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Development of a Multikilogram Synthesis of a Chiral Epoxide Precursor to a CCR1 Antagonist. Use of in Situ Monitoring for Informed Optimisation via Fragile Intermediates
Ainge, Debra, Booker, James E. M., Pedge, Nicholas, Sinclair, Rhona, Sleigh, Chris, Štefinović, Marijan, Vaz, Luis-Manuel, Way, EdwardVolume:
14
Language:
english
Journal:
Organic Process Research & Development
DOI:
10.1021/op900172t
Date:
January, 2010
File:
PDF, 1016 KB
english, 2010