Optimization of (2,3-Dihydro-1-benzofuran-3-yl)acetic Acids: Discovery of a Non-Free Fatty Acid-Like, Highly Bioavailable G Protein-Coupled Receptor 40/Free Fatty Acid Receptor 1 Agonist as a Glucose-Dependent Insulinotropic Agent
Negoro, Nobuyuki, Sasaki, Shinobu, Mikami, Satoshi, Ito, Masahiro, Tsujihata, Yoshiyuki, Ito, Ryo, Suzuki, Masami, Takeuchi, Koji, Suzuki, Nobuhiro, Miyazaki, Junichi, Santou, Takashi, Odani, TomoyukiVolume:
55
Language:
english
Journal:
Journal of Medicinal Chemistry
DOI:
10.1021/jm300170m
Date:
April, 2012
File:
PDF, 1.67 MB
english, 2012