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Discovery of novel tetrahydroisoquinoline derivatives as orally active N-type calcium channel blockers with high selectivity for hERG potassium channels
Ogiyama, Takashi, Inoue, Makoto, Honda, Shugo, Yamada, Hiroyoshi, Watanabe, Toshihiro, Gotoh, Takayasu, Kiso, Tetsuo, Koakutsu, Akiko, Kakimoto, Shuichiro, Shishikura, Jun-ichiVolume:
22
Language:
english
Journal:
Bioorganic & Medicinal Chemistry
DOI:
10.1016/j.bmc.2014.10.020
Date:
December, 2014
File:
PDF, 1.69 MB
english, 2014