Asymmetric Synthesis of Conformationally Constrained Fingolimod Analogues—Discovery of an Orally Active Sphingosine 1-Phosphate Receptor Type-1 Agonist and Receptor Type-3 Antagonist
Zhu, Ran, Snyder, Ashley H., Kharel, Yugesh, Schaffter, Lisa, Sun, Qin, Kennedy, Perry C., Lynch, Kevin R., Macdonald, Timothy L.Volume:
50
Language:
english
Journal:
Journal of Medicinal Chemistry
DOI:
10.1021/jm7010172
Date:
December, 2007
File:
PDF, 447 KB
english, 2007