Discovery of Selective and Orally Bioavailable Protein Kinase Cθ (PKCθ) Inhibitors from a Fragment Hit
George, Dawn M., Breinlinger, Eric C., Friedman, Michael, Zhang, Yang, Wang, Jianfei, Argiriadi, Maria, Bansal-Pakala, Pratima, Barth, Martine, Duignan, David B., Honore, Prisca, Lang, QingYu, MittelsVolume:
58
Language:
english
Journal:
Journal of Medicinal Chemistry
DOI:
10.1021/jm500669m
Date:
January, 2015
File:
PDF, 3.76 MB
english, 2015