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Synthesis and structure–activity relationships for 1-(4-(piperidin-1-ylsulfonyl)phenyl)pyrrolidin-2-ones as novel non-carboxylate inhibitors of the aldo-keto reductase enzyme AKR1C3
Heinrich, Daniel M., Flanagan, Jack U., Jamieson, Stephen M.F., Silva, Shevan, Rigoreau, Laurent J.M., Trivier, Elisabeth, Raynham, Tony, Turnbull, Andrew P., Denny, William A.Volume:
62
Language:
english
Journal:
European Journal of Medicinal Chemistry
DOI:
10.1016/j.ejmech.2013.01.047
Date:
April, 2013
File:
PDF, 1.09 MB
english, 2013