Orally Active 7-Substituted (4-Benzylphthalazin-1-yl)-2-methylpiperazin-1-yl]nicotinonitriles as Active-Site Inhibitors of Sphingosine 1-Phosphate Lyase for the Treatment of Multiple Sclerosis
Weiler, Sven, Braendlin, Nadine, Beerli, Christian, Bergsdorf, Christian, Schubart, Anna, Srinivas, Honnappa, Oberhauser, Berndt, Billich, AndreasVolume:
57
Language:
english
Journal:
Journal of Medicinal Chemistry
DOI:
10.1021/jm500338n
Date:
June, 2014
File:
PDF, 3.74 MB
english, 2014