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6-Hydroxybenzothiophene Ketones: Potent Inhibitors of 17β-Hydroxysteroid Dehydrogenase Type 1 (17β-HSD1) Owing to Favorable Molecule Geometry and Conformational Preorganization
Miralinaghi, Parisa, Schmitt, Christian, Hartmann, Rolf W., Frotscher, Martin, Engel, MatthiasVolume:
9
Language:
english
Journal:
ChemMedChem
DOI:
10.1002/cmdc.201402050
Date:
October, 2014
File:
PDF, 789 KB
english, 2014