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Bis(heteroaryl)piperazine (BHAP) reverse transcriptase inhibitors: structure-activity relationships of novel substituted indole analogs and the identification of 1-[(5-methanesulfonamido-1H-indol-2-yl)carbonyl]-4-[3-[(1-methylethyl)amino]pyridinyl]piperazinemonomethanesulfonate (U-90152S), a second-generation clinical candidate
Romero, Donna L., Morge, Raymond A., Genin, Michael J., Biles, Carolyn, Busso, Mariano, Resnick, Lionel, Althaus, Irene W., Reusser, Fritz, Thomas, Richard C., Tarpley, William G.Volume:
36
Language:
english
Journal:
Journal of Medicinal Chemistry
DOI:
10.1021/jm00062a027
Date:
May, 1993
File:
PDF, 606 KB
english, 1993