Discovery of an Orally Bioavailable NK1 Receptor Antagonist, (2S,3S)-(2-Methoxy-5-tetrazol-1-ylbenzyl)(2-phenylpiperidin-3-yl)amine (GR203040), with Potent Antiemetic Activity
Ward, Peter, Armour, Duncan R., Bays, David E., Evans, Brian, Giblin, Gerard M. P., Heron, Nicola, Hubbard, Tania, Liang, Kai, Middlemiss, DavidVolume:
38
Language:
english
Journal:
Journal of Medicinal Chemistry
DOI:
10.1021/jm00026a005
Date:
December, 1995
File:
PDF, 964 KB
english, 1995