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Biphenylsulfonamide Endothelin Receptor Antagonists. 4. Discovery of N -[[2‘-[[(4,5-Dimethyl-3-isoxazolyl)amino]sulfonyl]-4-(2-oxazolyl)[1,1‘-biphenyl]- 2-yl]methyl]- N ,3,3-trimethylbutanamide (BMS-207940), A Highly Potent and Orally Active ET A Selective Antagonist
Murugesan, Natesan, Gu, Zhengxiang, Spergel, Steven, Young, Marian, Chen, Ping, Mathur, Arvind, Leith, Leslie, Hermsmeier, Mark, Liu, Eddie C.-K., Zhang, Rongan, Bird, Eileen, Waldron, Tom, Marino, AnVolume:
46
Language:
english
Journal:
Journal of Medicinal Chemistry
DOI:
10.1021/jm020289q
Date:
January, 2003
File:
PDF, 241 KB
english, 2003