Structure−Activity Relationship of 6-Methylidene Penems Bearing Tricyclic Heterocycles as Broad-Spectrum β-Lactamase Inhibitors: Crystallographic Structures Show Unexpected Binding of 1,4-Thiazepine Intermediates
Venkatesan, Aranapakam M., Gu, Yansong, Santos, Osvaldo Dos, Abe, Takao, Agarwal, Atul, Yang, Youjun, Petersen, Peter J., Weiss, William J., Mansour, Tarek S., Nukaga, Michiyoshi, Hujer, Andrea M., BoVolume:
47
Language:
english
Journal:
Journal of Medicinal Chemistry
DOI:
10.1021/jm049680x
Date:
December, 2004
File:
PDF, 487 KB
english, 2004