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IV. Discovery of CXCR3 antagonists substituted with heterocycles as amide surrogates: Improved PK, hERG and metabolic profiles
Nair, Anilkumar G., Wong, Michael K.C., Shu, Youheng, Jiang, Yueheng, Jenh, Chung-Her, Kim, Seong Heon, Yang, De-Yi, Zeng, Qingbei, Shao, Yuefei, Zawacki, Lisa Guise, Duo, Jingqi, McGuinness, Brian F.Volume:
24
Language:
english
Journal:
Bioorganic & Medicinal Chemistry Letters
DOI:
10.1016/j.bmcl.2014.01.009
Date:
February, 2014
File:
PDF, 3.62 MB
english, 2014