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Thieno[2,3-d]pyrimidine-2-carboxamides bearing a carboxybenzene group at 5-position: Highly potent, selective, and orally available MMP-13 inhibitors interacting with the S1″ binding site
Nara, Hiroshi, Sato, Kenjiro, Naito, Takako, Mototani, Hideyuki, Oki, Hideyuki, Yamamoto, Yoshio, Kuno, Haruhiko, Santou, Takashi, Kanzaki, Naoyuki, Terauchi, Jun, Uchikawa, Osamu, Kori, MasakuniVolume:
22
Language:
english
Journal:
Bioorganic & Medicinal Chemistry
DOI:
10.1016/j.bmc.2014.07.025
Date:
October, 2014
File:
PDF, 2.98 MB
english, 2014