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Metabolic activation of indole-containing prostaglandin D2 receptor 1 antagonists: Impacts of glutathione trapping and glucuronide conjugation on covalent binding
Jean-François Lévesque, Stephen H. Day, Nathalie Chauret, Carmai Seto, Laird Trimble, Kevin P. Bateman, José M. Silva, Carl Berthelette, Nicolas Lachance, Michael Boyd, Lianhai Li, Claudio F. Sturino,Volume:
17
Year:
2007
Language:
english
Pages:
6
DOI:
10.1016/j.bmcl.2007.03.058
File:
PDF, 213 KB
english, 2007