:
10.1021/jm00092a002
Date:
July, 1992
File:
PDF, 1.60 MB
english, 1992