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Systematic evaluation of amide bioisosteres leading to the discovery of novel and potent thiazolylimidazolidinone inhibitors of SCD1 for the treatment of metabolic diseases
Sun, Shaoyi, Zhang, Zaihui, Kodumuru, Vishnumurthy, Pokrovskaia, Natalia, Fonarev, Julia, Jia, Qi, Leung, Po-Yee, Tran, Jennifer, Ratkay, Leslie G., McLaren, David G., Radomski, Chris, Chowdhury, SultVolume:
24
Language:
english
Journal:
Bioorganic & Medicinal Chemistry Letters
DOI:
10.1016/j.bmcl.2013.12.036
Date:
January, 2014
File:
PDF, 759 KB
english, 2014