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Design and synthesis of 5-[(2-chloro-6-fluorophenyl)acetylamino]-3-(4-fluorophenyl)-4-(4-pyrimidinyl)isoxazole (AKP-001), a novel inhibitor of p38 MAP kinase with reduced side effects based on the antedrug concept
Hasumi, Koichi, Sato, Shuichiro, Saito, Takahisa, Kato, Jun-ya, Shirota, Kazuhiko, Sato, Jun, Suzuki, Hiroyuki, Ohta, ShujiVolume:
22
Language:
english
Journal:
Bioorganic & Medicinal Chemistry
DOI:
10.1016/j.bmc.2014.05.045
Date:
August, 2014
File:
PDF, 2.32 MB
english, 2014