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Reversible Competitive α-Ketoheterocycle Inhibitors of Fatty Acid Amide Hydrolase Containing Additional Conformational Constraints in the Acyl Side Chain: Orally Active, Long-Acting Analgesics
Ezzili, Cyrine, Mileni, Mauro, McGlinchey, Nicholas, Long, Jonathan Z., Kinsey, Steven G., Hochstatter, Dustin G., Stevens, Raymond C., Lichtman, Aron H., Cravatt, Benjamin F., Bilsky, Edward J., BogeVolume:
54
Language:
english
Journal:
Journal of Medicinal Chemistry
DOI:
10.1021/jm101597x
Date:
April, 2011
File:
PDF, 4.34 MB
english, 2011