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Identification, Synthesis, and Biological Evaluation of 6-[(6 R )-2-(4-Fluorophenyl)-6-(hydroxymethyl)-4,5,6,7-tetrahydropyrazolo[1,5- a ]pyrimidin-3-yl]-2-(2-methylphenyl)pyridazin-3(2 H )-one (AS1940477), a Potent p38 MAP Kinase Inhibitor
Asano, Toru, Yamazaki, Hitoshi, Kasahara, Chiyoshi, Kubota, Hirokazu, Kontani, Toru, Harayama, Yu, Ohno, Kazuki, Mizuhara, Hidekazu, Yokomoto, Masaharu, Misumi, Keiji, Kinoshita, Tomohiko, Ohta, MitsuVolume:
57
Journal:
Journal of Medicinal Chemistry
DOI:
10.1021/jm501222p
Date:
August, 2014
File:
PDF, 119 KB
2014