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4-Nitrobenzyloxycarbonyl Derivatives of O 6 -Benzylguanine as Hypoxia-Activated Prodrug Inhibitors of O 6 -Alkylguanine-DNA Alkyltransferase (AGT), Which Produces Resistance to Agents Targeting the O -6 Position of DNA Guanine
Zhu, Rui, Liu, Mao-Chin, Luo, Mei-Zhen, Penketh, Philip G., Baumann, Raymond P., Shyam, Krishnamurthy, Sartorelli, Alan C.Volume:
54
Language:
english
Journal:
Journal of Medicinal Chemistry
DOI:
10.1021/jm201115f
Date:
November, 2011
File:
PDF, 1.11 MB
english, 2011