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A Novel Class of Cycloalkano[ b ]pyridines as Potent and Orally Active Opioid Receptor-like 1 Antagonists with Minimal Binding Affinity to the hERG K + Channel
Yoshizumi, Takashi, Takahashi, Hirobumi, Miyazoe, Hiroshi, Sugimoto, Yuichi, Tsujita, Tomohiro, Kato, Tetsuya, Ito, Hirokatsu, Kawamoto, Hiroshi, Hirayama, Mioko, Ichikawa, Daisuke, Azuma-Kanoh, TomokVolume:
51
Language:
english
Journal:
Journal of Medicinal Chemistry
DOI:
10.1021/jm701590h
Date:
July, 2008
File:
PDF, 222 KB
english, 2008