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Examining the Chirality, Conformation and Selective Kinase Inhibition of 3-((3 R ,4 R )-4-methyl-3-(methyl(7H-pyrrolo[2,3- d ]pyrimidin-4-yl)amino)piperidin-1-yl)-3-oxopropanenitrile (CP-690,550)
Jiang, Jian-kang, Ghoreschi, Kamran, Deflorian, Francesca, Chen, Zhi, Perreira, Melissa, Pesu, Marko, Smith, Jeremy, Nguyen, Dac-Trung, Liu, Eric H., Leister, William, Costanzi, Stefano, O’Shea, JohnVolume:
51
Language:
english
Journal:
Journal of Medicinal Chemistry
DOI:
10.1021/jm801142b
Date:
December, 2008
File:
PDF, 900 KB
english, 2008