Optimization of 6,7-Disubstituted-4-(arylamino)quinoline-3-carbonitriles as Orally Active, Irreversible Inhibitors of Human Epidermal Growth Factor Receptor-2 Kinase Activity
Tsou, Hwei-Ru, Overbeek-Klumpers, Elsebe G., Hallett, William A., Reich, Marvin F., Floyd, M. Brawner, Johnson, Bernard D., Michalak, Ronald S., Nilakantan, Ramaswamy, Discafani, Carolyn, Golas, JonatVolume:
48
Language:
english
Journal:
Journal of Medicinal Chemistry
DOI:
10.1021/jm040159c
Date:
February, 2005
File:
PDF, 642 KB
english, 2005