Discovery of a Potent, Orally Active 11β-Hydroxysteroid Dehydrogenase Type 1 Inhibitor for Clinical Study: Identification of ( S )-2-((1 S ,2 S ,4 R )-Bicyclo[2.2.1]heptan-2-ylamino)-5-isopropyl-5-methylthiazol-4(5 H )-one (AMG 221)
Véniant, Murielle M., Hale, Clarence, Hungate, Randall W., Gahm, Kyung, Emery, Maurice G., Jona, Janan, Joseph, Smriti, Adams, Jeffrey, Hague, Andrew, Moniz, George, Zhang, Jiandong, Bartberger, MichVolume:
53
Language:
english
Journal:
Journal of Medicinal Chemistry
DOI:
10.1021/jm100242d
Date:
June, 2010
File:
PDF, 2.15 MB
english, 2010